Synergistic Experimental and Computational Investigation of the Bioorthogonal Reactivity of Substituted Aryltetrazines
Battisti, Umberto M, García-Vázquez, Rocío, Svatunek, Dennis, Herrmann, Barbara, Löffler, Andreas, Mikula, Hannes, Herth, Matthias Manfred
Published in Bioconjugate chemistry (20.04.2022)
Published in Bioconjugate chemistry (20.04.2022)
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Journal Article
Analytical and preparative enantioseparation and main chiroptical properties of Iridium(III) bis(4,6-difluorophenylpyridinato)picolinato
Citti, Cinzia, Battisti, Umberto M., Ciccarella, Giuseppe, Maiorano, Vincenzo, Gigli, Giuseppe, Abbate, Sergio, Mazzeo, Giuseppe, Castiglioni, Ettore, Longhi, Giovanna, Cannazza, Giuseppe
Published in Journal of Chromatography A (07.10.2016)
Published in Journal of Chromatography A (07.10.2016)
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Journal Article
Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry
Stéen, E. Johanna L, Jørgensen, Jesper T, Denk, Christoph, Battisti, Umberto M, Nørregaard, Kamilla, Edem, Patricia E, Bratteby, Klas, Shalgunov, Vladimir, Wilkovitsch, Martin, Svatunek, Dennis, Poulie, Christian B. M, Hvass, Lars, Simón, Marina, Wanek, Thomas, Rossin, Raffaella, Robillard, Marc, Kristensen, Jesper L, Mikula, Hannes, Kjaer, Andreas, Herth, Matthias M
Published in ACS pharmacology & translational science (09.04.2021)
Published in ACS pharmacology & translational science (09.04.2021)
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Journal Article
Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET
Schlein, Eva, Rokka, Johanna, Odell, Luke R., van den Broek, Sara Lopes, Herth, Matthias M., Battisti, Umberto M., Syvänen, Stina, Sehlin, Dag, Eriksson, Jonas
Published in EJNMMI radiopharmacy and chemistry (06.03.2024)
Published in EJNMMI radiopharmacy and chemistry (06.03.2024)
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Journal Article
A Fluorescent Probe as a Lead Compound for a Selective α‑Synuclein PET Tracer: Development of a Library of 2‑Styrylbenzothiazoles and Biological Evaluation of [18F]PFSB and [18F]MFSB
Di Nanni, Adriana, Saw, Ran Sing, Battisti, Umberto M., Bowden, Gregory D., Boeckermann, Adam, Bjerregaard-Andersen, Kaare, Pichler, Bernd J., Herfert, Kristina, Herth, Matthias M., Maurer, Andreas
Published in ACS omega (29.08.2023)
Published in ACS omega (29.08.2023)
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Journal Article
Development of the First Aliphatic 18 F-Labeled Tetrazine Suitable for Pretargeted PET Imaging-Expanding the Bioorthogonal Tool Box
Battisti, Umberto M, Bratteby, Klas, Jørgensen, Jesper T, Hvass, Lars, Shalgunov, Vladimir, Mikula, Hannes, Kjær, Andreas, Herth, Matthias Manfred
Published in Journal of medicinal chemistry (28.10.2021)
Published in Journal of medicinal chemistry (28.10.2021)
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Journal Article
Evaluation of F-537-Tetrazine in a model for brain pretargeting imaging. Comparison to N-(3-[18F] fluoro-5-(1,2,4,5-tetrazin-3-yl)benzyl)propan-1-amine
Shalgunov, Vladimir, van den Broek, Sara Lopes, Andersen, Ida Vang, Raval, Nakul R., Schäfer, Gabriela, Barz, Matthias, Herth, Matthias M., Battisti, Umberto M.
Published in Nuclear medicine and biology (01.01.2024)
Published in Nuclear medicine and biology (01.01.2024)
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Journal Article
Spiroxatrine derivatives towards 5-HT1A receptor selectivity
Sorbi, Claudia, Tait, Annalisa, Battisti, Umberto M., Brasili, Livio
Published in Pharmacological reports (01.04.2020)
Published in Pharmacological reports (01.04.2020)
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Journal Article
Functional characterization of N-octyl 4-methylamphetamine variants and related bivalent compounds at the dopamine and serotonin transporters using Ca2+ channels as sensors
Ruchala, Iwona, Battisti, Umberto M., Nguyen, Vy T., Chen, Rita Yu-Tzu, Glennon, Richard A., Eltit, Jose M.
Published in Toxicology and applied pharmacology (15.05.2021)
Published in Toxicology and applied pharmacology (15.05.2021)
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Journal Article
Synthesis, biological evaluation and molecular modeling of 1-oxa-4-thiaspiro- and 1,4-dithiaspiro[4.5]decane derivatives as potent and selective 5-HT1A receptor agonists
Franchini, Silvia, Manasieva, Leda Ivanova, Sorbi, Claudia, Battisti, Umberto M., Fossa, Paola, Cichero, Elena, Denora, Nunzio, Iacobazzi, Rosa Maria, Cilia, Antonio, Pirona, Lorenza, Ronsisvalle, Simone, Aricò, Giuseppina, Brasili, Livio
Published in European journal of medicinal chemistry (05.01.2017)
Published in European journal of medicinal chemistry (05.01.2017)
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Journal Article
Direct Cu-mediated aromatic 18F-labeling of highly reactive tetrazines for pretargeted bioorthogonal PET imaging
García-Vázquez, Rocío, Battisti, Umberto M, Jørgensen, Jesper T, Shalgunov, Vladimir, Hvass, Lars, Stares, Daniel L, Petersen, Ida N, Crestey, François, Löffler, Andreas, Svatunek, Dennis, Kristensen, Jesper L, Mikula, Hannes, Kjaer, Andreas, Herth, Matthias M
Published in Chemical science (Cambridge) (15.09.2021)
Published in Chemical science (Cambridge) (15.09.2021)
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Journal Article
“Heart-cut” bidimensional achiral-chiral liquid chromatography applied to the evaluation of stereoselective metabolism, in vivo biological activity and brain response to chiral drug candidates targeting the central nervous system
Battisti, Umberto M., Citti, Cinzia, Larini, Martina, Ciccarella, Giuseppe, Stasiak, Natalia, Troisi, Luigino, Braghiroli, Daniela, Parenti, Carlo, Zoli, Michele, Cannazza, Giuseppe
Published in Journal of Chromatography A (22.04.2016)
Published in Journal of Chromatography A (22.04.2016)
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Journal Article
Diastereoselective Synthesis of (1,3-Dioxan-4-yl)pyrimidine and Purin Nucleoside Analogues
Battisti, Umberto M., Sorbi, Claudia, Quotadamo, Antonio, Franchini, Silvia, Tait, Annalisa, Schols, Dominique, Jeong, Lak Shin, Lee, Sang Kook, Song, Jayoung, Brasili, Livio
Published in European journal of organic chemistry (01.02.2015)
Published in European journal of organic chemistry (01.02.2015)
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Journal Article
Synthesis and Structure-Activity Relationships of Triazaspirodecanone Derivatives as Nociceptin/Orphanin FQ Receptor Ligands
Corrado, Sandra, Battisti, Umberto M., Sorbi, Claudia, Tait, Annalisa, Malfacini, Davide, Camarda, Valeria, Calò, Girolamo, Brasili, Livio
Published in Chemical biology & drug design (01.10.2015)
Published in Chemical biology & drug design (01.10.2015)
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Journal Article
Effects of N‑Alkyl-4-Methylamphetamine Optical Isomers on Plasma Membrane Monoamine Transporters and Abuse-Related Behavior
Battisti, Umberto M, Sitta, Ramsey, Harris, Alan, Sakloth, Farhana, Walther, Donna, Ruchala, Iwona, Negus, S. Stevens, Baumann, Michael H, Glennon, Richard A, Eltit, Jose M
Published in ACS chemical neuroscience (18.07.2018)
Published in ACS chemical neuroscience (18.07.2018)
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Journal Article
Synthesis, structural characterization and biological evaluation of 4′-C-methyl- and phenyl-dioxolane pyrimidine and purine nucleosides
Franchini, Silvia, Battisti, Umberto M., Sorbi, Claudia, Tait, Annalisa, Cornia, Andrea, Jeong, Lak Shin, Lee, Sang Kook, Song, Jayoung, Loddo, Roberta, Madeddu, Silvia, Sanna, Giuseppina, Brasili, Livio
Published in Archives of pharmacal research (01.05.2017)
Published in Archives of pharmacal research (01.05.2017)
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Journal Article
Structure–affinity/activity relationships of 1,4-dioxa-spiro[4.5]decane based ligands at α 1 and 5-HT1A receptors
Franchini, Silvia, Battisti, Umberto M., Baraldi, Annamaria, Prandi, Adolfo, Fossa, Paola, Cichero, Elena, Tait, Annalisa, Sorbi, Claudia, Marucci, Gabriella, Cilia, Antonio, Pirona, Lorenza, Brasili, Livio
Published in European journal of medicinal chemistry (24.11.2014)
Published in European journal of medicinal chemistry (24.11.2014)
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Journal Article
Structure-affinity/activity relationships of 1,4-dioxa-spiro[4.5]decane based ligands at α1 and 5-HT1A receptors
Franchini, Silvia, Battisti, Umberto M, Baraldi, Annamaria, Prandi, Adolfo, Fossa, Paola, Cichero, Elena, Tait, Annalisa, Sorbi, Claudia, Marucci, Gabriella, Cilia, Antonio, Pirona, Lorenza, Brasili, Livio
Published in European journal of medicinal chemistry (24.11.2014)
Published in European journal of medicinal chemistry (24.11.2014)
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Journal Article
7‑Chloro-5-(furan-3-yl)-3-methyl‑4H‑benzo[e][1,2,4]thiadiazine 1,1-Dioxide as Positive Allosteric Modulator of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor. The End of the Unsaturated-Inactive Paradigm?
Citti, Cinzia, Battisti, Umberto M, Cannazza, Giuseppe, Jozwiak, Krzysztof, Stasiak, Natalia, Puja, Giulia, Ravazzini, Federica, Ciccarella, Giuseppe, Braghiroli, Daniela, Parenti, Carlo, Troisi, Luigino, Zoli, Michele
Published in ACS chemical neuroscience (17.02.2016)
Published in ACS chemical neuroscience (17.02.2016)
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Journal Article
Regioselective cyclization of chloroacylaminobenzenesulfonamide derivatives
Carrozzo, Marina M., Battisti, Umberto M., Cannazza, Giuseppe, Citti, Cinzia, Parenti, Carlo, Troisi, Luigino
Published in Tetrahedron letters (13.06.2012)
Published in Tetrahedron letters (13.06.2012)
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Journal Article