Chemical genetic inhibition of DEAD-box proteins using covalent complementarity
Barkovich, Krister J, Moore, Megan K, Hu, Qi, Shokat, Kevan M
Published in Nucleic acids research (28.09.2018)
Published in Nucleic acids research (28.09.2018)
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Journal Article
Analog sensitive chemical inhibition of the DEAD‐box protein DDX3
Floor, Stephen N., Barkovich, Krister J., Condon, Kendall J., Shokat, Kevan M., Doudna, Jennifer A.
Published in Protein science (01.03.2016)
Published in Protein science (01.03.2016)
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Journal Article
Kinetics of inhibitor cycling underlie therapeutic disparities between EGFR-driven lung and brain cancers
Barkovich, Krister J, Hariono, Sujatmi, Garske, Adam L, Zhang, Jie, Blair, Jimmy A, Fan, Qi-Wen, Shokat, Kevan M, Nicolaides, Theodore, Weiss, William A
Published in Cancer discovery (01.05.2012)
Published in Cancer discovery (01.05.2012)
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Journal Article
p27 allosterically activates cyclin-dependent kinase 4 and antagonizes palbociclib inhibition
Guiley, Keelan Z, Stevenson, Jack W, Lou, Kevin, Barkovich, Krister J, Kumarasamy, Vishnu, Wijeratne, Tilini U, Bunch, Katharine L, Tripathi, Sarvind, Knudsen, Erik S, Witkiewicz, Agnieszka K, Shokat, Kevan M, Rubin, Seth M
Published in Science (American Association for the Advancement of Science) (13.12.2019)
Published in Science (American Association for the Advancement of Science) (13.12.2019)
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Journal Article
Physalis Mottle Virus-Like Nanocarriers with Expanded Internal Loading Capacity
Barkovich, Krister J., Wu, Zhuohong, Zhao, Zhongchao, Simms, Andrea, Chang, Eric Y., Steinmetz, Nicole F.
Published in Bioconjugate chemistry (20.09.2023)
Published in Bioconjugate chemistry (20.09.2023)
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Journal Article
Virus-like Particles Armored by an Endoskeleton
Wu, Zhuohong, Bayón, Jorge L., Kouznetsova, Tatiana B., Ouchi, Tetsu, Barkovich, Krister J., Hsu, Sean K., Craig, Stephen L., Steinmetz, Nicole F.
Published in Nano letters (13.03.2024)
Published in Nano letters (13.03.2024)
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Journal Article
Type II Kinase Inhibitors Targeting Cys-Gatekeeper Kinases Display Orthogonality with Wild Type and Ala/Gly-Gatekeeper Kinases
Ocasio, Cory A, Warkentin, Alexander A, McIntyre, Patrick J, Barkovich, Krister J, Vesely, Clare, Spencer, John, Shokat, Kevan M, Bayliss, Richard
Published in ACS chemical biology (19.10.2018)
Published in ACS chemical biology (19.10.2018)
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Journal Article
Analog sensitive chemical inhibition of the DEAD ‐box protein DDX 3
Floor, Stephen N., Barkovich, Krister J., Condon, Kendall J., Shokat, Kevan M., Doudna, Jennifer A.
Published in Protein science (01.03.2016)
Published in Protein science (01.03.2016)
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Journal Article
Combined BRAF^sup V600E^ and MEK blockade for BRAF^sup V600E^-mutant gliomas
Zhang, Jie, Yao, Tsun-wen, Hashizume, Rintaro, Hariono, Sujatmi, Barkovich, Krister J, Fan, Qi-wen, Prados, Michael, James, C David, Weiss, William A, Nicolaides, Theodore
Published in Journal of neuro-oncology (01.02.2017)
Published in Journal of neuro-oncology (01.02.2017)
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Journal Article
Combined BRAF super(V600E) and MEK blockade for BRAF super(V600E)-mutant gliomas
Zhang, Jie, Yao, Tsun-Wen, Hashizume, Rintaro, Hariono, Sujatmi, Barkovich, Krister J, Fan, Qi-Wen, Prados, Michael, James, CDavid, Weiss, William A, Nicolaides, Theodore
Published in Journal of neuro-oncology (01.02.2017)
Published in Journal of neuro-oncology (01.02.2017)
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Journal Article
Abstract 2314: Erlotinib response in lung- and glioma-derived EGFR alleles: Correlating kinase site occupancy with efficacy
Barkovich, Krister J., Nicolaides, Theodore, Hariono, Sujatmi, Garske, Adam, Fan, Qi Wen, Shokat, Kevan, Weiss, William A.
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Journal Article
Combined BRAF V600E and MEK blockade for BRAF V600E -mutant gliomas
Zhang, Jie, Yao, Tsun-Wen, Hashizume, Rintaro, Hariono, Sujatmi, Barkovich, Krister J, Fan, Qi-Wen, Prados, Michael, James, C David, Weiss, William A, Nicolaides, Theodore
Published in Journal of neuro-oncology (01.02.2017)
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Published in Journal of neuro-oncology (01.02.2017)
Journal Article