Imaging Mutant Huntingtin Aggregates: Development of a Potential PET Ligand
Liu, Longbin, Prime, Michael E, Lee, Matt R, Khetarpal, Vinod, Brown, Christopher J, Johnson, Peter D, Miranda-Azpiazu, Patricia, Chen, Xuemei, Clark-Frew, Daniel, Coe, Samuel, Davis, Randall, Dickie, Anthony, Ebneth, Andreas, Esposito, Simone, Gadouleau, Elise, Gai, Xinjie, Galan, Sebastien, Green, Samantha, Greenaway, Catherine, Giles, Paul, Halldin, Christer, Hayes, Sarah, Herbst, Todd, Herrmann, Frank, Heßmann, Manuela, Jia, Zhisheng, Kiselyov, Alexander, Kotey, Adrian, Krulle, Thomas, Mangette, John E, Marston, Richard W, Menta, Sergio, Mills, Matthew R, Monteagudo, Edith, Nag, Sangram, Nibbio, Martina, Orsatti, Laura, Schaertl, Sabine, Scheich, Christoph, Sproston, Joanne, Stepanov, Vladimir, Svedberg, Marie, Takano, Akihiro, Taylor, Malcolm, Thomas, Wayne, Toth, Miklós, Vaidya, Darshan, Vanräs, Katarina, Weddell, Derek, Wigginton, Ian, Wityak, John, Mrzljak, Ladislav, Munoz-Sanjuan, Ignacio, Bard, Jonathan A, Dominguez, Celia
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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[C-11]CHDI-626, a PET Tracer Candidate for Imaging Mutant Huntingtin Aggregates with Reduced Binding to AD Pathological Proteins
Liu, Longbin, Johnson, Peter D., Prime, Michael E., Khetarpal, Vinod, Lee, Matthew R., Brown, Christopher J., Chen, Xuemei, Clark-Frew, Daniel, Coe, Samuel, Conlon, Mike, Davis, Randall, Ensor, Samantha, Esposito, Simone, Moren, Anton Forsberg, Gai, Xinjie, Green, Samantha, Greenaway, Catherine, Haber, James, Halldin, Christer, Hayes, Sarah, Herbst, Todd, Herrmann, Frank, He-mann, Manuela, Hsai, Ming Min, Kotey, Adrian, Mangette, John E., Mills, Matthew R., Monteagudo, Edith, Nag, Sangram, Nibbio, Martina, Orsatti, Laura, Schaertl, Sabine, Scheich, Christoph, Sproston, Joanne, Stepanov, Vladimir, Varnas, Katarina, Varrone, Andrea, Wityak, John, Mrzljak, Ladislav, Munoz-Sanjuan, Ignacio, Bard, Jonathan A., Dominguez, Celia
Published in Journal of medicinal chemistry (26.08.2021)
Published in Journal of medicinal chemistry (26.08.2021)
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Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase
BARD, J. A, ZGOMBICK, J, ADHAM, N, VAYSSE, P, BRANCHEK, T. A, WEINSHANK, R. L
Published in The Journal of biological chemistry (05.11.1993)
Published in The Journal of biological chemistry (05.11.1993)
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Cloning and characterization of the guinea pig 5-HT1F receptor subtype: a comparison of the pharmacological profile to the human species homolog
Adham, N, Bard, J A, Zgombick, J M, Durkin, M M, Kucharewicz, S, Weinshank, R L, Branchek, T A
Published in Neuropharmacology (01.04.1997)
Published in Neuropharmacology (01.04.1997)
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Molecular cloning and pharmacological characterization of guinea pig 5-HT1B and 5-HT1D receptors
Zgombick, J M, Bard, J A, Kucharewicz, S A, Urquhart, D A, Weinshank, R L, Branchek, T A
Published in Neuropharmacology (01.04.1997)
Published in Neuropharmacology (01.04.1997)
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Differences in ligand binding profiles between cloned rabbit and human 5-HT1D alpha and 5-HT1D beta receptors: ketanserin and methiothepin distinguish rabbit 5-HT1D receptor subtypes
Bard, J A, Kucharewicz, S A, Zgombick, J M, Weinshank, R L, Branchek, T A, Cohen, M L
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.08.1996)
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Published in Naunyn-Schmiedeberg's archives of pharmacology (01.08.1996)
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Cloning and characterization of the guinea pig 5-HT sub(1F) receptor subtype: A comparison of the pharmacological profile to the human species homolog
Adham, N, Bard, JA, Zgombick, J M, Durkin, M M, Kucharewicz, S, Weinshank, R L, Branchek, T A
Published in Neuropharmacology (01.05.1997)
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Published in Neuropharmacology (01.05.1997)
Journal Article
Molecular cloning and pharmacological characterization of guinea pig 5-HT sub(1B) and 5-HT sub(1D) receptors
Zgombick, J M, Bard, JA, Kucharewicz, SA, Urquhart, DA, Weinshank, R L, Branchek, T A
Published in Neuropharmacology (01.05.1997)
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Published in Neuropharmacology (01.05.1997)
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The human serotonin 5-hydroxytryptamine sub(1D) receptor pseudogene is transcribed
Bard, JA, Nawoschik, S P, O'Dowd, B F, George, SR, Branchek, T A, Weinshank, R L
Published in Gene (01.01.1995)
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Published in Gene (01.01.1995)
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The 5-HT sub(4) receptor: Molecular cloning and pharmacological characterization of two splice variants
Gerald, C, Adham, N, Kao, Hung-Teh, Olsen, MA, Laz, T M, Schechter, LE, Bard, JA, Vaysse, PJ-J, Hartig, PR, Branchek, T A, Weinshank, R L
Published in The EMBO journal (01.01.1995)
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Published in The EMBO journal (01.01.1995)
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The rat homologue of the bovine alpha sub(1C)-adrenergic receptor shows the pharmacological properties of the classical alpha sub(1A) subtype
Laz, T M, ray, C, Smith, KE, Bard, JA, Vaysse, PJ-J, Branchek, T A, Weinshank, R L
Published in Molecular pharmacology (01.01.1994)
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Published in Molecular pharmacology (01.01.1994)
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The alpha sub(1)-adrenergic receptor that mediates smooth muscle contraction in human prostate has the pharmacological properties of the cloned human alpha sub(1c) subtype
ray, C, Bard, JA, Wetzel, J M, Chiu, G, Shapiro, E, Tang, R, Lepor, H, Hartig, PR, Weinshank, R L
Published in Molecular pharmacology (01.01.1994)
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Published in Molecular pharmacology (01.01.1994)
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