Concerted conformational dynamics and water movements in the ghrelin G protein-coupled receptor
Louet, Maxime, Casiraghi, Marina, Damian, Marjorie, Costa, Mauricio GS, Renault, Pedro, Gomes, Antoniel AS, Batista, Paulo R, M'Kadmi, Céline, Mary, Sophie, Cantel, Sonia, Denoyelle, Severine, Ben Haj Salah, Khoubaib, Perahia, David, Bisch, Paulo M, Fehrentz, Jean-Alain, Catoire, Laurent J, Floquet, Nicolas, Banères, Jean-Louis
Published in eLife (03.09.2021)
Published in eLife (03.09.2021)
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Journal Article
Bergofungin D, a peptaibol template for the introduction of chemical modifications, synthesis of analogs and comparative studies of their structures
Das, Sanjit, Salah, Khoubaib Haj Ben, Wenger, Emmanuel, Legrand, Baptiste, Didierjean, Claude, Inguimbert, Nicolas
Published in Journal of peptide science (01.08.2024)
Published in Journal of peptide science (01.08.2024)
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Journal Article
How are 1,2,3-triazoles accommodated in helical secondary structures?
Salah, Khoubaib Ben Haj, Das, Sanjit, Ruiz, Nicolas, Andreu, Vanessa, Martinez, Jean, Wenger, Emmanuel, Amblard, Muriel, Didierjean, Claude, Legrand, Baptiste, Inguimbert, Nicolas
Published in Organic & biomolecular chemistry (2018)
Published in Organic & biomolecular chemistry (2018)
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Journal Article
Enhancing the Antimicrobial Activity of Alamethicin F50/5 by Incorporating N‐terminal Hydrophobic Triazole Substituents
Das, Sanjit, Ben Haj Salah, Khoubaib, Wenger, Emmanuel, Martinez, Jean, Kotarba, Jules, Andreu, Vanessa, Ruiz, Nicolas, Savini, Filippo, Stella, Lorenzo, Didierjean, Claude, Legrand, Baptiste, Inguimbert, Nicolas
Published in Chemistry : a European journal (19.12.2017)
Published in Chemistry : a European journal (19.12.2017)
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Journal Article
Differential Effects of a Full and Biased Ghrelin Receptor Agonist in a Mouse Kindling Model
Buckinx, An, Van Den Herrewegen, Yana, Pierre, Anouk, Cottone, Eleonora, Ben Haj Salah, Khoubaib, Fehrentz, Jean-Alain, Kooijman, Ron, De Bundel, Dimitri, Smolders, Ilse
Published in International journal of molecular sciences (20.05.2019)
Published in International journal of molecular sciences (20.05.2019)
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Journal Article
Growth hormone secretagogues prevent dysregulation of skeletal muscle calcium homeostasis in a rat model of cisplatin‐induced cachexia
Conte, Elena, Camerino, Giulia Maria, Mele, Antonietta, De Bellis, Michela, Pierno, Sabata, Rana, Francesco, Fonzino, Adriano, Caloiero, Roberta, Rizzi, Laura, Bresciani, Elena, Ben Haj Salah, Khoubaib, Fehrentz, Jean‐Alain, Martinez, Jean, Giustino, Arcangela, Mariggiò, Maria Addolorata, Coluccia, Mauro, Tricarico, Domenico, Lograno, Marcello Diego, De Luca, Annamaria, Torsello, Antonio, Conte, Diana, Liantonio, Antonella
Published in Journal of cachexia, sarcopenia and muscle (01.06.2017)
Published in Journal of cachexia, sarcopenia and muscle (01.06.2017)
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Journal Article
JMV2894, a novel growth hormone secretagogue, accelerates body mass recovery in an experimental model of cachexia
Bresciani, Elena, Rizzi, Laura, Molteni, Laura, Ravelli, Monica, Liantonio, Antonella, Ben Haj Salah, Khoubaib, Fehrentz, Jean-Alain, Martinez, Jean, Omeljaniuk, Robert J., Biagini, Giuseppe, Locatelli, Vittorio, Torsello, Antonio
Published in Endocrine (01.10.2017)
Published in Endocrine (01.10.2017)
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Journal Article
Peptaibols as a model for the insertions of chemical modifications
Das, Sanjit, Ben Haj Salah, Khoubaib, Djibo, Mahamadou, Inguimbert, Nicolas
Published in Archives of biochemistry and biophysics (15.11.2018)
Published in Archives of biochemistry and biophysics (15.11.2018)
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Journal Article
GHSR-D2R heteromerization modulates dopamine signaling through an effect on G protein conformation
Damian, Marjorie, Pons, Véronique, Renault, Pedro, M’Kadmi, Céline, Delort, Bartholomé, Hartmann, Lucie, Kaya, Ali I., Louet, Maxime, Gagne, Didier, Salah, Khoubaib Ben Haj, Denoyelle, Séverine, Ferry, Gilles, Boutin, Jean A., Wagner, Renaud, Fehrentz, Jean-Alain, Martinez, Jean, Marie, Jacky, Floquet, Nicolas, Galès, Céline, Mary, Sophie, Hamm, Heidi E., Banères, Jean-Louis
Published in Proceedings of the National Academy of Sciences - PNAS (24.04.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (24.04.2018)
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Journal Article
Design and characterization of a triazole-based growth hormone secretagogue receptor modulator inhibiting the glucoregulatory and feeding actions of ghrelin
Péraldi-Roux, Sylvie, Bayle, Morgane, M'Kadmi, Céline, Damian, Marjorie, Vaillé, Justine, Fernandez, Gimena, Cornejo, Maria Paula, Marie, Jacky, Banères, Jean-Louis, Ben Haj Salah, Khoubaib, Fehrentz, Jean-Alain, Cantel, Sonia, Perello, Mario, Denoyelle, Séverine, Oiry, Catherine, Neasta, Jérémie
Published in Biochemical pharmacology (01.08.2022)
Published in Biochemical pharmacology (01.08.2022)
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Journal Article
Synthesis of [1,2,4]Triazolo[4,3‑a]piperazin-6-ones: An Approach to the Triazole-Fused Ketopiperazine Scaffold
Ben Haj Salah, Khoubaib, Legrand, Baptiste, Bibian, Mathieu, Wenger, Emmanuel, Fehrentz, Jean-Alain, Denoyelle, Séverine
Published in Organic letters (01.06.2018)
Published in Organic letters (01.06.2018)
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Journal Article
Development of Nonpeptidic Inverse Agonists of the Ghrelin Receptor (GHSR) Based on the 1,2,4-Triazole Scaffold
Haj Salah, Khoubaib Ben, Maingot, Mathieu, Blayo, Anne-Laure, M’Kadmi, Céline, Damian, Marjorie, Mary, Sophie, Cantel, Sonia, Neasta, Jérémie, Oiry, Catherine, Péraldi-Roux, Sylvie, Fernandez, Gimena, Romero, Guadalupe García, Perello, Mario, Marie, Jacky, Banères, Jean-Louis, Fehrentz, Jean-Alain, Denoyelle, Séverine
Published in Journal of medicinal chemistry (08.10.2020)
Published in Journal of medicinal chemistry (08.10.2020)
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Journal Article
Development and validation of LC–MS methods for peptaibol quantification in fungal extracts according to their lengths
Van Bohemen, Anne-Isaline, Zalouk-Vergnoux, Aurore, Poirier, Laurence, Phuong, Nam Ngoc, Inguimbert, Nicolas, Ben Haj Salah, Khoubaib, Ruiz, Nicolas, Pouchus, Yves François
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.01.2016)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.01.2016)
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Journal Article
Development of non-peptidic inverse agonists of the ghrelin receptor (GHSR) based on the 1,2,4-triazole scaffold
Ben Haj Salah, Khoubaib, Maingot, Mathieu, Blayo, Anne-Laure, M'Kadmi, Céline, Damian, Marjorie, Mary, Sophie, Cantel, Sonia, Neasta, Jérémie, Oiry, Catherine, Péraldi-Roux, Sylvie, Fernandez, Gimena, Romero, Guadalupe García, Perello, Mario, Marie, Jacky, Banères, Jean-Louis, Fehrentz, Jean-Alain, Denoyelle, Séverine
Published in Journal of medicinal chemistry (03.09.2020)
Published in Journal of medicinal chemistry (03.09.2020)
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