N‑[6-(4-Butanoyl-5-methyl‑1H‑pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]‑1H‑indole-3-carboxamide (SAR216471), a Novel Intravenous and Oral, Reversible, and Directly Acting P2Y12 Antagonist
Boldron, Christophe, Besse, Angélina, Bordes, Marie-Françoise, Tissandié, Stéphanie, Yvon, Xavier, Gau, Benjamin, Badorc, Alain, Rousseaux, Tristan, Barré, Guillaume, Meneyrol, Jérôme, Zech, Gernot, Nazare, Marc, Fossey, Valérie, Pflieger, Anne-Marie, Bonnet-Lignon, Sandrine, Millet, Laurence, Briot, Christophe, Dol, Frédérique, Hérault, Jean-Pascal, Savi, Pierre, Lassalle, Gilbert, Delesque, Nathalie, Herbert, Jean-Marc, Bono, Françoise
Published in Journal of medicinal chemistry (11.09.2014)
Published in Journal of medicinal chemistry (11.09.2014)
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Journal Article
N -[6-(4-Butanoyl-5-methyl-1 H -pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-1 H -indole-3-carboxamide (SAR216471), a Novel Intravenous and Oral, Reversible, and Directly Acting P2Y12 Antagonist
Boldron, Christophe, Besse, Angélina, Bordes, Marie-Françoise, Tissandié, Stéphanie, Yvon, Xavier, Gau, Benjamin, Badorc, Alain, Rousseaux, Tristan, Barré, Guillaume, Meneyrol, Jérôme, Zech, Gernot, Nazare, Marc, Fossey, Valérie, Pflieger, Anne-Marie, Bonnet-Lignon, Sandrine, Millet, Laurence, Briot, Christophe, Dol, Frédérique, Hérault, Jean-Pascal, Savi, Pierre, Lassalle, Gilbert, Delesque, Nathalie, Herbert, Jean-Marc, Bono, Françoise
Published in Journal of medicinal chemistry (11.09.2014)
Published in Journal of medicinal chemistry (11.09.2014)
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Journal Article
DERIVATIVES OF 1H-INDOLE-3-CARBOXAMIDE AND THEIR USE AS P2Y12 ANTAGONISTS
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Year of Publication 28.09.2016
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1H-Indole-3-Carboxamide Derivatives And Use Thereof As P2Y12 Antagonists
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DERIVATIVES OF 1H-INDOLE-3-CARBOXAMIDE AND THEIR USE AS P2Y12 ANTAGONISTS
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1H-INDOLE-3-CARBOXAMIDE DERIVATIVES, AND USE THEREOF AS P2Y12 ANTAGONIS TS
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derivados de 1 h-indol-3- carboxamida e sua utilização como antagonistas do p2y12
ANGELINA BESSE, CHRISTOPHE BOLDRON, GERNOT ZECH, VALÉRIE FOSSEY, ALAIN BADORC
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Year of Publication 04.07.2017
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Derivados de 1H-indol-3-carboxamida y sus usos como antagonistas de P2Y12
BESSE, Angelina, BOLDRON, Christophe, FOSSEY, Valérie, BADORC, Alain, ZECH, Gernot
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1 H-INDOLE-3-CARBOXAMIDE DERIVATIVES AND USE THEREOF AS P2Y12 ANTAGONISTS
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1H-INDOLE-3-CARBOXAMIDE DERIVATIVES AND USE THEREOF AS P2Y12 ANTAGONISTS
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