Highly Potent, Selective, and Orally Bioavailable 4‑Thiazol‑N‑(pyridin-2-yl)pyrimidin-2-amine Cyclin-Dependent Kinases 4 and 6 Inhibitors as Anticancer Drug Candidates: Design, Synthesis, and Evaluation
Tadesse, Solomon, Yu, Mingfeng, Mekonnen, Laychiluh B, Lam, Frankie, Islam, Saiful, Tomusange, Khamis, Rahaman, Muhammed H, Noll, Benjamin, Basnet, Sunita K. C, Teo, Theodosia, Albrecht, Hugo, Milne, Robert, Wang, Shudong
Published in Journal of medicinal chemistry (09.03.2017)
Published in Journal of medicinal chemistry (09.03.2017)
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Journal Article
Brassica rapa FLC homologue FLC2 is a key regulator of flowering time, identified through transcriptional co-expression networks
Xiao, Dong, Zhao, Jian J, Hou, Xi L, Basnet, Ram K, Carpio, Dunia P.D, Zhang, Ning W, Bucher, Johan, Lin, Ke, Cheng, Feng, Wang, Xiao W, Bonnema, Guusje
Published in Journal of experimental botany (01.11.2013)
Published in Journal of experimental botany (01.11.2013)
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Journal Article
Discovery of N ,4-Di(1 H -pyrazol-4-yl)pyrimidin-2-amine-Derived CDK2 Inhibitors as Potential Anticancer Agents: Design, Synthesis, and Evaluation
Fanta, Biruk Sintayehu, Lenjisa, Jimma, Teo, Theodosia, Kou, Lianmeng, Mekonnen, Laychiluh, Yang, Yuchao, Basnet, Sunita K C, Hassankhani, Ramin, Sykes, Matthew J, Yu, Mingfeng, Wang, Shudong
Published in Molecules (Basel, Switzerland) (25.03.2023)
Published in Molecules (Basel, Switzerland) (25.03.2023)
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Journal Article
Advanced maternal age may impact placental morphology in IVF pregnancies
Sacha, C.R., Basnet, K., Lee, A.M., James, K., Roberts, D.J.
Published in Fertility and sterility (01.03.2018)
Published in Fertility and sterility (01.03.2018)
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Journal Article
In Search of Novel CDK8 Inhibitors by Virtual Screening
Kumarasiri, Malika, Teo, Theodosia, Yu, Mingfeng, Philip, Stephen, Basnet, Sunita K. C, Albrecht, Hugo, Sykes, Matthew J, Wang, Peng, Wang, Shudong
Published in Journal of chemical information and modeling (27.03.2017)
Published in Journal of chemical information and modeling (27.03.2017)
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Journal Article
Discovery of 5-(2-(Phenylamino)pyrimidin-4-yl)thiazol-2(3H)-one Derivatives as Potent Mnk2 Inhibitors: Synthesis, SAR Analysis and Biological Evaluation
Diab, Sarah, Teo, Theodosia, Kumarasiri, Malika, Li, Peng, Yu, Mingfeng, Lam, Frankie, Basnet, Sunita K. C., Sykes, Matthew J., Albrecht, Hugo, Milne, Robert, Wang, Shudong
Published in ChemMedChem (01.05.2014)
Published in ChemMedChem (01.05.2014)
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Journal Article
An Orally Bioavailable and Highly Efficacious Inhibitor of CDK9/FLT3 for the Treatment of Acute Myeloid Leukemia
Anshabo, Abel Tesfaye, Bantie, Laychiluh, Diab, Sarah, Lenjisa, Jimma, Kebede, Alemwork, Long, Yi, Heinemann, Gary, Karanjia, Jasmine, Noll, Benjamin, Basnet, Sunita K C, Li, Manjun, Milne, Robert, Albrecht, Hugo, Wang, Shudong
Published in Cancers (22.02.2022)
Published in Cancers (22.02.2022)
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Journal Article
Discovery of CDK5 Inhibitors through Structure-Guided Approach
Khair, Nishat Z, Lenjisa, Jimma L, Tadesse, Solomon, Kumarasiri, Malika, Basnet, Sunita K. C, Mekonnen, Laychiluh B, Li, Manjun, Diab, Sarah, Sykes, Matthew J, Albrecht, Hugo, Milne, Robert, Wang, Shudong
Published in ACS medicinal chemistry letters (09.05.2019)
Published in ACS medicinal chemistry letters (09.05.2019)
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Journal Article
Close range photogrammetry for dynamically tracking drifted snow deposition
Basnet, K., Muste, M., Constantinescu, G., Ho, H., Xu, H.
Published in Cold regions science and technology (01.01.2016)
Published in Cold regions science and technology (01.01.2016)
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Journal Article
Quantitative Trait Locus Analysis of Seed Germination and Seedling Vigor in Brassica rapa Reveals QTL Hotspots and Epistatic Interactions
Basnet, Ram K, Duwal, Anita, Tiwari, Dev N, Xiao, Dong, Monakhos, Sokrat, Bucher, Johan, Visser, Richard G F, Groot, Steven P C, Bonnema, Guusje, Maliepaard, Chris
Published in Frontiers in plant science (01.12.2015)
Published in Frontiers in plant science (01.12.2015)
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Journal Article
Unveiling new chemical scaffolds as Mnk inhibitors
Diab, Sarah, Li, Peng, Basnet, Sunita K C, Lu, Jingfeng, Yu, Mingfeng, Albrecht, Hugo, Milne, Robert W, Wang, Shudong
Published in Future medicinal chemistry (01.01.2016)
Published in Future medicinal chemistry (01.01.2016)
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Journal Article
Discovery of N-phenyl-4-(1H-pyrrol-3-yl)pyrimidin-2-amine derivatives as potent Mnk2 inhibitors: design, synthesis, SAR analysis, and evaluation of in vitro anti-leukaemic activity
Abdelaziz, Ahmed M, Diab, Sarah, Islam, Saiful, Basnet, Sunita K C, Noll, Ben, Li, Peng, Mekonnen, Laychiluh B, Lu, Jingfeng, Albrecht, Hugo, Milne, Robert W, Gerber, Cobus, Yu, Mingfeng, Wang, Shudong
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2019)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2019)
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Journal Article
2-Anilino-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine-derived CDK2 inhibitors as anticancer agents: Design, synthesis & evaluation
Fanta, Biruk Sintayehu, Mekonnen, Laychiluh, Basnet, Sunita K.C., Teo, Theodosia, Lenjisa, Jimma, Khair, Nishat Z., Kou, Lianmeng, Tadesse, Solomon, Sykes, Matthew J., Yu, Mingfeng, Wang, Shudong
Published in Bioorganic & medicinal chemistry (15.02.2023)
Published in Bioorganic & medicinal chemistry (15.02.2023)
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Journal Article
Discovery of Potent Inhibitors of Cyclin‐Dependent Kinases 7 and 9: Design, Synthesis, Structure‐Activity Relationship Analysis and Biological Evaluation
Chen, Renjie, Hassankhani, Ramin, Long, Yi, Basnet, Sunita K. C., Teo, Theodosia, Yang, Yuchao, Mekonnen, Laychiluh, Yu, Mingfeng, Wang, Shudong
Published in ChemMedChem (01.02.2023)
Published in ChemMedChem (01.02.2023)
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Journal Article
Synthesis and evaluation of 2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a] pyridine]-1',5'-dione derivatives as Mnk inhibitors
Abdelaziz, Ahmed M., Basnet, Sunita K. C., Islam, Saiful, Li, Manjun, Tadesse, Solomon, Albrecht, Hugo, Gerber, Cobus, Yu, Mingfeng, Wang, Shudong
Published in Bioorganic & medicinal chemistry letters (15.09.2019)
Published in Bioorganic & medicinal chemistry letters (15.09.2019)
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Journal Article
Differential effects of endurance training and weight loss on plasma adiponectin multimers and adipose tissue macrophages in younger, moderately overweight men
Auerbach, Pernille, Nordby, Pernille, Bendtsen, Line Q, Mehlsen, Jesper L, Basnet, Smita K, Vestergaard, Henrik, Ploug, Thorkil, Stallknecht, Bente
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.09.2013)
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.09.2013)
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Journal Article
Pharmacologic Inhibition of MNKs in Acute Myeloid Leukemia
Teo, Theodosia, Lam, Frankie, Yu, Mingfeng, Yang, Yuchao, Basnet, Sunita K C, Albrecht, Hugo, Sykes, Matthew J, Wang, Shudong
Published in Molecular pharmacology (01.08.2015)
Published in Molecular pharmacology (01.08.2015)
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Journal Article
Dual Inhibition of Mnk2 and FLT3 for potential treatment of acute myeloid leukaemia
Diab, Sarah, Abdelaziz, Ahmad M., Li, Peng, Teo, Theodosia, Basnet, Sunita K.C., Noll, Ben, Rahaman, Muhammed H., Lu, Jingfeng, Hou, Jinqiang, Yu, Mingfeng, Le, Bich T., Albrecht, Hugo, Milne, Robert W., Wang, Shudong
Published in European journal of medicinal chemistry (20.10.2017)
Published in European journal of medicinal chemistry (20.10.2017)
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Journal Article
Inhibition of Mnk enhances apoptotic activity of cytarabine in acute myeloid leukemia cells
Li, Peng, Diab, Sarah, Yu, Mingfeng, Adams, Julian, Islam, Saiful, Basnet, Sunita K C, Albrecht, Hugo, Milne, Robert, Wang, Shudong
Published in Oncotarget (30.08.2016)
Published in Oncotarget (30.08.2016)
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Journal Article