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Published in Nature communications (21.02.2017)
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Published in Nature chemical biology (01.10.2016)
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RAF inhibitors prime wild-type RAF to activate the MAPK pathway and enhance growth
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Published in Nature (London) (18.03.2010)
Published in Nature (London) (18.03.2010)
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Mechanism of MEK inhibition determines efficacy in mutant KRAS- versus BRAF-driven cancers
Hatzivassiliou, Georgia, Haling, Jacob R, Chen, Huifen, Song, Kyung, Price, Steve, Heald, Robert, Hewitt, Joanne F M, Zak, Mark, Peck, Ariana, Orr, Christine, Merchant, Mark, Hoeflich, Klaus P, Chan, Jocelyn, Luoh, Shiuh-Ming, Anderson, Daniel J, Ludlam, Mary J C, Wiesmann, Christian, Ultsch, Mark, Friedman, Lori S, Malek, Shiva, Belvin, Marcia
Published in Nature (London) (12.09.2013)
Published in Nature (London) (12.09.2013)
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In vivo Antitumor Activity of MEK and Phosphatidylinositol 3-Kinase Inhibitors in Basal-Like Breast Cancer Models
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Published in Clinical cancer research (15.07.2009)
Published in Clinical cancer research (15.07.2009)
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Intermittent Administration of MEK Inhibitor GDC-0973 plus PI3K Inhibitor GDC-0941 Triggers Robust Apoptosis and Tumor Growth Inhibition
HOEFLICH, Klaus P, MERCHANT, Mark, ENGST, Stefan, JOHNSTON, Stuart, FRIEDMAN, Lori S, BELVIN, Marcia, ORR, Christine, CHAN, Jocelyn, DOUG DEN OTTER, BERRY, Leanne, KASMAN, Ian, KOEPPEN, Hartmut, RICE, Ken, YANG, Nai-Ying
Published in Cancer research (Chicago, Ill.) (2012)
Published in Cancer research (Chicago, Ill.) (2012)
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Predictive Biomarkers of Sensitivity to the Phosphatidylinositol 3' Kinase Inhibitor GDC-0941 in Breast Cancer Preclinical Models
O'BRIEN, Carol, WALLIN, Jeffrey J, BEIVIN, Marcia, FRIEDMAN, Lori S, LACKNER, Mark R, SAMPATH, Deepak, GUHATHAKURTA, Debraj, SAVAGE, Heidi, PUNNOOSE, Elizabeth A, GUAN, Jane, BERRY, Leanne, PRIOR, Wei Wei, AMLER, Lukas C
Published in Clinical cancer research (15.07.2010)
Published in Clinical cancer research (15.07.2010)
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An Integrated Genomic Screen Identifies LDHB as an Essential Gene for Triple-Negative Breast Cancer
MCCLELAND, Mark L, ADLER, Adam S, BELVIN, Marcia, HATZIVASSILIOU, Georgia, BLACKWOOD, Elizabeth M, CORSON, Laura, EVANGELISTA, Marie, JIPING ZHA, FIRESTEIN, Ron, YONGLEI SHANG, HUNSAKER, Thomas, TRUONG, Tom, PETERSON, David, TORRES, Eric, LI LI, HALEY, Benjamin, STEPHAN, Jean-Philippe
Published in Cancer research (Chicago, Ill.) (15.11.2012)
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Dual Detection of Fungal Infections in Drosophila via Recognition of Glucans and Sensing of Virulence Factors
Gottar, Marie, Gobert, Vanessa, Matskevich, Alexey A., Reichhart, Jean-Marc, Wang, Chengshu, Butt, Tariq M., Belvin, Marcia, Hoffmann, Jules A., Ferrandon, Dominique
Published in Cell (29.12.2006)
Published in Cell (29.12.2006)
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Combined MEK and ERK inhibition overcomes therapy-mediated pathway reactivation in RAS mutant tumors
Merchant, Mark, Moffat, John, Schaefer, Gabriele, Chan, Jocelyn, Wang, Xi, Orr, Christine, Cheng, Jason, Hunsaker, Thomas, Shao, Lily, Wang, Stephanie J, Wagle, Marie-Claire, Lin, Eva, Haverty, Peter M, Shahidi-Latham, Sheerin, Ngu, Hai, Solon, Margaret, Eastham-Anderson, Jeffrey, Koeppen, Hartmut, Huang, Shih-Min A, Schwarz, Jacob, Belvin, Marcia, Kirouac, Daniel, Junttila, Melissa R
Published in PloS one (05.10.2017)
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Targeting p21-activated kinase 1 (PAK1) to induce apoptosis of tumor cells
Ong, Christy C, Jubb, Adrian M, Haverty, Peter M, Zhou, Wei, Tran, Victoria, Truong, Tom, Turley, Helen, O'Brien, Tom, Vucic, Domagoj, Harris, Adrian L, Belvin, Marcia, Friedman, Lori S, Blackwood, Elizabeth M, Koeppen, Hartmut, Hoeflich, Klaus P
Published in Proceedings of the National Academy of Sciences - PNAS (26.04.2011)
Published in Proceedings of the National Academy of Sciences - PNAS (26.04.2011)
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ERK inhibition overcomes acquired resistance to MEK inhibitors
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Published in Molecular cancer therapeutics (01.05.2012)
Published in Molecular cancer therapeutics (01.05.2012)
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GDC-0941, a Novel Class I Selective PI3K Inhibitor, Enhances the Efficacy of Docetaxel in Human Breast Cancer Models by Increasing Cell Death In Vitro and In Vivo
WALLIN, Jeffrey J, GUAN, Jane, PRIOR, Wei Wei, LEE, Leslie B, BERRY, Leanne, BELMONT, Lisa D, KOEPPEN, Hartmut, BELVIN, Marcia, FRIEDMAN, Lori S, SAMPATH, Deepak
Published in Clinical cancer research (15.07.2012)
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Abstract 4898: Effects of chemotherapeutic agents on the tumor immune microenvironment
Belvin, Marcia P., Luoh, Shiuh-Ming, Cheung, Jeanne, McNamara, Erin, Cubas, Rafael, Kim, Jeong
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Metabolic Response to NAD Depletion across Cell Lines Is Highly Variable
Xiao, Yang, Kwong, Mandy, Daemen, Anneleen, Belvin, Marcia, Liang, Xiaorong, Hatzivassiliou, Georgia, O'Brien, Thomas
Published in PloS one (06.10.2016)
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Phosphoproteomic characterization of DNA damage response in melanoma cells following MEK/PI3K dual inhibition
Kirkpatrick, Donald S., Bustos, Daisy J., Dogan, Taner, Chan, Jocelyn, Phu, Lilian, Young, Amy, Friedman, Lori S., Belvin, Marcia, Song, Qinghua, Bakalarski, Corey E., Hoeflich, Klaus P.
Published in Proceedings of the National Academy of Sciences - PNAS (26.11.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (26.11.2013)
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Bridging the Gap between Preclinical and Clinical Studies Using Pharmacokinetic-Pharmacodynamic Modeling: An Analysis of GDC-0973, a MEK Inhibitor
WONG, Harvey, VERNILLET, Laurent, HOEFLICH, Klaus P, YONGCHANG SHI, AFTAB, Blake T, AOYAMA, Ron, TAN LAM, Sanh, BELVIN, Marcia, PRESCOTT, John, PETERSON, Amy, WARE, Joseph A, LEE, Lillian, MARTINI, Jean-Francois, PEIWEN YU, CONGFEN LI, DEL ROSARIO, Geoffrey, CHOO, Edna F
Published in Clinical cancer research (01.06.2012)
Published in Clinical cancer research (01.06.2012)
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Abstract 4905: Effects of MAPK pathway inhibitors in the tumor immune microenvironment
Belvin, Marcia P., Williams, Erin, Luoh, Shiuh-Ming, Cheung, Jeanne, Orr, Christine, Chan, Emily, Ebert, Peter, Mellman, Ira, Kim, Jeong, Merchant, Mark
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Suppression of HER2/HER3-Mediated Growth of Breast Cancer Cells with Combinations of GDC-0941 PI3K Inhibitor, Trastuzumab, and Pertuzumab
Yao, Evelyn, Zhou, Wei, Lee-Hoeflich, Si Tuen, Truong, Tom, Haverty, Peter M, Eastham-Anderson, Jeffrey, Lewin-Koh, Nicholas, Gunter, Bert, Belvin, Marcia, Murray, Lesley J, Friedman, Lori S, Sliwkowski, Mark X, Hoeflich, Klaus P
Published in Clinical cancer research (15.06.2009)
Published in Clinical cancer research (15.06.2009)
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Systematic generation of high-resolution deletion coverage of the Drosophila melanogaster genome
Friedman, Lori, Deal, Jennifer E, Howie, Elizabeth, Tan, Lory R, Edgar, Kyle A, Plowman, Gregory D, Marcinko, Marie, Winter, Christopher G, Milash, Brett, Winner, Millicent A, Cook, Kevin R, Parks, Annette L, Belvin, Marcia, Fawcett, Robert, Andrade, Rachel S, Kopczynski, Casey, Killpack, Keith, Duyk, Geoffrey, Grant, Deanna, Shaw, Kenneth J, Huppert, Kari, Miyazaki, Wesley Y, Margolis, Jonathan, Tabios, Mariano, Thao, Doua, Vysotskaia, Valentina, Kaufman, Thomas C, Zhao, Lora, Francis-Lang, Helen L, Robertson, Stephanie, Dompe, Nicholas A, Curtis, Daniel, Whittaker, Kellie, Deal-Herr, Megan E, Norton, Amanda, Bogart, Kevin P, Singer, Matthew A
Published in Nature genetics (01.03.2004)
Published in Nature genetics (01.03.2004)
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