Small molecule allosteric inhibitors of RORγt block Th17-dependent inflammation and associated gene expression in vivo
Saenz, Steven A, Local, Andrea, Carr, Tiffany, Shakya, Arvind, Koul, Shivsmriti, Hu, Haiqing, Chourb, Lisa, Stedman, Justin, Malley, Jenna, D'Agostino, Laura Akullian, Shanmugasundaram, Veerabahu, Malona, John, Schwartz, C Eric, Beebe, Lisa, Clements, Meghan, Rajaraman, Ganesh, Cho, John, Jiang, Lan, Dubrovskiy, Alex, Kreilein, Matt, Shimanovich, Roman, Hamann, Lawrence G, Escoubet, Laure, Ellis, J Michael
Published in PloS one (09.11.2021)
Published in PloS one (09.11.2021)
Get full text
Journal Article
Efficacy of a Covalent ERK1/2 Inhibitor, CC-90003, in KRAS-Mutant Cancer Models Reveals Novel Mechanisms of Response and Resistance
Aronchik, Ida, Dai, Yumin, Labenski, Matt, Barnes, Carmen, Jones, Terri, Qiao, Lixin, Beebe, Lisa, Malek, Mehnaz, Elis, Winfried, Shi, Tao, Mavrommatis, Konstantinos, Bray, Gordon L, Filvaroff, Ellen H
Published in Molecular cancer research (01.02.2019)
Published in Molecular cancer research (01.02.2019)
Get full text
Journal Article
Discovery of CC-99677, a selective targeted covalent MAPKAPK2 (MK2) inhibitor for autoimmune disorders
Malona, JOHN, CHUAQUI, CLAUDIO, SELETSKY, BORIS M., BEEBE, LISA, CANTIN, SUSAN, KALKEN, DANIEL VAN, FAHNOE, KELLY, WANG, ZHIGANG, BROWNING, BETH, SZABO, HILARY, KOOPMAN, LOUISE A., ORAVECZ, TAMAS, MCDONALD, JOSEPH J., RAMIREZ-VALLE, FRANCISCO, GAUR, RAJULA, MENSAH, KOFI A., THOMAS, MICHAEL, CONNARN, JAMIE N., HU, HAIQING, ALEXANDER, MATTHEW D., CORIN, ALAN F.
Published in Translational research : the journal of laboratory and clinical medicine (01.11.2022)
Published in Translational research : the journal of laboratory and clinical medicine (01.11.2022)
Get full text
Journal Article
Small molecule allosteric inhibitors of ROR[gamma]t block Th17-dependent inflammation and associated gene expression in vivo
Saenz, Steven A, Local, Andrea, Carr, Tiffany, Shakya, Arvind, Koul, Shivsmriti, Hu, Haiqing, Chourb, Lisa, Stedman, Justin, Malley, Jenna, D'Agostino, Laura Akullian, Shanmugasundaram, Veerabahu, Malona, John, Schwartz, C. Eric, Beebe, Lisa, Clements, Meghan, Rajaraman, Ganesh, Cho, John, Jiang, Lan, Dubrovskiy, Alex, Kreilein, Matt, Shimanovich, Roman, Hamann, Lawrence G, Escoubet, Laure, Ellis, J. Michael
Published in PloS one (09.11.2021)
Published in PloS one (09.11.2021)
Get full text
Journal Article
Promotion of N-nitrosodiethylamine-initiated hepatocellular tumors and hepatoblastomas by 2,3,7,8-tetrachlorodibenzo-p-dioxin or Aroclor 1254 in C57BL/6, DBA/2, and B6D2F1 mice
BEEBE, L. E, FORNWALD, L. W, DIWAN, B. A, ANVER, M. R, ANDERSON, L. M
Published in Cancer research (Chicago, Ill.) (01.11.1995)
Get full text
Published in Cancer research (Chicago, Ill.) (01.11.1995)
Journal Article
아프레밀라스트 및 TYK2 억제제를 포함하는 조합 요법
BUCHWALTER GILLES, PLENGE ROBERT, TZENG TE CHEN, ADAMS MARY, CARR TIFFANY, SCHAFER PETER HENRY, BEEBE LISA
Year of Publication 06.01.2022
Get full text
Year of Publication 06.01.2022
Patent
아프레밀라스트 및 TYK2 억제제를 포함하는 조합 요법
BUCHWALTER GILLES, PLENGE ROBERT, TZENG TE CHEN, ADAMS MARY, CARR TIFFANY, SCHAFER PETER HENRY, BEEBE LISA
Year of Publication 06.01.2022
Get full text
Year of Publication 06.01.2022
Patent
Small molecule allosteric inhibitors of RORγt block Th17-dependent inflammation and associated gene expression in vivo
Steven A. Saenz, Andrea Local, Tiffany Carr, Arvind Shakya, Shivsmriti Koul, Haiqing Hu, Lisa Chourb, Justin Stedman, Jenna Malley, Laura Akullian D’Agostino, Veerabahu Shanmugasundaram, John Malona, C. Eric Schwartz, Lisa Beebe, Meghan Clements, Ganesh Rajaraman, John Cho, Lan Jiang, Alex Dubrovskiy, Matt Kreilein, Roman Shimanovich, Lawrence G. Hamann, Laure Escoubet, J. Michael Ellis
Published in PloS one (01.01.2021)
Get full text
Published in PloS one (01.01.2021)
Journal Article
Paradigm of combination biologics: analytical challenges related to pharmacokinetic assays and interpretation of pharmacokinetic and immunogenicity results
Stevenson, Lauren, Zinnack, Kimberly, Donley, Jean, Beebe, Lisa, Amaravadi, Lakshmi
Published in Bioanalysis (01.03.2011)
Published in Bioanalysis (01.03.2011)
Get more information
Journal Article
Induction of hepatic CYP1A in male F344/NCr rats by dietary exposure to Aroclor 1254: examination of immunochemical, RNA, catalytic, and pharmacokinetic endpoints
Nims, R W, Beebe, L E, Dragnev, K H, Thomas, P E, Fox, S D, Issaq, H J, Jones, C R, Lubet, R A
Published in Environmental research (01.12.1992)
Published in Environmental research (01.12.1992)
Get more information
Journal Article
An IFN-beta-albumin fusion protein that displays improved pharmacokinetic and pharmacodynamic properties in nonhuman primates
Sung, Cynthia, Nardelli, Bernardetta, LaFleur, David W, Blatter, Erich, Corcoran, Marta, Olsen, Henrik S, Birse, Charles E, Pickeral, Oxana K, Zhang, Junli, Shah, Devanshi, Moody, Gordon, Gentz, Solange, Beebe, Lisa, Moore, Paul A
Published in Journal of interferon & cytokine research (01.01.2003)
Published in Journal of interferon & cytokine research (01.01.2003)
Get full text
Journal Article
COMBINATION THERAPIES COMPRISING APREMILAST AND TYK2 INHIBITORS
Carr, Tiffany, Schafer, Peter Henry, Tzeng, Te-chen, Plenge, Robert, Buchwalter, Gilles, Beebe, Lisa, Adams, Mary
Year of Publication 27.10.2022
Get full text
Year of Publication 27.10.2022
Patent
Combination therapies comprising apremilast and Tyk2 inhibitors
Carr, Tiffany, Schafer, Peter Henry, Tzeng, Te-chen, Plenge, Robert, Buchwalter, Gilles, Beebe, Lisa, Adams, Mary
Year of Publication 14.06.2022
Get full text
Year of Publication 14.06.2022
Patent
COMBINATION THERAPIES COMPRISING APREMILAST AND TYK2 INHIBITORS
BEEBE, Lisa, ADAMS, Mary, CARR, Tiffany, PLENGE, Robert, TZENG, Te-Chen, SCHAFER, Peter Henry, BUCHWALTER, Gilles
Year of Publication 09.03.2022
Get full text
Year of Publication 09.03.2022
Patent
POLYTHÉRAPIES COMPRENANT DE L'APRÉMILAST ET DES INHIBITEURS DE TYK2
BEEBE, Lisa, ADAMS, Mary, CARR, Tiffany, PLENGE, Robert, TZENG, Te-Chen, BUCHWALTER, Gilles, SCHAFER, Peter Henry
Year of Publication 09.03.2022
Get full text
Year of Publication 09.03.2022
Patent
COMBINATION THERAPIES COMPRISING APREMILAST AND TYK2 INHIBITORS
BEEBE, Lisa, ADAMS, Mary, CARR, Tiffany, PLENGE, Robert, TZENG, Te-Chen, SCHAFER, Peter Henry, BUCHWALTER, Gilles
Year of Publication 09.03.2022
Get full text
Year of Publication 09.03.2022
Patent
Combination therapies comprising apremilast and Tyk2 inhibitors
BEEBE, Lisa, ADAMS, Mary, CARR, Tiffany, PLENGE, Robert, TZENG, Te-Chen, SCHAFER, Peter Henry, BUCHWALTER, Gilles
Year of Publication 02.12.2021
Get full text
Year of Publication 02.12.2021
Patent
Combination therapies comprising apremilast and Tyk2 inhibitors
BEEBE, Lisa, ADAMS, Mary, CARR, Tiffany, PLENGE, Robert, TZENG, Te-Chen, SCHAFER, Peter Henry, BUCHWALTER, Gilles
Year of Publication 02.12.2021
Get full text
Year of Publication 02.12.2021
Patent
COMBINATION THERAPIES COMPRISING APREMILAST AND TYK2 INHIBITORS
BEEBE, Lisa, ADAMS, Mary, CARR, Tiffany, PLENGE, Robert, TZENG, Te-Chen, SCHAFER, Peter Henry, BUCHWALTER, Gilles
Year of Publication 29.11.2021
Get full text
Year of Publication 29.11.2021
Patent