Leveraging Compound Promiscuity to Identify Targetable Cysteines within the Kinome
Rao, Suman, Gurbani, Deepak, Du, Guangyan, Everley, Robert A, Browne, Christopher M, Chaikuad, Apirat, Tan, Li, Schröder, Martin, Gondi, Sudershan, Ficarro, Scott B, Sim, Taebo, Kim, Nam Doo, Berberich, Matthew J, Knapp, Stefan, Marto, Jarrod A, Westover, Kenneth D, Sorger, Peter K, Gray, Nathanael S
Published in Cell chemical biology (20.06.2019)
Published in Cell chemical biology (20.06.2019)
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Discovery and resistance mechanism of a selective CDK12 degrader
Jiang, Baishan, Gao, Yang, Che, Jianwei, Lu, Wenchao, Kaltheuner, Ines H, Dries, Ruben, Kalocsay, Marian, Berberich, Matthew J, Jiang, Jie, You, Inchul, Kwiatkowski, Nicholas, Riching, Kristin M, Daniels, Danette L, Sorger, Peter K, Geyer, Matthias, Zhang, Tinghu, Gray, Nathanael S
Published in Nature chemical biology (01.06.2021)
Published in Nature chemical biology (01.06.2021)
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Catalytic Degraders Effectively Address Kinase Site Mutations in EML4-ALK Oncogenic Fusions
Gao, Yang, Jiang, Baishan, Kim, Hellen, Berberich, Matthew J., Che, Jianwei, Donovan, Katherine A., Hatcher, John M., Huerta, Fidel, Kwiatkowski, Nicholas P., Liu, Yingpeng, Liuni, Peter P., Metivier, Rebecca J., Murali, Vineeth K., Nowak, Radosław P., Zhang, Tinghu, Fischer, Eric S., Gray, Nathanael S., Jones, Lyn H.
Published in Journal of medicinal chemistry (27.04.2023)
Published in Journal of medicinal chemistry (27.04.2023)
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Targeting immunosuppressive macrophages overcomes PARP inhibitor resistance in BRCA1-associated triple-negative breast cancer
Mehta, Anita K, Cheney, Emily M, Hartl, Christina A, Pantelidou, Constantia, Oliwa, Madisson, Castrillon, Jessica A, Lin, Jia-Ren, Hurst, Katie E, de Oliveira Taveira, Mateus, Johnson, Nathan T, Oldham, William M, Kalocsay, Marian, Berberich, Matthew J, Boswell, Sarah A, Kothari, Aditi, Johnson, Shawn, Dillon, Deborah A, Lipschitz, Mikel, Rodig, Scott, Santagata, Sandro, Garber, Judy E, Tung, Nadine, Yélamos, José, Thaxton, Jessica E, Mittendorf, Elizabeth A, Sorger, Peter K, Shapiro, Geoffrey I, Guerriero, Jennifer L
Published in Nature cancer (01.01.2021)
Published in Nature cancer (01.01.2021)
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The Activation State of CD4 T Cells Alters Cellular Peptidase Activities, HIV Antigen Processing, and MHC Class I Presentation in a Sequence-Dependent Manner
Boucau, Julie, Madouasse, Julien, Kourjian, Georgio, Carlin, Christopher S, Wambua, Daniel, Berberich, Matthew J, Le Gall, Sylvie
Published in The Journal of immunology (1950) (15.05.2019)
Published in The Journal of immunology (1950) (15.05.2019)
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HIV Protease Inhibitor-Induced Cathepsin Modulation Alters Antigen Processing and Cross-Presentation
Kourjian, Georgio, Rucevic, Marijana, Berberich, Matthew J, Dinter, Jens, Wambua, Daniel, Boucau, Julie, Le Gall, Sylvie
Published in The Journal of immunology (1950) (01.05.2016)
Published in The Journal of immunology (1950) (01.05.2016)
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Discovery of Covalent CDK14 Inhibitors with Pan-TAIRE Family Specificity
Ferguson, Fleur M, Doctor, Zainab M, Ficarro, Scott B, Browne, Christopher M, Marto, Jarrod A, Johnson, Jared L, Yaron, Tomer M, Cantley, Lewis C, Kim, Nam Doo, Sim, Taebo, Berberich, Matthew J, Kalocsay, Marian, Sorger, Peter K, Gray, Nathanael S
Published in Cell chemical biology (20.06.2019)
Published in Cell chemical biology (20.06.2019)
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Analysis of Major Histocompatibility Complex-Bound HIV Peptides Identified from Various Cell Types Reveals Common Nested Peptides and Novel T Cell Responses
Rucevic, Marijana, Kourjian, Georgio, Boucau, Julie, Blatnik, Renata, Garcia Bertran, Wilfredo, Berberich, Matthew J, Walker, Bruce D, Riemer, Angelika B, Le Gall, Sylvie
Published in Journal of virology (01.10.2016)
Published in Journal of virology (01.10.2016)
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Variable processing and cross-presentation of HIV by dendritic cells and macrophages shapes CTL immunodominance and immune escape
Dinter, Jens, Duong, Ellen, Lai, Nicole Y, Berberich, Matthew J, Kourjian, Georgio, Bracho-Sanchez, Edith, Chu, Duong, Su, Hang, Zhang, Shao Chong, Le Gall, Sylvie
Published in PLoS pathogens (01.03.2015)
Published in PLoS pathogens (01.03.2015)
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Impact of Zika virus on the human type I interferon osteoimmune response
Drouin, Arnaud, Wallbillich, Nicholas, Theberge, Marc, Liu, Sharon, Katz, Joshua, Bellovoda, Kamela, Se Yun Cheon, Scarlett, Gootkind, Frederick, Bierman, Emily, Zavras, Jason, Berberich, Matthew J., Kalocsay, Marian, Guastaldi, Fernando, Salvadori, Nicolas, Troulis, Maria, Fusco, Dahlene N.
Published in Cytokine (Philadelphia, Pa.) (01.01.2021)
Published in Cytokine (Philadelphia, Pa.) (01.01.2021)
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Proteomic profiling across breast cancer cell lines and models
Kalocsay, Marian, Berberich, Matthew J, Everley, Robert A, Nariya, Maulik K, Chung, Mirra, Gaudio, Benjamin, Victor, Chiara, Bradshaw, Gary A, Eisert, Robyn J, Hafner, Marc, Sorger, Peter K, Mills, Caitlin E, Subramanian, Kartik
Published in Scientific data (04.08.2023)
Published in Scientific data (04.08.2023)
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A dynamic view of the proteomic landscape during differentiation of ReNcell VM cells, an immortalized human neural progenitor line
Song, Yuyu, Subramanian, Kartik, Berberich, Matthew J, Rodriguez, Steven, Latorre, Isabel J, Luria, Catherine M, Everley, Robert, Albers, Mark W, Mitchison, Timothy J, Sorger, Peter K
Published in Scientific data (19.02.2019)
Published in Scientific data (19.02.2019)
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860 Targeting immunosuppressive macrophages overcomes PARP-inhibitor resistance in BRCA1-associated triple-negative breast cancer
Mehta, Anita, Cheney, Emily, Hartl, Christina, Pantelidou, Constantia, Oliwa, Madison, Castrillon, Jessica, Lin, Jia-Ren, Hurst, Katie, Taveira, Mateus de Oliveira, Johnson, Nathan, Oldham, William, Kalocsay, Marian, Berberich, Matthew, Boswell, Sarah, Kothari, Aditi, Johnson, Shawn, Dillon, Deborah, Lipschitz, Mikel, Rodig, Scott, Santagata, Sandro, Garber, Judy, Tung, Nadine, Yélamos, José, Thaxton, Jessica, Mittendorf, Elizabeth, Sorger, Peter, Shapiro, Geoffrey, Guerriero, Jennifer
Published in Journal for immunotherapy of cancer (01.11.2020)
Published in Journal for immunotherapy of cancer (01.11.2020)
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In vitro evaluation of digestive and endolysosomal enzymes to cleave CML‐modified Ara h 1 peptides
Mattison, Christopher P., Dinter, Jens, Berberich, Matthew J., Chung, Si‐Yin, Reed, Shawndrika S., Le Gall, Sylvie, Grimm, Casey C.
Published in Food science & nutrition (01.07.2015)
Published in Food science & nutrition (01.07.2015)
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Journal Article
The activation state of CD4 T cells alters cellular peptidase activities and HIV antigen processing and MHC-I presentation in a sequence-dependent manner
Boucau, Julie, Madouasse, Julien, Kourjian, Georgio, Carlin, Christopher S., Wambua, Daniel, Berberich, Matthew J., Le Gall, Sylvie
Published in The Journal of immunology (1950) (01.04.2019)
Published in The Journal of immunology (1950) (01.04.2019)
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Journal Article
The modulation of cathepsin activities by HIV protease inhibitors alters the processing and cross-presentation of pathogens
Le Gall, Sylvie, Kourjian, Georgio, Rucevic, Marijana, Berberich, Matthew J, Boucau, Julie
Published in The Journal of immunology (1950) (01.05.2016)
Published in The Journal of immunology (1950) (01.05.2016)
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Journal Article
Abstract P5-04-01: PARP inhibition modulates the infiltration, phenotype and function of tumor-associated macrophages (TAMs) in BRCA-associated breast cancer and can be augmented by harnessing the anti-tumor potential of TAMs
Guerriero, Jennifer L, Mehta, Anita K, Cheney, Emily M, Castrillon, Jessica A., Lin, Jia-Ren, Taveira, Mateus de Oliveira, Sonzogni, Olmo, Pantelidou, Constantia, Hartl, Christina A, Oldham, William M, Johnson, Nathan T, Boswell, Sarah A, Kalocsay, Marian, Berberich, Matthew J, Mei, Sholin, Wang, Dan, Johnson, Shawn, Gross, Brett, Dillon, Deborah A, Lipschitz, Mikel, Gjini, Evisa, Rodig, Scott, Santagata, Sandro, Garber, Judy E, Tung, Nadine, Sorger, Peter, Shapiro, Geoffrey I, Wulf, Gerburg M, Mittendorf, Elizabeth A
Published in Cancer research (Chicago, Ill.) (15.02.2020)
Published in Cancer research (Chicago, Ill.) (15.02.2020)
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Abstract 5333: Combining chemoproteomics with machine learning identifies functionally active covalent fragments for hard-to-drug cancer drivers
Hermann, Johannes C., Everley, Robert, Marholz, Laura, Berberich, Matthew, Yang, Tzu-Yi, Chao, Yu-Hsin, Awol, Abduselam K., Shaghafi, Michael, Yoon, Han, Varma, Rohan, Stein, Reed, Krug, Karsten, Lachtara, Emily, Erlanson, Daniel, Varma, Chris, Webster, Kevin R.
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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