Autoradiographic localization of 5-HT1A receptors in the post-mortem human brain using [3H]WAY-100635 and [11C]way-100635
Hall, H, Lundkvist, C, Halldin, C, Farde, L, Pike, V W, McCarron, J A, Fletcher, A, Cliffe, I A, Barf, T, Wikström, H, Sedvall, G
Published in Brain research (16.01.1997)
Published in Brain research (16.01.1997)
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5-HT1D Receptor Agonist Properties of Novel 2-[5-[[(Trifluoromethyl)sulfonyl]oxy]indolyl]ethylamines and Their Use as Synthetic Intermediates
Barf, Tjeerd A, de Boer, Peter, Wikström, Håkan, Peroutka, Stephen J, Svensson, Kjell, Ennis, Michael D, Ghazal, Nabil B, McGuire, James C, Smith, Martin W
Published in Journal of medicinal chemistry (22.11.1996)
Published in Journal of medicinal chemistry (22.11.1996)
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Arylsulfonamidothiazoles as a New Class of Potential Antidiabetic Drugs. Discovery of Potent and Selective Inhibitors of the 11β-Hydroxysteroid Dehydrogenase Type 1
Barf, Tjeerd, Vallgårda, Jerk, Emond, Rikard, Häggström, Charlotta, Kurz, Guido, Nygren, Alf, Larwood, Vivienne, Mosialou, Erifili, Axelsson, Kent, Olsson, Rolf, Engblom, Lars, Edling, Naimie, Rönquist-Nii, Yuko, Öhman, Birgitta, Alberts, Peteris, Abrahmsén, Lars
Published in Journal of medicinal chemistry (29.08.2002)
Published in Journal of medicinal chemistry (29.08.2002)
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Substituted benzylamino-6-(trifluoromethyl)pyrimidin-4(1 H)-ones: a novel class of selective human A-FABP inhibitors
Ringom, Rune, Axen, Eva, Uppenberg, Jonas, Lundbäck, Thomas, Rondahl, Lena, Barf, Tjeerd
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
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Discovery of inhibitors of human adipocyte fatty acid-binding protein, a potential type 2 diabetes target
Lehmann, Fredik, Haile, Saba, Axen, Eva, Medina, Carmen, Uppenberg, Jonas, Svensson, Stefan, Lundbäck, Thomas, Rondahl, Lena, Barf, Tjeerd
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
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Active site variability of type 1 11β-hydroxysteroid dehydrogenase revealed by selective inhibitors and cross-species comparisons
Hult, Malin, Shafqat, Naeem, Elleby, Björn, Mitschke, Doreen, Svensson, Stefan, Forsgren, Margareta, Barf, Tjeerd, Vallgårda, Jerk, Abrahmsen, Lars, Oppermann, Udo
Published in Molecular and cellular endocrinology (27.03.2006)
Published in Molecular and cellular endocrinology (27.03.2006)
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Synthesis and Biological Activity of a Novel Class of Small Molecular Weight Peptidomimetic Competitive Inhibitors of Protein Tyrosine Phosphatase 1B
Larsen, Scott D, Barf, Tjeerd, Liljebris, Charlotta, May, Paul D, Ogg, Derek, O'Sullivan, Theresa J, Palazuk, Barbara J, Schostarez, Heinrich J, Stevens, F. Craig, Bleasdale, John E
Published in Journal of medicinal chemistry (31.01.2002)
Published in Journal of medicinal chemistry (31.01.2002)
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Active site variability of type 1 11beta-hydroxysteroid dehydrogenase revealed by selective inhibitors and cross-species comparisons
Hult, Malin, Shafqat, Naeem, Elleby, Björn, Mitschke, Doreen, Svensson, Stefan, Forsgren, Margareta, Barf, Tjeerd, Vallgårda, Jerk, Abrahmsen, Lars, Oppermann, Udo
Published in Molecular and cellular endocrinology (27.03.2006)
Published in Molecular and cellular endocrinology (27.03.2006)
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Characterization of the radioactive metabolites of the 5-HT1A receptor radioligand, [O-methyl-11C]WAY-100635, in monkey and human plasma by HPLC : Comparison of the behaviour of an identified radioactive metabolite with parent radioligand in monkey using PET
OSMAN, S, LUNDKVIST, C, WIKSTRÖM, H, BARF, T, CLIFFE, I. A, FLETCHER, A, FARDE, L, PIKE, V. W, HALLDIN, C, MCCARRON, J. A, SWAHN, C.-G, GINOVART, N, LUTHRA, S. K, BENCH, C. J, GRASBY, P. M
Published in Nuclear medicine and biology (01.07.1996)
Published in Nuclear medicine and biology (01.07.1996)
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5-(Sulfonyl)oxy-tryptamines and ethylamino side chain restricted derivatives. Structure-affinity relationships for h5-HT1B and h5-HT1D receptors
Barf, T, Wikström, H, Pauwels, P J, Palmier, C, Tardif, S, Lundmark, M, Sundell, S
Published in Bioorganic & medicinal chemistry (01.09.1998)
Published in Bioorganic & medicinal chemistry (01.09.1998)
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SYNTHESIS AND EVALUATION OF PHARMACOLOGICAL AND PHARMACOKINETIC PROPERTIES OF MONOPROPYL ANALOGS OF 5-[[(TRIFLUOROMETHYL)SULFONYL]OXY]-2-AMINOTETRALIN, 7-[[(TRIFLUOROMETHYL)SULFONYL]OXY]-2-AMINOTETRALIN, AND 8-[[(TRIFLUOROMETHYL)SULFONYL]OXY]-2-AMINOTETRALIN - CENTRAL DOPAMINE AND SEROTONIN RECEPTOR ACTIVITY
SONESSON, C, BARF, T, NILSSON, J, DIJKSTRA, D, CARLSSON, A, SVENSSON, K, SMITH, MW, MARTIN, IJ, DUNCAN, JN, KING, LJ, WIKSTROM, H
Published in Journal of medicinal chemistry (14.04.1995)
Published in Journal of medicinal chemistry (14.04.1995)
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Potential anxiolytic properties of R-(+)-8-OSO2CF3-PAT, a 5-HT 1A receptor agonist
Barf, T, Korte, S M, Korte-Bouws, G, Sonesson, C, Damsma, G, Bohus, B, Wikström, H
Published in European journal of pharmacology (22.02.1996)
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Published in European journal of pharmacology (22.02.1996)
Journal Article
Potential anxiolytic properties of R-(+)-8-OSO sub(2)CF sub(3)-PAT, a 5-HT sub(1A) receptor agonist
Barf, T, Korte, S M, Korte-Bouws, G, Sonesson, C, Damsma, G, Bohus, B, Wikstroem, H
Published in European journal of pharmacology (01.02.1996)
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Published in European journal of pharmacology (01.02.1996)
Journal Article
Potential anxiolytic properties of R-(+)-8-OSO2CF3-PAT, a 5-HT1A receptor agonist
BARF, T, KORTE, S. M, KORTE-BOWS, G, SONESSON, C, DAMSMA, G, BOHUS, B, WIKSTRÖM, H
Published in European journal of pharmacology (22.02.1996)
Published in European journal of pharmacology (22.02.1996)
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Journal Article
Autoradiographic localization of 5-HT 1A receptors in the post-mortem human brain using [ 3H]WAY-100635 and [ 11C]WAY-100635
Hall, H, Lundkvist, C, Halldin, C, Farde, L, Pike, V.W, McCarron, J.A, Fletcher, A, Cliffe, I.A, Barf, T, Wikström, H, Sedvall, G
Published in Brain research (1997)
Published in Brain research (1997)
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Journal Article
Autoradiographic localization of 5-HT sub(1A) receptors in the post-mortem human brain using [ super(3)H]WAY-100635 and [ super(11)C]WAY-100635
Hall, H, Lundkvist, C, Halldin, C, Farde, L, Pike, V W, McCarron, JA, Fletcher, A, Cliffe, IA, Barf, T, Wikstrom, H, Sedvall, G
Published in Brain research (01.01.1997)
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Published in Brain research (01.01.1997)
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Investigations with GMC2021 in experimental models predictive of antimigraine activity and coronary side-effect potential
Saxena, Pramod R., De Vries, Peter, Heiligers, Jan P.C., VanDenBrink, Antoinette Maassen, Bax, Willem A., Barf, Tjeerd, Wikström, Håkan
Published in European journal of pharmacology (19.09.1996)
Published in European journal of pharmacology (19.09.1996)
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Synthesis and Evaluation of Pharmacological and Pharmacokinetic Properties of Monopropyl Analogs of 5-, 7-, and 8-[[(Trifluoromethyl)sulfonyl]oxy]-2-aminotetralins: Central Dopamine and Serotonin Receptor Activity
Sonesson, Clas, Barf, Tjeerd, Nilsson, Jonas, Dijkstra, Durk, Carlsson, Arvid, Svensson, Kjell, Smith, Martin W, Martin, Iain J, Duncan, J. Neil
Published in Journal of medicinal chemistry (01.04.1995)
Published in Journal of medicinal chemistry (01.04.1995)
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