Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa
Cotman, Andrej Emanuel, Durcik, Martina, Benedetto Tiz, Davide, Fulgheri, Federica, Secci, Daniela, Sterle, Maša, Možina, Štefan, Skok, Žiga, Zidar, Nace, Zega, Anamarija, Ilaš, Janez, Peterlin Mašič, Lucija, Tomašič, Tihomir, Hughes, Diarmaid, Huseby, Douglas L., Cao, Sha, Garoff, Linnéa, Berruga Fernández, Talía, Giachou, Paraskevi, Crone, Lisa, Simoff, Ivailo, Svensson, Richard, Birnir, Bryndis, Korol, Sergiy V., Jin, Zhe, Vicente, Francisca, Ramos, Maria C., de la Cruz, Mercedes, Glinghammar, Björn, Lenhammar, Lena, Henderson, Sara R., Mundy, Julia E. A., Maxwell, Anthony, Stevenson, Clare E. M., Lawson, David M., Janssen, Guido V., Sterk, Geert Jan, Kikelj, Danijel
Published in Journal of medicinal chemistry (26.01.2023)
Published in Journal of medicinal chemistry (26.01.2023)
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Antibiotic class with potent in vivo activity targeting lipopolysaccharide synthesis in Gram-negative bacteria
Huseby, Douglas L, Cao, Sha, Zamaratski, Edouard, Sooriyaarachchi, Sanjeewani, Ahmad, Shabbir, Bergfors, Terese, Krasnova, Laura, Pelss, Juris, Ikaunieks, Martins, Loza, Einars, Katkevics, Martins, Bobileva, Olga, Cirule, Helena, Gukalova, Baiba, Grinberga, Solveiga, Backlund, Maria, Simoff, Ivailo, Leber, Anna T, Berruga-Fernández, Talía, Antonov, Dmitry, Konda, Vivekananda R, Lindström, Stefan, Olanders, Gustav, Brandt, Peter, Baranczewski, Pawel, Vingsbo Lundberg, Carina, Liepinsh, Edgars, Suna, Edgars, Jones, T Alwyn, Mowbray, Sherry L, Hughes, Diarmaid, Karlén, Anders
Published in Proceedings of the National Academy of Sciences - PNAS (09.04.2024)
Published in Proceedings of the National Academy of Sciences - PNAS (09.04.2024)
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New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate Staphylococcus aureus
Durcik, Martina, Cotman, Andrej Emanuel, Toplak, Žan, Možina, Štefan, Skok, Žiga, Szili, Petra Eva, Czikkely, Márton, Maharramov, Elvin, Vu, Thu Hien, Piras, Maria Vittoria, Zidar, Nace, Ilaš, Janez, Zega, Anamarija, Trontelj, Jurij, Pardo, Luis A., Hughes, Diarmaid, Huseby, Douglas, Berruga-Fernández, Tália, Cao, Sha, Simoff, Ivailo, Svensson, Richard, Korol, Sergiy V., Jin, Zhe, Vicente, Francisca, Ramos, Maria C., Mundy, Julia E. A., Maxwell, Anthony, Stevenson, Clare E. M., Lawson, David M., Glinghammar, Björn, Sjöström, Eva, Bohlin, Martin, Oreskär, Joanna, Alvér, Sofie, Janssen, Guido V., Sterk, Geert Jan, Kikelj, Danijel, Pal, Csaba, Tomašič, Tihomir, Peterlin Mašič, Lucija
Published in Journal of medicinal chemistry (23.03.2023)
Published in Journal of medicinal chemistry (23.03.2023)
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Antibacterial activity of apramycin at acidic pH warrants wide therapeutic window in the treatment of complicated urinary tract infections and acute pyelonephritis
Becker, Katja, Cao, Sha, Nilsson, Anna, Erlandsson, Maria, Hotop, Sven-Kevin, Kuka, Janis, Hansen, Jon, Haldimann, Klara, Grinberga, Solveiga, Berruga-Fernández, Talia, Huseby, Douglas L., Shariatgorji, Reza, Lindmark, Evelina, Platzack, Björn, Böttger, Erik C., Crich, David, Friberg, Lena E., Vingsbo Lundberg, Carina, Hughes, Diarmaid, Brönstrup, Mark, Andrén, Per E., Liepinsh, Edgars, Hobbie, Sven N.
Published in EBioMedicine (01.11.2021)
Published in EBioMedicine (01.11.2021)
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Risk assessment for the transmission of Middle East respiratory syndrome coronavirus (MERS-CoV) on aircraft: a systematic review
Berruga-Fernández, T., Robesyn, E., Korhonen, T., Penttinen, P., Jansa, J. M.
Published in Epidemiology & Infection (10.06.2021)
Published in Epidemiology & Infection (10.06.2021)
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Book Review
Sleep Architecture in Night Shift Workers Police Officers with Obstructive Sleep Apnea-hypopnea Syndrome
Verde-Tinoco, Selene, Santana-Miranda, Rafael, Gutiérrez-Escobar, Romel, Haro, Reyes, Miranda-Ortiz, Joana, Berruga-Fernandez, Talia, Jimenez-Correa, Ulises, Poblano, Adrián
Published in Sleep science (Sao Paulo, Brazil) (01.01.2017)
Published in Sleep science (Sao Paulo, Brazil) (01.01.2017)
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