Discovery of N-Isoxazolyl Biphenylsulfonamides as Potent Dual Angiotensin II and Endothelin A Receptor Antagonists
Murugesan, Natesan, Tellew, John E, Gu, Zhengxiang, Kunst, Bridgette L, Fadnis, Leena, Cornelius, Lyndon A, Baska, Rose Ann F, Yang, Yifan, Beyer, Sophie M, Monshizadegan, Hossain, Dickinson, Kenneth E, Panchal, Balkrushna, Valentine, Maria T, Chong, Saeho, Morrison, Richard A, Carlson, Kenneth E, Powell, James R, Moreland, Suzanne, Barrish, Joel C, Kowala, Mark C, Macor, John E
Published in Journal of medicinal chemistry (29.08.2002)
Published in Journal of medicinal chemistry (29.08.2002)
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Discovery of 4′-[(Imidazol-1-yl)methyl]biphenyl-2-sulfonamides as dual endothelin/Angiotensin II receptor antagonists
Tellew, John E, Baska, Rose Ann F, Beyer, Sophie M, Carlson, Kenneth E, Cornelius, Lyndon A, Fadnis, Leena, Gu, Zhengxiang, Kunst, Bridgette L, Kowala, Mark C, Monshizadegan, Hossain, Murugesan, Natesan, Ryan, Carol S, Valentine, Maria T, Yang, Yifan, Macor, John E
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
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Dual Angiotensin II and Endothelin A Receptor Antagonists: Synthesis of 2‘-Substituted N-3-Isoxazolyl Biphenylsulfonamides with Improved Potency and Pharmacokinetics
Murugesan, Natesan, Gu, Zhengxiang, Fadnis, Leena, Tellew, John E, Baska, Rose Ann F, Yang, Yifan, Beyer, Sophie M, Monshizadegan, Hossain, Dickinson, Kenneth E, Valentine, Maria T, Humphreys, W. Griffith, Lan, Shih-Jung, Ewing, William R, Carlson, Kenneth E, Kowala, Mark C, Zahler, Robert, Macor, John E
Published in Journal of medicinal chemistry (13.01.2005)
Published in Journal of medicinal chemistry (13.01.2005)
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Novel Dual Action AT1 and ETA Receptor Antagonists Reduce Blood Pressure in Experimental Hypertension
Kowala, Mark C, Murugesan, Natesan, Tellew, John, Carlson, Kenneth, Monshizadegan, Hossain, Ryan, Carol, Gu, Zhengxiang, Kane, Bridgette, Fadnis, Leena, Baska, Rose Ann, Beyer, Sophie, Arthur, Susan, Dickinson, Kenneth, Zhang, Donglu, Perrone, Mark, Ferrer, Pam, Giancarli, Mary, Baumann, Jergen, Bird, Eileen, Panchal, Balkrushna, Yang, Yifan, Trippodo, Nick, Barrish, Joel, Macor, John E
Published in The Journal of pharmacology and experimental therapeutics (01.04.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2004)
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Journal Article
Novel Dual Action AT 1 and ET A Receptor Antagonists Reduce Blood Pressure in Experimental Hypertension
Kowala, Mark C., Murugesan, Natesan, Tellew, John, Carlson, Kenneth, Monshizadegan, Hossain, Ryan, Carol, Gu, Zhengxiang, Kane, Bridgette, Fadnis, Leena, Baska, Rose Ann, Beyer, Sophie, Arthur, Susan, Dickinson, Kenneth, Zhang, Donglu, Perrone, Mark, Ferrer, Pam, Giancarli, Mary, Baumann, Jergen, Bird, Eileen, Panchal, Balkrushna, Yang, Yifan, Trippodo, Nick, Barrish, Joel, Macor, John E.
Published in The Journal of pharmacology and experimental therapeutics (01.04.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2004)
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Identification of [ 3H]P1075 binding sites and P1075-activated K + currents in ovine choroid plexus cells
Dickinson, Kenneth E.J, Baska, Rose Ann, Cohen, Robert B, Bryson, Catherine C, Smith, Mark A, Schroeder, Kirk, Lodge, Nicholas J
Published in European journal of pharmacology (12.03.1998)
Published in European journal of pharmacology (12.03.1998)
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