Discovery of Orally Available and Brain Penetrant AEP Inhibitors
Krummenacher, Daniela, He, Weiping, Kuhn, Bernd, Schnider, Christian, Beurier, Angélica, Brom, Virginie, Sivasothy, Thulase, Marty, Christine, Tosstorff, Andreas, Hewings, David S., Mesch, Stefanie, Pinard, Emmanuel, Brändlin, Mathis, Hochstrasser, Remo, Westwood, Paul, Rothe, Judith, Kronenberger, Alexandra, Morandi, Federica, Gutbier, Simon, Schuler, Angelika, Heer, Dominik, Gloria, Ludivine Esteves, Joedicke, Lisa, Rudolph, Markus G., Müller, Lutz, Grüninger, Fiona, Baumann, Karlheinz, Kaniyappan, Senthilvelrajan, Manevski, Nenad, Bartels, Björn
Published in Journal of medicinal chemistry (28.12.2023)
Published in Journal of medicinal chemistry (28.12.2023)
Get full text
Journal Article
A Streamlined, Safe and Sustainable Process for Gemlapodect
Fantasia, Serena, Bartels, Björn, Bliss, Fritz, Koch, Fritz, Scalone, Michelangelo, Spiess, Daniel, Steiner, Markus, Wang, Shaoning, Püntener, Kurt
Published in Helvetica chimica acta (01.10.2023)
Published in Helvetica chimica acta (01.10.2023)
Get full text
Journal Article
Selective and brain-penetrant HCN1 inhibitors reveal links between synaptic integration, cortical function, and working memory
Harde, Eva, Hierl, Markus, Weber, Michael, Waiz, David, Wyler, Roger, Wach, Jean-Yves, Haab, Rachel, Gundlfinger, Anja, He, Weiping, Schnider, Patrick, Paina, Manuel, Rolland, Jean-Francois, Greiter-Wilke, Andrea, Gasser, Rodolfo, Reutlinger, Michael, Dupont, Amanda, Roberts, Sonia, O'Connor, Eoin C., Bartels, Björn, Hall, Benjamin J.
Published in Cell chemical biology (21.03.2024)
Published in Cell chemical biology (21.03.2024)
Get full text
Journal Article
Formal Modeling and Verification of Low-Level Software Programs
Bartels, Björn, Glesner, Sabine
Published in 2010 10th International Conference on Quality Software (01.07.2010)
Published in 2010 10th International Conference on Quality Software (01.07.2010)
Get full text
Conference Proceeding
SYNTHESIS OF TRANS-8-CHLORO-5-METHYL-1 -[4-(PYRIDIN-2-YLOXY)-CYCLOHEXYL]-5,6-DIHYDRO-4H-2,3,5,10B-TETRAAZA-BENZO[E]AZULENE AND CRYTALLINE FORMS THEREOF
Ran, Frederic, Diodone, Ralph, Bartels, Bjorn, Pfleger, Christophe, Trussardi, Rene, Rothenhaeusler, Benno, Grassmann, Olaf, Hartung, Thomas, Schwitter, Urs, Hoffmann-Emery, Fabienne, Adam, Jean-Michel
Year of Publication 16.09.2021
Get full text
Year of Publication 16.09.2021
Patent
Synthesis of trans-8-chloro-5-methyl-1-[4-(pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4H-2,3,5,10B-tetraaza-benzo[e]azulene and crytalline forms thereof
Ran, Frederic, Diodone, Ralph, Bartels, Bjorn, Pfleger, Christophe, Trussardi, Rene, Rothenhaeusler, Benno, Grassmann, Olaf, Hartung, Thomas, Schwitter, Urs, Hoffmann-Emery, Fabienne, Adam, Jean-Michel
Year of Publication 22.06.2021
Get full text
Year of Publication 22.06.2021
Patent
SYNTHESIS OF TRANS-8-CHLORO-5-METHYL-1 -[4-(PYRIDIN-2-YLOXY)-CYCLOHEXYL]-5,6-DIHYDRO-4H-2,3,5,10B-TETRAAZA-BENZO[E]AZULENE AND CRYTALLINE FORMS THEREOF
Ran, Frederic, Diodone, Ralph, Bartels, Bjorn, Pfleger, Christophe, Trussardi, Rene, Rothenhaeusler, Benno, Grassmann, Olaf, Hartung, Thomas, Schwitter, Urs, Hoffmann-Emery, Fabienne, Adam, Jean-Michel
Year of Publication 27.06.2019
Get full text
Year of Publication 27.06.2019
Patent
Synthesis of trans-8-chloro-5-methyl-1-[4-(pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4H-2,3,5,10B-tetraaza-benzo[E]azulene and crytalline forms thereof
Ran, Frederic, Diodone, Ralph, Bartels, Bjorn, Pfleger, Christophe, Trussardi, Rene, Rothenhaeusler, Benno, Grassmann, Olaf, Hartung, Thomas, Schwitter, Urs, Hoffmann-Emery, Fabienne, Adam, Jean-Michel
Year of Publication 02.04.2019
Get full text
Year of Publication 02.04.2019
Patent
Verification of Distributed Embedded Real-Time Systems and their Low-Level Implementations Using Timed CSP
Bartels, B., Glesner, S.
Published in 2011 18th Asia-Pacific Software Engineering Conference (01.12.2011)
Published in 2011 18th Asia-Pacific Software Engineering Conference (01.12.2011)
Get full text
Conference Proceeding
SYNTHESIS OF TRANS-8-CHLORO-5-METHYL-1 -[4-(PYRIDIN-2-YLOXY)-CYCLOHEXYL]-5,6-DIHYDRO-4H-2,3,5,10B-TETRAAZA-BENZO[E]AZULENE AND CRYTALLINE FORMS THEREOF
Diodone Ralph, Trussardi Rene, Schwitter Urs, Rothenhaeusler Benno, Hartung Thomas, Pfleger Christophe, Bartels Bjorn, Hoffmann-Emery Fabienne, Ran Frederic, Adam Jean-Michel, Grassmann Olaf
Year of Publication 29.09.2016
Get full text
Year of Publication 29.09.2016
Patent