Exploring the Chemical Space of Benzothiazole-Based DNA Gyrase B Inhibitors
Skok, Žiga, Barančoková, Michaela, Benek, Ondřej, Cruz, Cristina Durante, Tammela, Päivi, Tomašič, Tihomir, Zidar, Nace, Mašič, Lucija Peterlin, Zega, Anamarija, Stevenson, Clare E. M, Mundy, Julia E. A, Lawson, David M, Maxwell, Anthony, Kikelj, Danijel, Ilaš, Janez
Published in ACS medicinal chemistry letters (10.12.2020)
Published in ACS medicinal chemistry letters (10.12.2020)
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Journal Article
Discovery of Benzothiazole Scaffold-Based DNA Gyrase B Inhibitors
Gjorgjieva, Marina, Tomašič, Tihomir, Barančokova, Michaela, Katsamakas, Sotirios, Ilaš, Janez, Tammela, Päivi, Peterlin Mašič, Lucija, Kikelj, Danijel
Published in Journal of medicinal chemistry (13.10.2016)
Published in Journal of medicinal chemistry (13.10.2016)
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Journal Article
Recent progress in the discovery and development of DNA gyrase B inhibitors
Baran oková, Michaela, Kikelj, Danijel, Ilaš, Janez
Published in Future medicinal chemistry (01.05.2018)
Published in Future medicinal chemistry (01.05.2018)
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Journal Article
Design, synthesis and biological evaluation of 4,5-dibromo-N-(thiazol-2-yl)-1H-pyrrole-2-carboxamide derivatives as novel DNA gyrase inhibitors
Tomašič, Tihomir, Mirt, Matic, Barančoková, Michaela, Ilaš, Janez, Zidar, Nace, Tammela, Päivi, Kikelj, Danijel
Published in Bioorganic & medicinal chemistry (01.01.2017)
Published in Bioorganic & medicinal chemistry (01.01.2017)
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Journal Article
Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors
Jakopin, Žiga, Ilaš, Janez, Barančoková, Michaela, Brvar, Matjaž, Tammela, Päivi, Sollner Dolenc, Marija, Tomašič, Tihomir, Kikelj, Danijel
Published in European journal of medicinal chemistry (21.04.2017)
Published in European journal of medicinal chemistry (21.04.2017)
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Journal Article
Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floor: A medicinal chemistry and QTAIM study
Zidar, Nace, Emanuel Cotman, Andrej, Sinnige, Wessel, Benek, Ondrej, Barančokova, Michaela, Zega, Anamarija, Peterlin Mašič, Lucija, Tomašič, Tihomir, Ilaš, Janez, Henderson, Sara R., Mundy, Julia E.A., Maxwell, Anthony, Stevenson, Clare E.M., Lawson, David M., Jan Sterk, Geert, Tosso, Rodrigo, Gutierrez, Lucas, Enriz, Ricardo D., Kikelj, Danijel
Published in Bioorganic & medicinal chemistry (15.07.2024)
Published in Bioorganic & medicinal chemistry (15.07.2024)
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Journal Article
Design, synthesis, and biological evaluation of 1‐ethyl‐3‐(thiazol‐2‐yl)urea derivatives as Escherichia coli DNA gyrase inhibitors
Tomašič, Tihomir, Barančoková, Michaela, Zidar, Nace, Ilaš, Janez, Tammela, Päivi, Kikelj, Danijel
Published in Archiv der Pharmazie (Weinheim) (01.01.2018)
Published in Archiv der Pharmazie (Weinheim) (01.01.2018)
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Journal Article
A New Cell‐Based AI‐2‐Mediated Quorum Sensing Interference Assay in Screening of LsrK‐Targeted Inhibitors
Gatta, Viviana, Tomašič, Tihomir, Ilaš, Janez, Zidar, Nace, Peterlin Mašič, Lucija, Barančoková, Michaela, Frlan, Rok, Anderluh, Marko, Kikelj, Danijel, Tammela, Päivi
Published in Chembiochem : a European journal of chemical biology (01.07.2020)
Published in Chembiochem : a European journal of chemical biology (01.07.2020)
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Journal Article
Discovery of new ATP-competitive inhibitors of human DNA topoisomerase IIα through screening of bacterial topoisomerase inhibitors
Skok, Žiga, Durcik, Martina, Gramec Skledar, Darja, Barančoková, Michaela, Peterlin Mašič, Lucija, Tomašič, Tihomir, Zega, Anamarija, Kikelj, Danijel, Zidar, Nace, Ilaš, Janez
Published in Bioorganic chemistry (01.09.2020)
Published in Bioorganic chemistry (01.09.2020)
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Journal Article
Design, synthesis and biological evaluation of novel DNA gyrase inhibitors and their siderophore mimic conjugates
Lamut, Andraž, Cruz, Cristina D., Skok, Žiga, Barančoková, Michaela, Zidar, Nace, Zega, Anamarija, Mašič, Lucija Peterlin, Ilaš, Janez, Tammela, Päivi, Kikelj, Danijel, Tomašič, Tihomir
Published in Bioorganic chemistry (01.01.2020)
Published in Bioorganic chemistry (01.01.2020)
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Journal Article
Synthesis and Evaluation of N‐Phenylpyrrolamides as DNA Gyrase B Inhibitors
Durcik, Martina, Tammela, Päivi, Barančoková, Michaela, Tomašič, Tihomir, Ilaš, Janez, Kikelj, Danijel, Zidar, Nace
Published in ChemMedChem (22.01.2018)
Published in ChemMedChem (22.01.2018)
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Journal Article
Second-generation 4,5,6,7-tetrahydrobenzo[ d ]thiazoles as novel DNA gyrase inhibitors
Lamut, Andraž, Skok, Žiga, Barančoková, Michaela, Gutierrez, Lucas J, Cruz, Cristina D, Tammela, Päivi, Draskovits, Gábor, Szili, Petra Éva, Nyerges, Ákos, Pál, Csaba, Molek, Peter, Bratkovič, Tomaž, Ilaš, Janez, Zidar, Nace, Zega, Anamarija, Enriz, Ricardo D, Kikelj, Danijel, Tomašič, Tihomir
Published in Future medicinal chemistry (01.02.2020)
Published in Future medicinal chemistry (01.02.2020)
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Journal Article
Synthesis and Evaluation of N-Phenylpyrrolamides as DNA GyraseB Inhibitors
Durcik, Martina, Tammela, Paivi, Barancokova, Michaela, Tomasic, Tihomir, Ilas, Janez, Kikelj, Danijel, Zidar, Nace
Published in ChemMedChem (22.01.2018)
Published in ChemMedChem (22.01.2018)
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Journal Article