HIV-1 re-suppression on a first-line regimen despite the presence of phenotypic drug resistance
Basson, Adriaan E, Charalambous, Salome, Hoffmann, Christopher J, Morris, Lynn, Apetrei, Cristian
Published in PloS one (18.06.2020)
Published in PloS one (18.06.2020)
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ω‑Functionalized Lipid Prodrugs of HIV NtRTI Tenofovir with Enhanced Pharmacokinetic Properties
Pribut, Nicole, D’Erasmo, Michael, Dasari, Madhuri, Giesler, Kyle E, Iskandar, Sabrina, Sharma, Savita K, Bartsch, Perry W, Raghuram, Akshay, Bushnev, Anatoliy, Hwang, Soyon S, Burton, Samantha L, Derdeyn, Cynthia A, Basson, Adriaan E, Liotta, Dennis C, Miller, Eric J
Published in Journal of medicinal chemistry (09.09.2021)
Published in Journal of medicinal chemistry (09.09.2021)
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Application of the Huisgen cycloaddition and ‘click’ reaction toward various 1,2,3-triazoles as HIV non-nucleoside reverse transcriptase inhibitors
Pribut, Nicole, Veale, Clinton G.L., Basson, Adriaan E., van Otterlo, Willem A.L., Pelly, Stephen C.
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
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Journal Article
Expanding the toolbox of metabolically stable lipid prodrug strategies
Toti, Kiran S, Pribut, Nicole, D'Erasmo, Michael, Dasari, Madhuri, Sharma, Savita K, Bartsch, Perry W, Burton, Samantha L, Gold, Hannah B, Bushnev, Anatoliy, Derdeyn, Cynthia A, Basson, Adriaan E, Liotta, Dennis C, Miller, Eric J
Published in Frontiers in pharmacology (06.01.2023)
Published in Frontiers in pharmacology (06.01.2023)
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Impact of drug resistance-associated amino acid changes in HIV-1 subtype C on susceptibility to newer nonnucleoside reverse transcriptase inhibitors
Basson, Adriaan E, Rhee, Soo-Yon, Parry, Chris M, El-Khatib, Ziad, Charalambous, Salome, De Oliveira, Tulio, Pillay, Deenan, Hoffmann, Christopher, Katzenstein, David, Shafer, Robert W, Morris, Lynn
Published in Antimicrobial agents and chemotherapy (01.02.2015)
Published in Antimicrobial agents and chemotherapy (01.02.2015)
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Contribution of Gag and Protease to HIV-1 Phenotypic Drug Resistance in Pediatric Patients Failing Protease Inhibitor-Based Therapy
Giandhari, Jennifer, Basson, Adriaan E, Sutherland, Katherine, Parry, Chris M, Cane, Patricia A, Coovadia, Ashraf, Kuhn, Louise, Hunt, Gillian, Morris, Lynn
Published in Antimicrobial agents and chemotherapy (01.04.2016)
Published in Antimicrobial agents and chemotherapy (01.04.2016)
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K103N, V106M and Y188L Significantly Reduce HIV-1 Subtype C Phenotypic Susceptibility to Doravirine
Reddy, Nikita, Papathanasopoulos, Maria, Steegen, Kim, Basson, Adriaan Erasmus
Published in Viruses (20.09.2024)
Published in Viruses (20.09.2024)
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Journal Article
Genetic Changes in HIV-1 Gag-Protease Associated with Protease Inhibitor-Based Therapy Failure in Pediatric Patients
Giandhari, Jennifer, Basson, Adriaan E, Coovadia, Ashraf, Kuhn, Louise, Abrams, Elaine J, Strehlau, Renate, Morris, Lynn, Hunt, Gillian M
Published in AIDS research and human retroviruses (01.08.2015)
Published in AIDS research and human retroviruses (01.08.2015)
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Novel indole based NNRTIs with improved potency against wild type and resistant HIV
Müller, Ronel, Mulani, Iqbal, Basson, Adriaan E., Pribut, Nicole, Hassam, Mohammad, Morris, Lynn, van Otterlo, Willem A.L., Pelly, Stephen C.
Published in Bioorganic & medicinal chemistry letters (15.09.2014)
Published in Bioorganic & medicinal chemistry letters (15.09.2014)
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Antibacterial activities and cytotoxicity of terpenoids isolated from Spirostachys africana
Mathabe, Matlakala Christina, Hussein, Ahmed A., Nikolova, Roumiana V., Basson, Adriaan E., Meyer, J.J. Marion, Lall, Namrita
Published in Journal of ethnopharmacology (28.02.2008)
Published in Journal of ethnopharmacology (28.02.2008)
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Development of phenotypic HIV-1 drug resistance after exposure to single-dose nevirapine
Basson, Adriaan E, Ntsala, Matshediso, Martinson, Neil, Tlale, Emily, Corrigan, Gary E, Shao, Xingwu, Gray, Glenda, McIntyre, James, Puren, Adrian, Morris, Lynn
Published in Journal of acquired immune deficiency syndromes (1999) (01.12.2008)
Published in Journal of acquired immune deficiency syndromes (1999) (01.12.2008)
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Building Metabolically Stable and Potent Anti-HIV Thioether-Lipid Analogues of Tenofovir Exalidex: A thorough Pharmacological Analysis
D'Erasmo, Michael P, Sharma, Savita K, Pribut, Nicole, Basson, Adriaan, Dasari, Madhuri, Bartsch, Perry, Iskandar, Sabrina E, Giesler, Kyle E, Burton, Samantha, Derdeyn, Cindy A, Liotta, Dennis C, Miller, Eric J
Published in Journal of medicinal chemistry (16.10.2024)
Published in Journal of medicinal chemistry (16.10.2024)
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Synthesis of novel pyridine and pyrimidine derivatives as potential inhibitors of HIV-1 reverse transcriptase using palladium-catalysed C-N cross-coupling and nucleophilic aromatic substitution reactions
Changunda, Charles R. K., Rousseau, Amanda L., Basson, Adriaan E., Bode, Moira L.
Published in ARKIVOC free online journal of organic chemistry (30.04.2021)
Published in ARKIVOC free online journal of organic chemistry (30.04.2021)
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