TAC‐tics for Leveraging Proximity Biology in Drug Discovery
Nalawansha, Dhanusha A., Mangano, Kyle, Besten, Willem, Potts, Patrick Ryan
Published in Chembiochem : a European journal of chemical biology (16.02.2024)
Published in Chembiochem : a European journal of chemical biology (16.02.2024)
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Journal Article
NEDD8 links cullin-RING ubiquitin ligase function to the p97 pathway
den Besten, Willem, Verma, Rati, Kleiger, Gary, Oania, Robert S, Deshaies, Raymond J
Published in Nature structural & molecular biology (01.05.2012)
Published in Nature structural & molecular biology (01.05.2012)
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Journal Article
Primary Amine Tethered Small Molecules Promote the Degradation of X‑Linked Inhibitor of Apoptosis Protein
Besten, Willem den, Verma, Kshitij, Yamazoe, Sayumi, Blaquiere, Nicole, Phung, Wilson, Izrael-Tomasevic, Anita, Mulvihill, Melinda M, Helgason, Elizabeth, Prakash, Sumit, Goncharov, Tatiana, Vucic, Domagoj, Dueber, Erin, Fairbrother, Wayne J, Wertz, Ingrid, Yu, Kebing, Staben, Steven T
Published in Journal of the American Chemical Society (21.07.2021)
Published in Journal of the American Chemical Society (21.07.2021)
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Journal Article
Conjugation of Indoles to Antibodies through a Novel Self‐Immolating Linker
Dragovich, Peter S., Blake, Robert A., Chen, Chunjiao, Chen, Jinhua, Chuh, Josefa, den Besten, Willem, Fan, Fang, Fourie, Aimee, Hartman, Steven J., He, Changrong, He, Jintang, Ingalla, Ellen Rei, Kozak, Katherine R., Leong, Steven R., Lu, Jiawei, Ma, Yong, Meng, Lingyao, Nannini, Michelle, Oeh, Jason, Ohri, Rachana, Lewis Phillips, Gail, Pillow, Thomas H., Rowntree, Rebecca K., Sampath, Deepak, Vandlen, Richard, Vollmar, Breanna, Wai, John, Wertz, Ingrid E., Xu, Keyang, Xu, Zijin, Zhang, Donglu
Published in Chemistry : a European journal (03.04.2018)
Published in Chemistry : a European journal (03.04.2018)
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Journal Article
Cytokine-dependent imatinib resistance in mouse BCR-ABL+, Arf-null lymphoblastic leukemia
Williams, Richard T, den Besten, Willem, Sherr, Charles J
Published in Genes & development (15.09.2007)
Published in Genes & development (15.09.2007)
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Journal Article
Degradation of the Deubiquitinating Enzyme USP33 Is Mediated by p97 and the Ubiquitin Ligase HERC2
Chan, Nickie C., den Besten, Willem, Sweredoski, Michael J., Hess, Sonja, Deshaies, Raymond J., Chan, David C.
Published in The Journal of biological chemistry (11.07.2014)
Published in The Journal of biological chemistry (11.07.2014)
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Journal Article
Options for a National Framework for Benefit Distribution and Their Relation to Community-Based and National REDD+ Monitoring
Skutsch, Margaret, Turnhout, Esther, Vijge, Marjanneke, Herold, Martin, Wits, Tjeerd, den Besten, Jan, Torres, Arturo
Published in Forests (2014)
Published in Forests (2014)
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Journal Article
Arf-induced turnover of the nucleolar nucleophosmin-associated SUMO-2/3 protease Senp3
Kuo, Mei-Ling, den Besten, Willem, Thomas, Mary C., Sherr, Charles J.
Published in Cell cycle (Georgetown, Tex.) (01.11.2008)
Published in Cell cycle (Georgetown, Tex.) (01.11.2008)
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Journal Article
The evolution of REDD+: An analysis of discursive-institutional dynamics
den Besten, Jan Willem, Arts, Bas, Verkooijen, Patrick
Published in Environmental science & policy (01.01.2014)
Published in Environmental science & policy (01.01.2014)
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Journal Article
Protein Interaction Profiling of the p97 Adaptor UBXD1 Points to a Role for the Complex in Modulating ERGIC-53 Trafficking
Haines, Dale S., Lee, J. Eugene, Beauparlant, Stephen L., Kyle, Dane B., den Besten, Willem, Sweredoski, Michael J., Graham, Robert L.J., Hess, Sonja, Deshaies, Raymond J.
Published in Molecular & cellular proteomics (01.06.2012)
Published in Molecular & cellular proteomics (01.06.2012)
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Journal Article
N-Terminal Polyubiquitination of the ARF Tumor Suppressor, A Natural Lysine-Less Protein
Kuo, Mei-Ling, Besten, Willem den, Sherr, Charles J.
Published in Cell cycle (Georgetown, Tex.) (01.11.2004)
Published in Cell cycle (Georgetown, Tex.) (01.11.2004)
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Journal Article
Catalytic in vivo protein knockdown by small-molecule PROTACs
Bondeson, Daniel P, Mares, Alina, Smith, Ian E D, Ko, Eunhwa, Campos, Sebastien, Miah, Afjal H, Mulholland, Katie E, Routly, Natasha, Buckley, Dennis L, Gustafson, Jeffrey L, Zinn, Nico, Grandi, Paola, Shimamura, Satoko, Bergamini, Giovanna, Faelth-Savitski, Maria, Bantscheff, Marcus, Cox, Carly, Gordon, Deborah A, Willard, Ryan R, Flanagan, John J, Casillas, Linda N, Votta, Bartholomew J, den Besten, Willem, Famm, Kristoffer, Kruidenier, Laurens, Carter, Paul S, Harling, John D, Churcher, Ian, Crews, Craig M
Published in Nature chemical biology (01.08.2015)
Published in Nature chemical biology (01.08.2015)
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Journal Article
Antibody-mediated delivery of chimeric protein degraders which target estrogen receptor alpha (ERα)
Dragovich, Peter S., Adhikari, Pragya, Blake, Robert A., Blaquiere, Nicole, Chen, Jinhua, Cheng, Yun-Xing, den Besten, Willem, Han, Jinping, Hartman, Steven J., He, Jintang, He, Mingtao, Rei Ingalla, Ellen, Kamath, Amrita V., Kleinheinz, Tracy, Lai, Tommy, Leipold, Douglas D., Li, Chun Sing, Liu, Qi, Lu, Jiawei, Lu, Ying, Meng, Fanwei, Meng, Lingyao, Ng, Carl, Peng, Kaishan, Lewis Phillips, Gail, Pillow, Thomas H., Rowntree, Rebecca K., Sadowsky, Jack D., Sampath, Deepak, Staben, Leanna, Staben, Steven T., Wai, John, Wan, Kunpeng, Wang, Xinxin, Wei, BinQing, Wertz, Ingrid E., Xin, Jianfeng, Xu, Keyang, Yao, Hui, Zang, Richard, Zhang, Donglu, Zhou, Hao, Zhao, Yongxin
Published in Bioorganic & medicinal chemistry letters (15.02.2020)
Published in Bioorganic & medicinal chemistry letters (15.02.2020)
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Journal Article
PYCR1 and PYCR2 Interact and Collaborate with RRM2B to Protect Cells from Overt Oxidative Stress
Kuo, Mei-Ling, Lee, Mabel Bin-Er, Tang, Michelle, den Besten, Willem, Hu, Shuya, Sweredoski, Michael J, Hess, Sonja, Chou, Chih-Ming, Changou, Chun A, Su, Mingming, Jia, Wei, Su, Leila, Yen, Yun
Published in Scientific reports (06.01.2016)
Published in Scientific reports (06.01.2016)
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