An Update on Development of Small-Molecule Plasmodial Kinase Inhibitors
Moolman, Chantalle, Sluis, Rencia van der, Beteck, Richard M, Legoabe, Lesetja J
Published in Molecules (Basel, Switzerland) (07.11.2020)
Published in Molecules (Basel, Switzerland) (07.11.2020)
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2-Aroyl quinazolinone: Synthesis and in vitro anti-parasitic activity
Setshedi, Koketso J. J., Beteck, Richard M. M., Jesumoroti, Omobolanle J. J., Ilbeigi, Kayhan, Mabille, Dorien, Caljon, Guy, Van der Kooy, Frank, Legoabe, Lesetja J. J.
Published in Chemical biology & drug design (01.10.2023)
Published in Chemical biology & drug design (01.10.2023)
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Recent progress in the development of anti-malarial quinolones
Beteck, Richard M, Smit, Frans J, Haynes, Richard K, N'Da, David D
Published in Malaria journal (30.08.2014)
Published in Malaria journal (30.08.2014)
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Assessment of the Activity of Decoquinate and Its Quinoline- O -Carbamate Derivatives against Toxoplasma gondii In Vitro and in Pregnant Mice Infected with T. gondii Oocysts
Ramseier, Jessica, Imhof, Dennis, Anghel, Nicoleta, Hänggeli, Kai, Beteck, Richard M, Balmer, Vreni, Ortega-Mora, Luis-Miguel, Sanchez-Sanchez, Roberto, Ferre, Ignacio, Haynes, Richard K, Hemphill, Andrew
Published in Molecules (Basel, Switzerland) (22.10.2021)
Published in Molecules (Basel, Switzerland) (22.10.2021)
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Easy-To-Access Quinolone Derivatives Exhibiting Antibacterial and Anti-Parasitic Activities
Beteck, Richard M, Jordaan, Audrey, Seldon, Ronnett, Laming, Dustin, Hoppe, Heinrich C, Warner, Digby F, Khanye, Setshaba D
Published in Molecules (Basel, Switzerland) (20.02.2021)
Published in Molecules (Basel, Switzerland) (20.02.2021)
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New Quinolone-Based Thiosemicarbazones Showing Activity Against Plasmodium falciparum and Mycobacterium tuberculosis
Beteck, Richard M, Seldon, Ronnett, Jordaan, Audrey, Warner, Digby F, Hoppe, Heinrich C, Laming, Dustin, Khanye, Setshaba D
Published in Molecules (Basel, Switzerland) (04.05.2019)
Published in Molecules (Basel, Switzerland) (04.05.2019)
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Cinnamoyl-Oxaborole Amides: Synthesis and Their in Vitro Biological Activity
Gumbo, Maureen, Beteck, Richard M, Mandizvo, Tawanda, Seldon, Ronnett, Warner, Digby F, Hoppe, Heinrich C, Isaacs, Michelle, Laming, Dustin, Tam, Christina C, Cheng, Luisa W, Liu, Nicole, Land, Kirkwood M, Khanye, Setshaba D
Published in Molecules (Basel, Switzerland) (15.08.2018)
Published in Molecules (Basel, Switzerland) (15.08.2018)
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Synthesis and In Vitro Antibacterial Evaluation of Mannich Base Nitrothiazole Derivatives
Dube, Phelelisiwe S, Hart, Dylan, Legoabe, Lesetja J, Jordaan, Audrey, Warner, Digby F, Beteck, Richard M
Published in MolBank (01.03.2024)
Published in MolBank (01.03.2024)
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Journal Article
In Vitro versus in Mice: Efficacy and Safety of Decoquinate and Quinoline- O -Carbamate Derivatives against Experimental Infection with Neospora caninum Tachyzoites
Ramseier, Jessica, Imhof, Dennis, Hänggeli, Kai Pascal Alexander, Anghel, Nicoleta, Boubaker, Ghalia, Beteck, Richard M, Ortega-Mora, Luis-Miguel, Haynes, Richard K, Hemphill, Andrew
Published in Pathogens (Basel) (13.03.2023)
Published in Pathogens (Basel) (13.03.2023)
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Anti-Trypanosomal and Antimalarial Properties of Tetralone Derivatives and Structurally Related Benzocycloalkanones
Beteck, Richard M, Legoabe, Lesetja J, Isaacs, Michelle, Khanye, Setshaba D, Laming, Dustin, Hoppe, Heinrich C
Published in Medicina (Kaunas, Lithuania) (24.05.2019)
Published in Medicina (Kaunas, Lithuania) (24.05.2019)
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Antimalarial application of quinones: A recent update
Patel, Om P.S., Beteck, Richard M., Legoabe, Lesetja J.
Published in European journal of medicinal chemistry (15.01.2021)
Published in European journal of medicinal chemistry (15.01.2021)
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Journal Article
Quinolone: a versatile therapeutic compound class
Dube, Phelelisiwe S., Legoabe, Lesetja J., Beteck, Richard M.
Published in Molecular diversity (01.06.2023)
Published in Molecular diversity (01.06.2023)
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Steroid-triazole conjugates: A brief overview of synthesis and their application as anticancer agents
Agarwal, Devesh S., Sakhuja, Rajeev, Beteck, Richard M., Legoabe, Lesetja J.
Published in Steroids (01.09.2023)
Published in Steroids (01.09.2023)
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Quinolone analogues of benzothiazinone: Synthesis, antitubercular structure-activity relationship and ADME profiling
Dube, Phelelisiwe S., Legoabe, Lesetja J., Jordaan, Audrey, Sigauke, Lester, Warner, Digby F., Beteck, Richard M.
Published in European journal of medicinal chemistry (05.10.2023)
Published in European journal of medicinal chemistry (05.10.2023)
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Hydrazinated geraniol derivatives as potential broad‐spectrum antiprotozoal agents
Jooste, Joelien, Legoabe, Lesetja J., Ilbeigi, Kayhan, Caljon, Guy, Beteck, Richard M.
Published in Archiv der Pharmazie (Weinheim) (01.10.2024)
Published in Archiv der Pharmazie (Weinheim) (01.10.2024)
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Journal Article
Synthesis and in vitro antitrypanosomal evaluation of novel 6-heteroarylidene-substituted quinolone derivatives
Angula, Klaudia T., Legoabe, Lesetja J., Swart, Tarryn, Hoppe, Heinrich C., Beteck, Richard M.
Published in European journal of medicinal chemistry (05.01.2022)
Published in European journal of medicinal chemistry (05.01.2022)
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