Active site-directed probes targeting dipeptidyl peptidases 8 and 9
Espadinha, Margarida, De Loose, Joni, Corthaut, Sam, Thys, Sofie, Van Rymenant, Yentl, Verhulst, Emile, Benramdane, Siham, Filippi, Nicolò, Augustyns, Koen, Van Wielendaele, Pieter, Pintelon, Isabel, De Meester, Ingrid, Van der Veken, Pieter
Published in European journal of medicinal chemistry (15.04.2024)
Published in European journal of medicinal chemistry (15.04.2024)
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Highly Selective Inhibitors of Dipeptidyl Peptidase 9 (DPP9) Derived from the Clinically Used DPP4-Inhibitor Vildagliptin
Benramdane, Siham, De Loose, Joni, Filippi, Nicolò, Espadinha, Margarida, Beyens, Olivier, Rymenant, Yentl Van, Dirkx, Laura, Bozdag, Murat, Feijens, Pim-Bart, Augustyns, Koen, Caljon, Guy, De Winter, Hans, De Meester, Ingrid, Van der Veken, Pieter
Published in Journal of medicinal chemistry (28.09.2023)
Published in Journal of medicinal chemistry (28.09.2023)
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Journal Article
Vildagliptin‐Derived Dipeptidyl Peptidase 9 (DPP9) Inhibitors: Identification of a DPP8/9‐Specific Lead
Benramdane, Siham, De Loose, Joni, Beyens, Olivier, Van Rymenant, Yentl, Vliegen, Gwendolyn, Augustyns, Koen, De Winter, Hans, De Meester, Ingrid, Van der Veken, Pieter
Published in ChemMedChem (03.08.2022)
Published in ChemMedChem (03.08.2022)
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α‑Amino Diphenyl Phosphonates as Novel Inhibitors of Escherichia coli ClpP Protease
Moreno-Cinos, Carlos, Sassetti, Elisa, Salado, Irene G, Witt, Gesa, Benramdane, Siham, Reinhardt, Laura, Cruz, Cristina D, Joossens, Jurgen, Van der Veken, Pieter, Brötz-Oesterhelt, Heike, Tammela, Päivi, Winterhalter, Mathias, Gribbon, Philip, Windshügel, Björn, Augustyns, Koen
Published in Journal of medicinal chemistry (24.01.2019)
Published in Journal of medicinal chemistry (24.01.2019)
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Journal Article
DPP9 BINDING COMPOUNDS
AUGUSTYNS, Koen, DE WINTER, Hans, BENRAMDANE, Siham, DE MEESTER, Ingrid, BEYENS, Olivier, ESPADINHA, Margarida, DE LOOSE, Joni, FILIPPI, Nicolò, VAN DER VEKEN, Pieter
Year of Publication 07.12.2023
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Year of Publication 07.12.2023
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