Theranostic Perspectives in Prostate Cancer with the Gastrin-Releasing Peptide Receptor Antagonist NeoBOMB1: Preclinical and First Clinical Results
Nock, Berthold A, Kaloudi, Aikaterini, Lymperis, Emmanouil, Giarika, Athina, Kulkarni, Harshad R, Klette, Ingo, Singh, Aviral, Krenning, Eric P, de Jong, Marion, Maina, Theodosia, Baum, Richard P
Published in Journal of Nuclear Medicine (01.01.2017)
Published in Journal of Nuclear Medicine (01.01.2017)
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Journal Article
"To serve and protect": enzyme inhibitors as radiopeptide escorts promote tumor targeting
Nock, Berthold A, Maina, Theodosia, Krenning, Eric P, de Jong, Marion
Published in Journal of Nuclear Medicine (01.01.2014)
Published in Journal of Nuclear Medicine (01.01.2014)
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Journal Article
Peptide Radioligands in Cancer Theranostics: Agonists and Antagonists
Nock, Berthold A, Kanellopoulos, Panagiotis, Joosten, Lieke, Mansi, Rosalba, Maina, Theodosia
Published in Pharmaceuticals (Basel, Switzerland) (30.04.2023)
Published in Pharmaceuticals (Basel, Switzerland) (30.04.2023)
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Journal Article
Radiolabeled Bombesin Analogs
Mansi, Rosalba, Nock, Berthold A., Dalm, Simone U., Busstra, Martijn B., van Weerden, Wytske M., Maina, Theodosia
Published in Cancers (17.11.2021)
Published in Cancers (17.11.2021)
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Journal Article
[68Ga]Ga-DATA5m-LM4, a PET Radiotracer in the Diagnosis of SST2R-Positive Tumors: Preclinical and First Clinical Results
Kanellopoulos, Panagiotis, Nock, Berthold A., Greifenstein, Lukas, Baum, Richard P., Roesch, Frank, Maina, Theodosia
Published in International journal of molecular sciences (23.11.2022)
Published in International journal of molecular sciences (23.11.2022)
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Journal Article
Bis(Disulfide)-Bridged Somatostatin-14 Analogs and Their [ 111 In]In-Radioligands: Synthesis and Preclinical Profile
Tatsi, Aikaterini, Maina, Theodosia, Waser, Beatrice, Krenning, Eric P, de Jong, Marion, Reubi, Jean Claude, Cordopatis, Paul, Nock, Berthold A
Published in International journal of molecular sciences (01.02.2024)
Published in International journal of molecular sciences (01.02.2024)
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Journal Article
[ 99m Tc]Tc-DB1 Mimics with Different-Length PEG Spacers: Preclinical Comparison in GRPR-Positive Models
Kanellopoulos, Panagiotis, Lymperis, Emmanouil, Kaloudi, Aikaterini, de Jong, Marion, Krenning, Eric P, Nock, Berthold A, Maina, Theodosia
Published in Molecules (Basel, Switzerland) (28.07.2020)
Published in Molecules (Basel, Switzerland) (28.07.2020)
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Journal Article
Preclinical and first clinical experience with the gastrin-releasing peptide receptor-antagonist [68Ga]SB3 and PET/CT
Maina, Theodosia, Bergsma, Hendrik, Kulkarni, Harshad R., Mueller, Dirk, Charalambidis, David, Krenning, Eric P., Nock, Berthold A., de Jong, Marion, Baum, Richard P.
Published in European journal of nuclear medicine and molecular imaging (01.05.2016)
Published in European journal of nuclear medicine and molecular imaging (01.05.2016)
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Journal Article
Combination of the amide‐to‐triazole substitution strategy with alternative structural modifications for the metabolic stabilization of tumor‐targeting, radiolabeled peptides
Guarrochena, Xabier, Anderla, Maximilian, Salomon, Philipp, Feiner, Irene V. J., Nock, Berthold A., Maina, Theodosia, Mindt, Thomas L.
Published in Journal of peptide science (11.09.2024)
Published in Journal of peptide science (11.09.2024)
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Journal Article
NeoBOMB1, a GRPR-Antagonist for Breast Cancer Theragnostics: First Results of a Preclinical Study with [ 67 Ga]NeoBOMB1 in T-47D Cells and Tumor-Bearing Mice
Kaloudi, Aikaterini, Lymperis, Emmanouil, Giarika, Athina, Dalm, Simone, Orlandi, Francesca, Barbato, Donato, Tedesco, Mattia, Maina, Theodosia, de Jong, Marion, Nock, Berthold A
Published in Molecules (Basel, Switzerland) (11.11.2017)
Published in Molecules (Basel, Switzerland) (11.11.2017)
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Journal Article
GRPR-Antagonists Carrying DOTAGA-Chelator via Positively Charged Linkers: Perspectives for Prostate Cancer Theranostics
Obeid, Karim, Kanellopoulos, Panagiotis, Abouzayed, Ayman, Mattsson, Adam, Tolmachev, Vladimir, Nock, Berthold A, Maina, Theodosia, Orlova, Anna
Published in Pharmaceutics (01.04.2024)
Published in Pharmaceutics (01.04.2024)
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Journal Article
Structure of alpha-synuclein fibrils derived from human Lewy body dementia tissue
Dhavale, Dhruva D, Barclay, Alexander M, Borcik, Collin G, Basore, Katherine, Berthold, Deborah A, Gordon, Isabelle R, Liu, Jialu, Milchberg, Moses H, O'Shea, Jennifer Y, Rau, Michael J, Smith, Zachary, Sen, Soumyo, Summers, Brock, Smith, John, Warmuth, Owen A, Perrin, Richard J, Perlmutter, Joel S, Chen, Qian, Fitzpatrick, James A J, Schwieters, Charles D, Tajkhorshid, Emad, Rienstra, Chad M, Kotzbauer, Paul T
Published in Nature communications (29.03.2024)
Published in Nature communications (29.03.2024)
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Journal Article
[99mTc]Tc-DB15 in GRPR-Targeted Tumor Imaging with SPECT: From Preclinical Evaluation to the First Clinical Outcomes
Nock, Berthold A., Kaloudi, Aikaterini, Kanellopoulos, Panagiotis, Janota, Barbara, Bromińska, Barbara, Iżycki, Dariusz, Mikołajczak, Renata, Czepczynski, Rafał, Maina, Theodosia
Published in Cancers (12.10.2021)
Published in Cancers (12.10.2021)
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Journal Article
Theranostic approaches in nuclear oncology: From bench to bed
Nock, Berthold A., Maina, Theodosia
Published in Journal of labelled compounds & radiopharmaceuticals (01.08.2019)
Published in Journal of labelled compounds & radiopharmaceuticals (01.08.2019)
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Journal Article
Rhenium(I) Tricarbonyl Complexes with (2-Hydroxyphenyl)diphenylphosphine as PO Bidentate Ligand
Shegani, Antonio, Triantis, Charalampos, Nock, Berthold A, Maina, Theodosia, Kiritsis, Christos, Psycharis, Vassilis, Raptopoulou, Catherine, Pirmettis, Ioannis, Tisato, Francesco, Papadopoulos, Minas S
Published in Inorganic chemistry (17.07.2017)
Published in Inorganic chemistry (17.07.2017)
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Journal Article
Functional relevance of genes implicated by obesity genome-wide association study signals for human adipocyte biology
Bernhard, F., Landgraf, K., Klöting, N., Berthold, A., Büttner, P., Friebe, D., Kiess, W., Kovacs, P., Blüher, M., Körner, A.
Published in Diabetologia (01.02.2013)
Published in Diabetologia (01.02.2013)
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Journal Article