New Halogen-Containing Drugs Approved by FDA in 2021: An Overview on Their Syntheses and Pharmaceutical Use
Benedetto Tiz, Davide, Bagnoli, Luana, Rosati, Ornelio, Marini, Francesca, Sancineto, Luca, Santi, Claudio
Published in Molecules (Basel, Switzerland) (02.03.2022)
Published in Molecules (Basel, Switzerland) (02.03.2022)
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Journal Article
FDA-Approved Small Molecules in 2022: Clinical Uses and Their Synthesis
Benedetto Tiz, Davide, Bagnoli, Luana, Rosati, Ornelio, Marini, Francesca, Santi, Claudio, Sancineto, Luca
Published in Pharmaceutics (21.11.2022)
Published in Pharmaceutics (21.11.2022)
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Journal Article
Biorefining Twin Transition: Digitalisation for Bio-based Chemicals/Materials - Discovery, Design and Optimisation
Žula, Matej, Grilc, Miha, Kostyniuk, Andrii, Tofani, Giorgio, Jasiukaitytė-Grojzdek, Edita, Ročnik Kozmelj, Tina, Kumar Chowdari, Ramesh, Lavrič, Žan, Teržan, Janvit, Hočevar, Brigita, Jakob, Ana, Rakić, Emilija, Pomeroy, Brett, Cajnko, Miša Mojca, A Vicente, Filipa, Marinič, Dana, Oberlintner, Ana, Novak, Uroš, Benedetto Tiz, Davide, Huš, Matej, Likozar, Blaž
Published in Chimia (20.12.2023)
Published in Chimia (20.12.2023)
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Journal Article
Practical Synthesis and Application of Halogen-Doped Pyrrole Building Blocks
Cotman, Andrej Emanuel, Guérin, Thomas, Kovačević, Ivana, Benedetto Tiz, Davide, Durcik, Martina, Fulgheri, Federica, Možina, Štefan, Secci, Daniela, Sterle, Maša, Ilaš, Janez, Zega, Anamarija, Zidar, Nace, Mašič, Lucija Peterlin, Tomašič, Tihomir, Leroux, Frédéric R, Hanquet, Gilles, Kikelj, Danijel
Published in ACS omega (13.04.2021)
Published in ACS omega (13.04.2021)
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Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa
Cotman, Andrej Emanuel, Durcik, Martina, Benedetto Tiz, Davide, Fulgheri, Federica, Secci, Daniela, Sterle, Maša, Možina, Štefan, Skok, Žiga, Zidar, Nace, Zega, Anamarija, Ilaš, Janez, Peterlin Mašič, Lucija, Tomašič, Tihomir, Hughes, Diarmaid, Huseby, Douglas L., Cao, Sha, Garoff, Linnéa, Berruga Fernández, Talía, Giachou, Paraskevi, Crone, Lisa, Simoff, Ivailo, Svensson, Richard, Birnir, Bryndis, Korol, Sergiy V., Jin, Zhe, Vicente, Francisca, Ramos, Maria C., de la Cruz, Mercedes, Glinghammar, Björn, Lenhammar, Lena, Henderson, Sara R., Mundy, Julia E. A., Maxwell, Anthony, Stevenson, Clare E. M., Lawson, David M., Janssen, Guido V., Sterk, Geert Jan, Kikelj, Danijel
Published in Journal of medicinal chemistry (26.01.2023)
Published in Journal of medicinal chemistry (26.01.2023)
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Journal Article
Improved N-phenylpyrrolamide inhibitors of DNA gyrase as antibacterial agents for high-priority bacterial strains
Zidar, Nace, Onali, Alessia, Peršolja, Peter, Benedetto Tiz, Davide, Dernovšek, Jaka, Skok, Žiga, Durcik, Martina, Cotman, Andrej Emanuel, Hrast Rambaher, Martina, Cruz, Cristina D., Tammela, Päivi, Senerovic, Lidija, Jovanovic, Milija, Szili, Petra Éva, Czikkely, Márton Simon, Pál, Csaba, Zega, Anamarija, Peterlin Mašič, Lucija, Ilaš, Janez, Tomašič, Tihomir, Kikelj, Danijel
Published in European journal of medicinal chemistry (15.11.2024)
Published in European journal of medicinal chemistry (15.11.2024)
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Journal Article
New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity
Durcik, Martina, Lovison, Denise, Skok, Žiga, Durante Cruz, Cristina, Tammela, Päivi, Tomašič, Tihomir, Benedetto Tiz, Davide, Draskovits, Gábor, Nyerges, Ákos, Pál, Csaba, Ilaš, Janez, Peterlin Mašič, Lucija, Kikelj, Danijel, Zidar, Nace
Published in European journal of medicinal chemistry (25.06.2018)
Published in European journal of medicinal chemistry (25.06.2018)
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Journal Article
New N -phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity
Cotman, Andrej Emanuel, Fulgheri, Federica, Piga, Martina, Peršolja, Peter, Tiz, Davide Benedetto, Skok, Žiga, Durcik, Martina, Sterle, Maša, Dernovšek, Jaka, Cruz, Cristina D, Tammela, Päivi, Szili, Petra Éva, Daruka, Lejla, Pál, Csaba, Zega, Anamarija, Mašič, Lucija Peterlin, Ilaš, Janez, Tomašič, Tihomir, Kikelj, Danijel, Zidar, Nace
Published in RSC advances (04.09.2024)
Published in RSC advances (04.09.2024)
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Journal Article
Developing novel classes of protein kinase CK1δ inhibitors by fusing [1,2,4]triazole with different bicyclic heteroaromatic systems
Grieco, Ilenia, Bissaro, Maicol, Tiz, Davide Benedetto, Perez, Daniel I., Perez, Conception, Martinez, Ana, Redenti, Sara, Mariotto, Elena, Bortolozzi, Roberta, Viola, Giampietro, Cozza, Giorgio, Spalluto, Giampiero, Moro, Stefano, Federico, Stephanie
Published in European journal of medicinal chemistry (15.04.2021)
Published in European journal of medicinal chemistry (15.04.2021)
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Journal Article
An optimised series of substituted N-phenylpyrrolamides as DNA gyrase B inhibitors
Tiz, Davide Benedetto, Skok, Žiga, Durcik, Martina, Tomašič, Tihomir, Mašič, Lucija Peterlin, Ilaš, Janez, Zega, Anamarija, Draskovits, Gábor, Révész, Tamás, Nyerges, Ákos, Pál, Csaba, Cruz, Cristina D., Tammela, Päivi, Žigon, Dušan, Kikelj, Danijel, Zidar, Nace
Published in European journal of medicinal chemistry (01.04.2019)
Published in European journal of medicinal chemistry (01.04.2019)
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