Second-Generation Pharmacological Chaperones: Beyond Inhibitors
Tran, My Lan, Génisson, Yves, Ballereau, Stéphanie, Dehoux, Cécile
Published in Molecules (Basel, Switzerland) (09.07.2020)
Published in Molecules (Basel, Switzerland) (09.07.2020)
Get full text
Journal Article
Natural and Bioinspired Lipidic Alkynylcarbinols as Leishmanicidal, Antiplasmodial, Trypanocidal, Fungicidal, Antibacterial, and Antimycobacterial Agents
Bouvet, Jon, Maraval, Valérie, Ballereau, Stéphanie, Bernardes-Génisson, Vania, Génisson, Yves
Published in Journal of natural products (Washington, D.C.) (20.09.2024)
Published in Journal of natural products (Washington, D.C.) (20.09.2024)
Get full text
Journal Article
Pharmacological Chaperone Therapy for Pompe Disease
Borie-Guichot, Marc, Tran, My Lan, Génisson, Yves, Ballereau, Stéphanie, Dehoux, Cécile
Published in Molecules (Basel, Switzerland) (29.11.2021)
Published in Molecules (Basel, Switzerland) (29.11.2021)
Get full text
Journal Article
Synthesis and biological evaluation of natural Lachnophyllum methyl ester, Lachnophyllum lactone and their synthetic analogs
Adande, Kodjo, Simalou, Oudjaniyobi, Ardanuy, Juline, Eloh, Kodjo, Mehalla, Chérine, Constant, Patricia, Fabing, Isabelle, Génisson, Yves, Ballereau, Stéphanie
Published in Organic & biomolecular chemistry (09.10.2024)
Published in Organic & biomolecular chemistry (09.10.2024)
Get full text
Journal Article
Phosphopantetheinyl transferase binding and inhibition by amidino-urea and hydroxypyrimidinethione compounds
Carivenc, Coralie, Maveyraud, Laurent, Blanger, Claire, Ballereau, Stéphanie, Roy-Camille, Coralie, Nguyen, Minh Chau, Génisson, Yves, Guilhot, Christophe, Chalut, Christian, Pedelacq, Jean-Denis, Mourey, Lionel
Published in Scientific reports (10.09.2021)
Published in Scientific reports (10.09.2021)
Get full text
Journal Article
Phenyl dialkynylcarbinols, a Bioinspired Series of Synthetic Antitumor Acetylenic Lipids
Bossuat, Margaux, Rullière, Pauline, Preuilh, Nadège, Peixoto, Antonio, Joly, Etienne, Gomez, Jean-Guillaume, Bourkhis, Maroua, Rodriguez, Frédéric, Gonçalves, Fernanda, Fabing, Isabelle, Gaspard, Hafida, Bernardes-Génisson, Vania, Maraval, Valérie, Ballereau, Stéphanie, Chauvin, Remi, Britton, Sébastien, Génisson, Yves
Published in Journal of medicinal chemistry (26.10.2023)
Published in Journal of medicinal chemistry (26.10.2023)
Get full text
Journal Article
Enantioselective Stereodivergent Synthesis of Jaspine B and 4-epi-Jaspine B from Axially Chiral Allenols
Alnazer, Heba, Castellan, Tessa, Salma, Yahya, Genisson, Yves, Ballereau, Stephanie
Published in Synlett (01.01.2019)
Published in Synlett (01.01.2019)
Get more information
Journal Article
Chemical modification of clay nanocomposites for the improvement of the catalytic properties of Lipase A from Candida antarctica
Cavalcante, Antônio Luthierre Gama, Chaves, Anderson Valério, Fechine, Pierre Basílio Almeida, Holanda Alexandre, Jeferson Yves Nunes, Freire, Tiago Melo, Davi, Dalila Maria Barbosa, Neto, Francisco Simão, de Sousa, Isamayra Germano, da Silva Moreira, Katerine, de Oliveira, André Luiz Barros, de Mattos, Marcos Carlos, Oliveira, Maria Conceição Ferreira, de Brito, Maria Vieira, Ballereau, Stéphanie, Bernardes-Génisson, Vania, da Fonseca, Aluísio Marques, dos Santos, José C.S.
Published in Process biochemistry (1991) (01.09.2022)
Published in Process biochemistry (1991) (01.09.2022)
Get full text
Journal Article
Phosphorus Dendrimers for Metal-Free Ligation: Design of Multivalent Pharmacological Chaperones against Gaucher Disease
Tran, My Lan, Borie-Guichot, Marc, Garcia, Virginie, Oukhrib, Abdelouahd, Génisson, Yves, Levade, Thierry, Ballereau, Stéphanie, Turrin, Cédric-Olivier, Dehoux, Cécile
Published in Chemistry : a European journal (21.09.2023)
Published in Chemistry : a European journal (21.09.2023)
Get full text
Journal Article
Rapid access to jaspine B and its enantiomer
Santos, Cécile, Fabing, Isabelle, Saffon, Nathalie, Ballereau, Stéphanie, Génisson, Yves
Published in Tetrahedron (01.09.2013)
Published in Tetrahedron (01.09.2013)
Get full text
Journal Article
Fragment-Based Ligand Discovery Applied to the Mycolic Acid Methyltransferase Hma (MmaA4) from Mycobacterium tuberculosis : A Crystallographic and Molecular Modelling Study
Galy, Romain, Ballereau, Stéphanie, Génisson, Yves, Mourey, Lionel, Plaquevent, Jean-Christophe, Maveyraud, Laurent
Published in Pharmaceuticals (Basel, Switzerland) (08.12.2021)
Published in Pharmaceuticals (Basel, Switzerland) (08.12.2021)
Get full text
Journal Article
Chemistry and Biology of HPAs: A Family of Ceramide Trafficking Inhibitors
Berkeš, Dušan, Daïch, Adam, Santos, Cécile, Ballereau, Stéphanie, Génisson, Yves
Published in Chemistry : a European journal (05.12.2016)
Published in Chemistry : a European journal (05.12.2016)
Get full text
Journal Article
Concise asymmetric synthesis of new enantiomericC-alkyl pyrrolidines acting as pharmacological chaperones against Gaucher disease
Castellan, Tessa, Garcia, Virginie, Rodriguez, Frederic, Fabing, Isabelle, Shchukin, Yevhenii, Tran, My Lan, Ballereau, Stephanie, Levade, Thierry, Genisson, Yves, Dehoux, Cecile
Published in Organic & biomolecular chemistry (21.10.2020)
Published in Organic & biomolecular chemistry (21.10.2020)
Get full text
Journal Article
N,O-Dialkyl deoxynojirimycin derivatives as CERT START domain ligands
Castellan, Tessa, Santos, Cécile, Rodriguez, Frédéric, Lepage, Mathieu L., Liang, Yan, Bodlenner, Anne, Compain, Philippe, Génisson, Yves, Dehoux, Cécile, Ballereau, Stéphanie
Published in Bioorganic & medicinal chemistry letters (15.01.2020)
Published in Bioorganic & medicinal chemistry letters (15.01.2020)
Get full text
Journal Article
Alkyne‐Tagged Analogue of Jaspine B: New Tool for Identifying Jaspine B Mode of Action
Rozié, Alexandrine, Santos, Cécile, Fabing, Isabelle, Calsou, Patrick, Britton, Sébastien, Génisson, Yves, Ballereau, Stéphanie
Published in Chembiochem : a European journal of chemical biology (04.12.2018)
Published in Chembiochem : a European journal of chemical biology (04.12.2018)
Get full text
Journal Article
Iminosugar-based ceramide mimicry for the design of new CERT START domain ligands
Santos, Cécile, Stauffert, Fabien, Ballereau, Stéphanie, Dehoux, Cécile, Rodriguez, Frédéric, Bodlenner, Anne, Compain, Philippe, Génisson, Yves
Published in Bioorganic & medicinal chemistry (15.03.2017)
Published in Bioorganic & medicinal chemistry (15.03.2017)
Get full text
Journal Article
Synthesis and biological evaluation of aziridine-containing analogs of phytosphingosine
Ballereau, Stéphanie, Andrieu-Abadie, Nathalie, Saffon, Nathalie, Génisson, Yves
Published in Tetrahedron (08.04.2011)
Published in Tetrahedron (08.04.2011)
Get full text
Journal Article
Multivalent pyrrolidines acting as pharmacological chaperones against Gaucher disease
Borie-Guichot, Marc, Lan Tran, My, Garcia, Virginie, Oukhrib, Abdelouahd, Rodriguez, Frédéric, Turrin, Cédric-Olivier, Levade, Thierry, Génisson, Yves, Ballereau, Stéphanie, Dehoux, Cécile
Published in Bioorganic chemistry (01.05.2024)
Published in Bioorganic chemistry (01.05.2024)
Get full text
Journal Article
The CERT antagonist HPA-12: First practical synthesis and individual binding evaluation of the four stereoisomers
Santos, Cécile, Fleury, Laurence, Rodriguez, Frédéric, Markus, Jozef, Berkeš, Dušan, Daïch, Adam, Ausseil, Frédéric, Baudoin-Dehoux, Cécile, Ballereau, Stéphanie, Génisson, Yves
Published in Bioorganic & medicinal chemistry (01.05.2015)
Published in Bioorganic & medicinal chemistry (01.05.2015)
Get full text
Journal Article
Flexible and enantioselective access to jaspine B and biologically active chain-modified analogues thereof
Salma, Yahya, Ballereau, Stephanie, Maaliki, Carine, Ladeira, Sonia, Andrieu-Abadie, Nathalie, Genisson, Yves
Published in Organic & biomolecular chemistry (21.07.2010)
Published in Organic & biomolecular chemistry (21.07.2010)
Get full text
Journal Article