Autoimmune pathways in mice and humans are blocked by pharmacological stabilization of the TYK2 pseudokinase domain
Burke, James R, Cheng, Lihong, Gillooly, Kathleen M, Strnad, Joann, Zupa-Fernandez, Adriana, Catlett, Ian M, Zhang, Yifan, Heimrich, Elizabeth M, McIntyre, Kim W, Cunningham, Mark D, Carman, Julie A, Zhou, Xiadi, Banas, Dana, Chaudhry, Charu, Li, Sha, D'Arienzo, Celia, Chimalakonda, Anjaneya, Yang, XiaoXia, Xie, Jenny H, Pang, Jian, Zhao, Qihong, Rose, Shawn M, Huang, Jinwen, Moslin, Ryan M, Wrobleski, Stephen T, Weinstein, David S, Salter-Cid, Luisa M
Published in Science translational medicine (24.07.2019)
Published in Science translational medicine (24.07.2019)
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Bruton's tyrosine kinase inhibitor BMS-986142 in experimental models of rheumatoid arthritis enhances efficacy of agents representing clinical standard-of-care
Gillooly, Kathleen M, Pulicicchio, Claudine, Pattoli, Mark A, Cheng, Lihong, Skala, Stacey, Heimrich, Elizabeth M, McIntyre, Kim W, Taylor, Tracy L, Kukral, Daniel W, Dudhgaonkar, Shailesh, Nagar, Jignesh, Banas, Dana, Watterson, Scott H, Tino, Joseph A, Fura, Aberra, Burke, James R
Published in PloS one (24.07.2017)
Published in PloS one (24.07.2017)
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Identification of Tricyclic Agonists of Sphingosine-1-phosphate Receptor 1 (S1P1) Employing Ligand-Based Drug Design
Xiao, Hai-Yun, Watterson, Scott H, Langevine, Charles M, Srivastava, Anurag S, Ko, Soo S, Zhang, Yanlei, Cherney, Robert J, Guo, Wei-Wei, Gilmore, John L, Sheppeck, James E, Wu, Dauh-Rurng, Li, Peng, Ramasamy, Duraisamy, Arunachalam, Piramanayagam, Mathur, Arvind, Taylor, Tracy L, Shuster, David J, McIntyre, Kim W, Shen, Ding-Ren, Yarde, Melissa, Cvijic, Mary Ellen, Marino, Anthony M, Balimane, Praveen V, Yang, Zheng, Banas, Dana M, Cornelius, Georgia, D’Arienzo, Celia J, Warrack, Bethanne M, Lehman-McKeeman, Lois, Salter-Cid, Luisa M, Xie, Jenny, Barrish, Joel C, Carter, Percy H, Dyckman, Alaric J, Dhar, T. G. Murali
Published in Journal of medicinal chemistry (10.11.2016)
Published in Journal of medicinal chemistry (10.11.2016)
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DGKα/ζ inhibitors combine with PD-1 checkpoint therapy to promote T cell-mediated antitumor immunity
Wichroski, Michael, Benci, Joseph, Liu, Si-Qi, Chupak, Louis, Fang, Jie, Cao, Carolyn, Wang, Cindy, Onorato, Joelle, Qiu, Hongchen, Shan, Yongli, Banas, Dana, Powles, Ryan, Locke, Gregory, Witt, Abigail, Stromko, Caitlyn, Qi, Huilin, Zheng, Xiaofan, Martin, Scott, Ding, Min, Gentles, Robert, Meanwell, Nicholas, Velaparthi, Upender, Olson, Richard, Wee, Susan, Tenney, Daniel, Parker, Christopher G, Cravatt, Benjamin F, Lawrence, Michael, Borzilleri, Robert, Lees, Emma
Published in Science translational medicine (25.10.2023)
Published in Science translational medicine (25.10.2023)
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Potent and Selective Agonists of Sphingosine 1‑Phosphate 1 (S1P1): Discovery and SAR of a Novel Isoxazole Based Series
Watterson, Scott H, Guo, Junqing, Spergel, Steve H, Langevine, Charles M, Moquin, Robert V, Shen, Ding Ren, Yarde, Melissa, Cvijic, Mary Ellen, Banas, Dana, Liu, Richard, Suchard, Suzanne J, Gillooly, Kathleen, Taylor, Tracy, Rex-Rabe, Sandra, Shuster, David J, McIntyre, Kim W, Cornelius, Georgia, D’Arienzo, Celia, Marino, Anthony, Balimane, Praveen, Warrack, Bethanne, Salter-Cid, Luisa, McKinnon, Murray, Barrish, Joel C, Carter, Percy H, Pitts, William J, Xie, Jenny, Dyckman, Alaric J
Published in Journal of medicinal chemistry (24.03.2016)
Published in Journal of medicinal chemistry (24.03.2016)
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B cells from African American lupus patients exhibit an activated phenotype
Menard, Laurence C, Habte, Sium, Gonsiorek, Waldemar, Lee, Deborah, Banas, Dana, Holloway, Deborah A, Manjarrez-Orduno, Nataly, Cunningham, Mark, Stetsko, Dawn, Casano, Francesca, Kansal, Selena, Davis, Patricia M, Carman, Julie, Zhang, Clarence K, Abidi, Ferva, Furie, Richard, Nadler, Steven G, Suchard, Suzanne J
Published in JCI insight (16.06.2016)
Published in JCI insight (16.06.2016)
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Identification and synthesis of potent and selective pyridyl-isoxazole based agonists of sphingosine-1-phosphate 1 (S1P1)
Guo, Junqing, Watterson, Scott H., Spergel, Steven H., Kempson, James, Langevine, Charles M., Shen, Ding Ren, Yarde, Melissa, Cvijic, Mary Ellen, Banas, Dana, Liu, Richard, Suchard, Suzanne J., Gillooly, Kathleen, Taylor, Tracy, Rex-Rabe, Sandra, Shuster, David J., McIntyre, Kim W., Cornelius, Georgia, D’Arienzo, Celia, Marino, Anthony, Balimane, Praveen, Salter-Cid, Luisa, McKinnon, Murray, Barrish, Joel C., Carter, Percy H., Pitts, William J., Xie, Jenny, Dyckman, Alaric J.
Published in Bioorganic & medicinal chemistry letters (15.05.2016)
Published in Bioorganic & medicinal chemistry letters (15.05.2016)
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Human phosphatase RET31, and variants thereof
SIEMERS NATHAN, JACKSON DONALD G, RAMANATHAN CHANDRA S, SUCHARD SUZANNE J, FINGER JOSHUA, TODDERUD C. GORDON, BANAS DANA, LEE LIANA
Year of Publication 15.04.2008
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Year of Publication 15.04.2008
Patent
Human phosphatase RET31, and variants thereof
Jackson, Donald G, Ramanathan, Chandra S, Lee, Liana, Siemers, Nathan, Suchard, Suzanne J, Finger, Joshua, Todderud, C. Gordon, Banas, Dana
Year of Publication 15.04.2008
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Year of Publication 15.04.2008
Patent
Polynucleotides encoding the novel human phosphatase, RET31, and variants thereof
Jackson, Donald G, Ramanathan, Chandra S, Feder, John N, Lee, Liana, Nelson, Thomas C, Siemers, Nathan, Suchard, Suzanne J, Finger, Joshua, Todderud, C. Gordon, Banas, Dana
Year of Publication 26.12.2006
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Year of Publication 26.12.2006
Patent
Human phosphatase RET31, and variants thereof
SIEMERS NATHAN, MINTIER GABE, JACKSON DONALD G, BOL DAVID, RAMANATHAN CHANDRA S, TODDERRUD C. G, BANAS DANA, FEDER JOHN N, NELSON THOMAS C, LEE LIANA, SCHIEVEN GARY, BASSOLINO DONNA, MCATEE PATRICK, FINGER JOSHUA, KRYSTEK STANLEY, SUCHARD SUZANNE
Year of Publication 19.01.2006
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Year of Publication 19.01.2006
Patent
POLYNUCLEOTIDES ENCODING NOVEL HUMAN PHOSPHATASES
SIEMERS NATHAN, MINTIER GABE, JACKSON DONALD G, BOL DAVID, RAMANATHAN CHANDRA S, TODDERRUD C. G, BANAS DANA, FEDER JOHN N, NELSON THOMAS C, LEE LIANA, SCHIEVEN GARY, BASSOLINO DONNA, MCATEE PATRICK, FINGER JOSHUA, KRYSTEK STANLEY, SUCHARD SUZANNE
Year of Publication 16.06.2005
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Year of Publication 16.06.2005
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POLYNUCLEOTIDES ENCODING HUMAN PHOSPHATASES
BASSOLINO, DONNA, MINTIER, GABE, SUCHARD, SUZANNE, LEE, LIANA, BOL, DAVID, JACKSON, DONALD, G, SCHIEVEN, GARY, BANAS, DANA, SIEMERS, NATHAN, KRYSTEK, STANLEY, FINGER, JOSHUA, MCATEE, PATRICK, RAMANATHAN, CHANDRA, TODDERUD, C, GORDON
Year of Publication 24.09.2003
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Year of Publication 24.09.2003
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POLYNUCLEOTIDES ENCODING HUMAN PHOSPHATASES
BASSOLINO, DONNA, MINTIER, GABE, LEE, LIANA, BOL, DAVID, JACKSON, DONALD, G, SCHIEVEN, GARY, BANAS, DANA, SIEMERS, NATHAN, NELSON, THOMAS, KRYSTEK, STANLEY, SUCHARD, SUSAN, FINGER, JOSHUA, FEDER, JOHN, MCATEE, PATRICK, RAMANATHAN, CHANDRA, TODDERUD, C, GORDON
Year of Publication 10.04.2003
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Year of Publication 10.04.2003
Patent
POLYNUCLEOTIDES ENCODING NOVEL HUMAN PHOSPHATASES
BASSOLINO, DONNA, MINTIER, GABE, LEE, LIANA, BOL, DAVID, JACKSON, DONALD, G, SCHIEVEN, GARY, BANAS, DANA, SIEMERS, NATHAN, NELSON, THOMAS, KRYSTEK, STANLEY, SUCHARD, SUSAN, FINGER, JOSHUA, FEDER, JOHN, MCATEE, PATRICK, RAMANATHAN, CHANDRA, TODDERUD, C, GORDON
Year of Publication 25.07.2002
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Year of Publication 25.07.2002
Patent
POLYNUCLEOTIDES ENCODING HUMAN PHOSPHATASES
JACKSON, DONALD G, BASSOLINO, DONNA, MINTIER, GABE, TODDERUD, GORDON C, LEE, LIANA, BOL, DAVID, BANAS, DANA, SCHIEVEN, GARY, SIEMERS, NATHAN, NELSON, THOMAS, SUCHARD, SUSAN, KRYSTEK, STANLEY, FINGER, JOSHUA, FEDER, JOHN, MCATEE, PATRICK, RAMANATHAN, CHANDRA
Year of Publication 25.07.2002
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Year of Publication 25.07.2002
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