Structural insights and in vitro reconstitution of membrane targeting and activation of human PI4KB by the ACBD3 protein
Klima, Martin, Tóth, Dániel J, Hexnerova, Rozalie, Baumlova, Adriana, Chalupska, Dominika, Tykvart, Jan, Rezabkova, Lenka, Sengupta, Nivedita, Man, Petr, Dubankova, Anna, Humpolickova, Jana, Nencka, Radim, Veverka, Vaclav, Balla, Tamas, Boura, Evzen
Published in Scientific reports (24.03.2016)
Published in Scientific reports (24.03.2016)
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A large scale high-throughput screen identifies chemical inhibitors of phosphatidylinositol 4-kinase type II alpha[S]
Sengupta, Nivedita, Jović, Marko, Barnaeva, Elena, Kim, David W., Hu, Xin, Southall, Noel, Dejmek, Milan, Mejdrova, Ivana, Nencka, Radim, Baumlova, Adriana, Chalupska, Dominika, Boura, Evzen, Ferrer, Marc, Marugan, Juan, Balla, Tamas
Published in Journal of lipid research (01.03.2019)
Published in Journal of lipid research (01.03.2019)
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Rational Design of Novel Highly Potent and Selective Phosphatidylinositol 4‑Kinase IIIβ (PI4KB) Inhibitors as Broad-Spectrum Antiviral Agents and Tools for Chemical Biology
Mejdrová, Ivana, Chalupská, Dominika, Plačková, Pavla, Müller, Christin, Šála, Michal, Klíma, Martin, Baumlová, Adriana, Hřebabecký, Hubert, Procházková, Eliška, Dejmek, Milan, Strunin, Dmytro, Weber, Jan, Lee, Gary, Matoušová, Marika, Mertlíková-Kaiserová, Helena, Ziebuhr, John, Birkus, Gabriel, Boura, Evzen, Nencka, Radim
Published in Journal of medicinal chemistry (12.01.2017)
Published in Journal of medicinal chemistry (12.01.2017)
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Highly Selective Phosphatidylinositol 4‑Kinase IIIβ Inhibitors and Structural Insight into Their Mode of Action
Mejdrová, Ivana, Chalupská, Dominika, Kögler, Martin, Šála, Michal, Plačková, Pavla, Baumlová, Adriana, Hřebabecký, Hubert, Procházková, Eliška, Dejmek, Milan, Guillon, Rémi, Strunin, Dmytro, Weber, Jan, Lee, Gary, Birkus, Gabriel, Mertlíková-Kaiserová, Helena, Boura, Evzen, Nencka, Radim
Published in Journal of medicinal chemistry (14.05.2015)
Published in Journal of medicinal chemistry (14.05.2015)
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Kobuviral Non-structural 3A Proteins Act as Molecular Harnesses to Hijack the Host ACBD3 Protein
Klima, Martin, Chalupska, Dominika, Różycki, Bartosz, Humpolickova, Jana, Rezabkova, Lenka, Silhan, Jan, Baumlova, Adriana, Dubankova, Anna, Boura, Evzen
Published in Structure (London) (07.02.2017)
Published in Structure (London) (07.02.2017)
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The crystal structure of the phosphatidylinositol 4-kinase IIα
Baumlova, Adriana, Chalupska, Dominika, Róźycki, Bartosz, Jovic, Marko, Wisniewski, Eva, Klima, Martin, Dubankova, Anna, Kloer, Daniel P, Nencka, Radim, Balla, Tamas, Boura, Evzen
Published in EMBO reports (01.10.2014)
Published in EMBO reports (01.10.2014)
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The high-resolution crystal structure of phosphatidylinositol 4-kinase IIβ and the crystal structure of phosphatidylinositol 4-kinase IIα containing a nucleoside analogue provide a structural basis for isoform-specific inhibitor design
Klima, Martin, Baumlova, Adriana, Chalupska, Dominika, Hřebabecký, Hubert, Dejmek, Milan, Nencka, Radim, Boura, Evzen
Published in Acta crystallographica. Section D, Biological crystallography. (01.07.2015)
Published in Acta crystallographica. Section D, Biological crystallography. (01.07.2015)
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Journal Article
The crystal structure of the phosphatidylinositol 4-kinase II[alpha]
Baumlova, Adriana, Chalupska, Dominika, Roycki, Bartosz, Jovic, Marko, Wisniewski, Eva, Klima, Martin, Dubankova, Anna, Kloer, Daniel P, Nencka, Radim, Balla, Tamas, Boura, Evzen
Published in EMBO reports (01.10.2014)
Published in EMBO reports (01.10.2014)
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Journal Article
The high-resolution crystal structure of phosphatidylinositol 4-kinase II[beta] and the crystal structure of phosphatidylinositol 4-kinase II[alpha] containing a nucleoside analogue provide a structural basis for isoform-specific inhibitor design
Klima, Martin, Baumlova, Adriana, Chalupska, Dominika, Hrebabecky, Hubert, Dejmek, Milan, Nencka, Radim, Boura, Evzen
Published in Acta crystallographica. Section D, Biological crystallography. (01.07.2015)
Published in Acta crystallographica. Section D, Biological crystallography. (01.07.2015)
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