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Published in Scientific reports (01.08.2017)
Published in Scientific reports (01.08.2017)
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Structure-activity relationships of natural and non-natural amino acid-based amide and 2-oxoamide inhibitors of human phospholipase A2 enzymes
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Published in Bioorganic & medicinal chemistry (15.12.2008)
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Enzymatic Removal of Carboxyl Protecting Groups. 2. Cleavage of the Benzyl and Methyl Moieties
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Published in Journal of organic chemistry (28.10.2005)
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Autotaxin inhibitors: a patent review
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Published in Expert opinion on therapeutic patents (01.09.2013)
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Development of Potent and Selective Inhibitors for Group VIA Calcium-Independent Phospholipase A(2) Guided by Molecular Dynamics and Structure-Activity Relationships
Mouchlis, Varnavas D., Limnios, Dimitris, Kokotou, Maroula G., Barbayianni, Efrosini, Kokotos, George, McCammon, J. Andrew, Dennis, Edward A.
Published in Journal of medicinal chemistry (12.05.2016)
Published in Journal of medicinal chemistry (12.05.2016)
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Development of a potent 2-oxoamide inhibitor of secreted phospholipase A(2) guided by molecular docking calculations and molecular dynamics simulations
Vasilakaki, Sofia, Barbayianni, Efrosini, Leonis, Georgios, Papadopoulos, Manthos G., Mavromoustakos, Thomas, Gelb, Michael H., Kokotos, George
Published in Bioorganic & medicinal chemistry (15.04.2016)
Published in Bioorganic & medicinal chemistry (15.04.2016)
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Inhibitors of secreted phospholipase A(2) suppress the release of PGE(2) in renal mesangial cells
Vasilakaki, Sofia, Barbayianni, Efrosini, Magrioti, Victoria, Pastukhov, Oleksandr, Constantinou-Kokotou, Violetta, Huwiler, Andrea, Kokotos, George
Published in Bioorganic & medicinal chemistry (01.07.2016)
Published in Bioorganic & medicinal chemistry (01.07.2016)
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Development of Potent and Selective Inhibitors for Group VIA Calcium-Independent Phospholipase A2 Guided by Molecular Dynamics and Structure–Activity Relationships
Mouchlis, Varnavas D, Limnios, Dimitris, Kokotou, Maroula G, Barbayianni, Efrosini, Kokotos, George, McCammon, J. Andrew, Dennis, Edward A
Published in Journal of medicinal chemistry (12.05.2016)
Published in Journal of medicinal chemistry (12.05.2016)
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Inhibition of Group IVA Cytosolic Phospholipase A(2) by Thiazolyl Ketones in Vitro, ex Vivo, and in Vivo
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Published in Journal of medicinal chemistry (25.09.2014)
Published in Journal of medicinal chemistry (25.09.2014)
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Inhibitors of secreted phospholipase A2 suppress the release of PGE2 in renal mesangial cells
Vasilakaki, Sofia, Barbayianni, Efrosini, Magrioti, Victoria, Pastukhov, Oleksandr, Constantinou-Kokotou, Violetta, Huwiler, Andrea, Kokotos, George
Published in Bioorganic & medicinal chemistry (01.07.2016)
Published in Bioorganic & medicinal chemistry (01.07.2016)
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Development of a potent 2-oxoamide inhibitor of secreted phospholipase A2 guided by molecular docking calculations and molecular dynamics simulations
Vasilakaki, Sofia, Barbayianni, Efrosini, Leonis, Georgios, Papadopoulos, Manthos G., Mavromoustakos, Thomas, Gelb, Michael H., Kokotos, George
Published in Bioorganic & medicinal chemistry (15.04.2016)
Published in Bioorganic & medicinal chemistry (15.04.2016)
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2-Oxoamide inhibitors of cytosolic group IVA phospholipase A(2) with reduced lipophilicity
Antonopoulou, Georgia, Magrioti, Victoria, Kokotou, Maroula G., Nikolaou, Aikaterini, Barbayianni, Efrosini, Mouchlis, Varnavas D., Dennis, Edward A., Kokotos, George
Published in Bioorganic & medicinal chemistry (01.10.2016)
Published in Bioorganic & medicinal chemistry (01.10.2016)
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2-Oxoamides based on dipeptides as selective calcium-independent phospholipase A(2) inhibitors
Smyrniotou, Anneta, Kokotou, Maroula G., Mouchlis, Varnavas D., Barbayianni, Efrosini, Kokotos, George, Dennis, Edward A., Constantinou-Kokotou, Violetta
Published in Bioorganic & medicinal chemistry (01.02.2017)
Published in Bioorganic & medicinal chemistry (01.02.2017)
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Inhibitors of secreted phospholipase A 2 suppress the release of PGE 2 in renal mesangial cells
Vasilakaki, Sofia, Barbayianni, Efrosini, Magrioti, Victoria, Pastukhov, Oleksandr, Constantinou-Kokotou, Violetta, Huwiler, Andrea, Kokotos, George
Published in Bioorganic & medicinal chemistry (01.07.2016)
Published in Bioorganic & medicinal chemistry (01.07.2016)
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Development of Potent and Selective Inhibitors for Group VIA Calcium-Independent Phospholipase A 2 Guided by Molecular Dynamics and Structure–Activity Relationships
Mouchlis, Varnavas D., Limnios, Dimitris, Kokotou, Maroula G., Barbayianni, Efrosini, Kokotos, George, McCammon, J. Andrew, Dennis, Edward A.
Published in Journal of medicinal chemistry (12.05.2016)
Published in Journal of medicinal chemistry (12.05.2016)
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2-Oxoamides based on dipeptides as selective calcium-independent phospholipase A2 inhibitors
Smyrniotou, Anneta, Kokotou, Maroula G., Mouchlis, Varnavas D., Barbayianni, Efrosini, Kokotos, George, Dennis, Edward A., Constantinou-Kokotou, Violetta
Published in Bioorganic & medicinal chemistry (01.02.2017)
Published in Bioorganic & medicinal chemistry (01.02.2017)
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Journal Article
2-Oxoamides based on dipeptides as selective calcium-independent phospholipase A 2 inhibitors
Smyrniotou, Anneta, Kokotou, Maroula G, Mouchlis, Varnavas D, Barbayianni, Efrosini, Kokotos, George, Dennis, Edward A, Constantinou-Kokotou, Violetta
Published in Bioorganic & medicinal chemistry (01.02.2017)
Published in Bioorganic & medicinal chemistry (01.02.2017)
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