Identification of a human estrogen receptor α tetrapeptidic fragment with dual antiproliferative and anti-nociceptive action
Jouffre, Baptiste, Acramel, Alexandre, Belnou, Mathilde, Santolla, Maria Francesca, Talia, Marianna, Lappano, Rosamaria, Nemati, Fariba, Decaudin, Didier, Khemtemourian, Lucie, Liu, Wang-Qing, Maggiolini, Marcello, Eschalier, Alain, Mallet, Christophe, Jacquot, Yves
Published in Scientific reports (24.01.2023)
Published in Scientific reports (24.01.2023)
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Interaction of the Anti-Proliferative GPER Inverse Agonist ERα17p with the Breast Cancer Cell Plasma Membrane: From Biophysics to Biology
Trichet, Michaël, Lappano, Rosamaria, Belnou, Mathilde, Salazar Vazquez, Lilian Shadai, Alves, Isabel, Ravault, Delphine, Sagan, Sandrine, Khemtemourian, Lucie, Maggiolini, Marcello, Jacquot, Yves
Published in Cells (Basel, Switzerland) (15.02.2020)
Published in Cells (Basel, Switzerland) (15.02.2020)
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Bio-inspired hybrid fluorescent ligands for the FK1 domain of FKBP52
Li de La Sierra Gallay, Ines, Belnou, Mathilde, Chambraud, Beatrice, Genet, Melanie, van Tilbeurgh, Herman, Nicaise, Magali, Desmadril, Michel, Baulieu, Etienne-Emile, Jacquot, Yves, Byrne, Cillian
Published in Journal of medicinal chemistry (2020)
Published in Journal of medicinal chemistry (2020)
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Journal Article
Bioinspired Hybrid Fluorescent Ligands for the FK1 Domain of FKBP52
de la Sierra-Gallay, Inès Li, Belnou, Mathilde, Chambraud, Béatrice, Genet, Melanie, van Tilbeurgh, Herman, Aumont-Nicaise, Magali, Desmadril, Michel, Baulieu, Etienne-Emile, Jacquot, Yves, Byrne, Cillian
Published in Journal of medicinal chemistry (24.09.2020)
Published in Journal of medicinal chemistry (24.09.2020)
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Journal Article
Improvement of the anti-proliferative activity of the peptide ERα17p in MCF-7 breast cancer cells using nanodiamonds
Yip, François, Nemati, Fariba, El Botty, Rania, Belnou, Mathilde, Decaudin, Didier, Mansuy, Christelle, Jacquot, Yves
Published in Annales pharmaceutiques françaises (01.11.2019)
Published in Annales pharmaceutiques françaises (01.11.2019)
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A β‑Turn Motif in the Steroid Hormone Receptor’s Ligand-Binding Domains Interacts with the Peptidyl-prolyl Isomerase (PPIase) Catalytic Site of the Immunophilin FKBP52
Byrne, Cillian, Henen, Morkos A, Belnou, Mathilde, Cantrelle, François-Xavier, Kamah, Amina, Qi, Haoling, Giustiniani, Julien, Chambraud, Béatrice, Baulieu, Etienne-Emile, Lippens, Guy, Landrieu, Isabelle, Jacquot, Yves
Published in Biochemistry (Easton) (27.09.2016)
Published in Biochemistry (Easton) (27.09.2016)
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