Prodrugs of Perzinfotel with Improved Oral Bioavailability
Baudy, Reinhardt B, Butera, John A, Abou-Gharbia, Magid A, Chen, Hong, Harrison, Boyd, Jain, Uday, Magolda, Ronald, Sze, Jean Y, Brandt, Michael R, Cummons, Terri A, Kowal, Diane, Pangalos, Menelas N, Zupan, Bojana, Hoffmann, Matthew, May, Michael, Mugford, Cheryl, Kennedy, Jeffrey, Childers, Wayne E
Published in Journal of medicinal chemistry (12.02.2009)
Published in Journal of medicinal chemistry (12.02.2009)
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Journal Article
Characterization of Two Novel N-Methyl-D-aspartate Antagonists: EAA-090 (2-[8,9-Dioxo-2,6-diazabicyclo [5.2.0]non-1(7)-en2-yl]ethylphosphonic Acid) and EAB-318 (R-α-Amino-5-chloro-1-(phosphonomethyl)-1H-benzimidazole-2-propanoic Acid Hydrochloride)
Sun, Lucy, Chiu, Doreen, Kowal, Dianne, Simon, Rachelle, Smeyne, Michelle, Zukin, R Suzanne, Olney, John, Baudy, Reinhardt, Lin, Stephen
Published in The Journal of pharmacology and experimental therapeutics (01.08.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2004)
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Journal Article
Design, Synthesis, SAR, and Biological Evaluation of Highly Potent Benzimidazole-Spaced Phosphono-α-Amino Acid Competitive NMDA Antagonists of the AP-6 Type
Baudy, Reinhardt B, Yardley, John P, Zaleska, Margaret M, Bramlett, Donna R, Tasse, Rene P, Kowal, Dianne M, Katz, Alan H, Moyer, John A, Abou-Gharbia, Magid
Published in Journal of medicinal chemistry (10.05.2001)
Published in Journal of medicinal chemistry (10.05.2001)
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Journal Article
Potent quinoxaline-spaced phosphono .alpha.-amino acids of the AP-6 type as competitive NMDA antagonists: synthesis and biological evaluation
Baudy, Reinhardt B, Greenblatt, Lynne P, Jirkovsky, Ivo L, Conklin, Mary, Russo, Ralph J, Bramlett, Donna R, Emrey, Tracy A, Simmonds, Joanne T, Kowal, Dianne M
Published in Journal of medicinal chemistry (01.02.1993)
Published in Journal of medicinal chemistry (01.02.1993)
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Journal Article
Advances toward New Antidepressants with Dual Serotonin Transporter and 5-HT1A Receptor Affinity within a Class of 3-Aminochroman Derivatives. Part 2
Hatzenbuhler, Nicole T, Baudy, Reinhardt, Evrard, Deborah A, Failli, Amedeo, Harrison, Boyd L, Lenicek, Steven, Mewshaw, Richard E, Saab, Annmarie, Shah, Uresh, Sze, Jean, Zhang, Minsheng, Zhou, Dahui, Chlenov, Michael, Kagan, Michael, Golembieski, Jeannette, Hornby, Geoffrey, Lai, Margaret, Smith, Deborah L, Sullivan, Kelly M, Schechter, Lee E, Andree, Terrance H
Published in Journal of medicinal chemistry (13.11.2008)
Published in Journal of medicinal chemistry (13.11.2008)
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Journal Article
Advances toward New Antidepressants with Dual Serotonin Transporter and 5-HT 1A Receptor Affinity within a Class of 3-Aminochroman Derivatives. Part 2
Hatzenbuhler, Nicole T., Baudy, Reinhardt, Evrard, Deborah A., Failli, Amedeo, Harrison, Boyd L., Lenicek, Steven, Mewshaw, Richard E., Saab, Annmarie, Shah, Uresh, Sze, Jean, Zhang, Minsheng, Zhou, Dahui, Chlenov, Michael, Kagan, Michael, Golembieski, Jeannette, Hornby, Geoffrey, Lai, Margaret, Smith, Deborah L., Sullivan, Kelly M., Schechter, Lee E., Andree, Terrance H.
Published in Journal of medicinal chemistry (13.11.2008)
Published in Journal of medicinal chemistry (13.11.2008)
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Journal Article
Octahydropyrazino[2',3':3,4]pyrido[1,2-a]indoles. A new class of potent antihypertensive agents
Jirkovsky, Ivo, Santroch, George, Baudy, Reinhardt, Oshiro, George
Published in Journal of medicinal chemistry (01.02.1987)
Published in Journal of medicinal chemistry (01.02.1987)
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Journal Article
Characterization of Two Novel N -Methyl-D-aspartate Antagonists: EAA-090 (2-[8,9-Dioxo-2,6-diazabicyclo [5.2.0]non-1(7)-en2-yl]ethylphosphonic Acid) and EAB-318 ( R -α-Amino-5-chloro-1-(phosphonomethyl)-1 H -benzimidazole-2-propanoic Acid Hydrochloride)
Sun, Lucy, Chiu, Doreen, Kowal, Dianne, Simon, Rachelle, Smeyne, Michelle, Zukin, R. Suzanne, Olney, John, Baudy, Reinhardt, Lin, Stephen
Published in The Journal of pharmacology and experimental therapeutics (01.08.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2004)
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Journal Article
Corrigendum to “Synthesis, characterization, and evaluation of pro-drugs of VLA-4 antagonists”
Huryn, D.M., Ashwell, Susan, Baudy, Reinhardt, Dressen, Darren B., Gallaway, William, Grant, Francine S., Konradi, Andrei, Ley, Robert W., Petusky, Susan, Pleiss, Michael A., Sarantakis, Dimitri, Semko, Christopher M., Sherman, Mary M., Tio, Cesar, Zhang, Lu
Published in Bioorganic & medicinal chemistry letters (01.11.2004)
Published in Bioorganic & medicinal chemistry letters (01.11.2004)
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Journal Article
Synthesis of the Four 3-Aminotricyclo [2.2.1.0(2,6)] Heptane-1,3-Dicarboxylic Acid Isomers
Baudy, Reinhardt B., Sze, Jean Y., Butera, John A.
Published in Synthetic communications (31.12.2004)
Published in Synthetic communications (31.12.2004)
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Journal Article
Synthesis, characterization and evaluation of pro-drugs of VLA-4 antagonists
Huryn, Donna M, Ashwell, Susan, Baudy, Reinhardt, Dressen, Darren B, Gallaway, William, Grant, Francine S, Konradi, Andrei, Ley, Robert W, Petusky, Susan, Pleiss, Michael A, Sarantakis, Dimitri, Semko, Christopher M, Sherman, Mary M, Tio, Cesar, Zhang, Lu
Published in Bioorganic & medicinal chemistry letters (05.04.2004)
Published in Bioorganic & medicinal chemistry letters (05.04.2004)
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