Design, synthesis, and biological evaluation of phenyl thiazole-based AR-V7 degraders
Bhumireddy, Archana, Bandaru, N.V.M. Rao, Raghurami Reddy, B., Gore, Suraj T., Mukherjee, Subhendu, Balasubramanian, Wesley Roy, Sumanth Kumar, V., Alapati, Krishna Satya, Venkata Gowri Chandra Sekhar, Kondapalli, Nellore, Kavitha, Abbineni, Chandrasekhar, Samajdar, Susanta
Published in Bioorganic & medicinal chemistry letters (01.01.2022)
Published in Bioorganic & medicinal chemistry letters (01.01.2022)
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Journal Article
COMPOUNDS AND COMPOSITIONS FOR TREATING HEMATOLOGICAL DISORDERS
NELLORE KAVITHA, GUMMADI VENKATESHWAR RAO, SAMAJDAR SUSANTA, DAGINAKATTE GIRISH, BALASUBRAMANIAN WESLEY ROY
Year of Publication 14.02.2024
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Year of Publication 14.02.2024
Patent
Discovery of CA-4948, an Orally Bioavailable IRAK4 Inhibitor for Treatment of Hematologic Malignancies
Gummadi, Venkateshwar Rao, Boruah, Anima, Ainan, Bharathi Raja, Vare, Brahma Reddy, Manda, Srinivas, Gondle, Hari Prakash, Kumar, Shiva Nagendra, Mukherjee, Subhendu, Gore, Suraj T, Krishnamurthy, Narasimha Rao, Marappan, Sivapriya, Nayak, Shilpa S, Nellore, Kavitha, Balasubramanian, Wesley Roy, Bhumireddy, Archana, Giri, Sanjeev, Gopinath, Sreevalsam, Samiulla, Dodheri S, Daginakatte, Girish, Basavaraju, Aravind, Chelur, Shekar, Eswarappa, Rajesh, Belliappa, Charamanna, Subramanya, Hosahalli S, Booher, Robert N, Ramachandra, Murali, Samajdar, Susanta
Published in ACS medicinal chemistry letters (10.12.2020)
Published in ACS medicinal chemistry letters (10.12.2020)
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Journal Article
Abstract 3852: Combination efficacy and safety profile of an orally bioavailable small molecule agent targeting CD47/SIRPα axis
Daginakatte, Girish, Pottayil, Sasikumar, Chennakrishna, Gundala, Balasubramanian, Wesley Roy, Naremaddepalli, Sudarshan, Bhumireddy, Archana, Patil, Sandeep, Nellore, Kavitha, Chand, Priyabrata, Aithal, Kiran, Dhudashiya, Amit, DS, Samiulla, Eswarappa, Rajesh, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract C127: Discovery of AUR-112, a novel MALT1 protease inhibitor for the treatement of B cell lymphomas
Balasubramanian, Wesley Roy, Raju, Sammeta Srinivasa, K.Y, Vasantha, Reddy, Archana Bhumi, Maben, Janith Mary, Patil, Sandeep Sadashiv, N.R, Raghavendra, B, Kiran Aithal, K.B, Charamanna, Chikkanna, Dinesh, Nellore, Kavitha, D.S, Samiulla, Daginakatte, Girish, Chelur, Shekar, Ramachandra, Murali, Samajdar, Susanta
Published in Molecular cancer therapeutics (01.12.2023)
Published in Molecular cancer therapeutics (01.12.2023)
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Journal Article
Abstract B007: Potent antitumor activity of a novel and orally available small-molecule antagonist targeting the CD47/SIRPα pathway
Sasikumar, Pottayil G., Gundala, Chennakrishnareddy, Balasubramanian, Wesley R., Naremaddepalli, Sudarshan S., Bhumireddy, Archana, Patil, Sandeep S., Dhudashiya, Amit A., Rayavarapu, Vijaysai, Lakshminarasimhan, Anirudha, Samiulla, Dodheri S., Aithal, Kiran, Daginakatte, Girish, Ramachandra, Murali
Published in Molecular cancer therapeutics (01.01.2018)
Published in Molecular cancer therapeutics (01.01.2018)
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Journal Article
Abstract 1650: Targeting CD47- SIRPα interaction by novel peptide-based antagonists
Sasikumar, Pottayil G., Gundala, Chennakrishnareddy, Gowda, Nagaraj M., Naremaddepalli, Sudarshan S., Bhumireddy, Archana, Nair, Rashmi, Balasubramanian, Wesley Roy, Lakshminarasimhan, Anirudha, Dodheri, Samiulla S., Aithal, Kiran, Ramachandra, Raghuveer K., Daginakatte, Girish, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Journal Article
Abstract 5108: Potent small molecule compounds that selectively inhibit proliferation of ABC-DLBCL cell lines
Satyam, Leena Khare, Chikkanna, Dinesh, Khairnar, Vinayak, Pothuganti, Manoj, Panigrahi, Sunil, Lakshminarasimhan, Anirudha, Rao, Narasimha, Balasubramanian, Wesley, Patil, Sandeep, Gopinath, Sreevalsam, Upendra, Gunta, Nagaraj, Jwala, Aithal, Kiran, Ahuja, Vijay, Giri, Sanjeev, Pandit, Chetan, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Journal Article
Abstract 3646: Novel IRAK-4 inhibitors exhibit highly potent anti-proliferative activity in DLBCL cell lines with activating MYD88 L265P mutation
Balasubramanian, Wesley Roy, Gummadi, Venkateshwar Rao, D, Ravi Krishna Babu, Marappan, Sivapriya, Choudhary, Bhavesh, Gopinath, Sreevalsam, Nellore, Kavitha, Chelur, Shekar, Daginakatte, Girish, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Journal Article
Abstract 4798: Efficacy and safety of highly selective novel IRAK4 inhibitors for treatment of ABC-DLBCL
Balasubramanian, Wesley Roy, Gummadi, Venkateshwar Rao, Nellore, Kavitha, Mukherjee, Subhendu, Marappan, Sivapriya, Basavaraju, Aravind, Ainan, Bharathi Raja, Daginakatte, Girish, Gopinath, Sreevalsam, Giri, Sanjeev, Antony, Thomas, Chelur, Shekar, Samajdar, Susanta, Pandit, Chetan, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
Abstract 3500: AUR103 an oral small molecule CD47 antagonist in combination with azacytidine and bortezomib exhibits potent anti-tumor activity in myeloma and leukemia models in vitro and in vivo
Daginakatte, Girish C., Pottayil, Sasikumar, Naremaddepalli, Sudarshan, Chennakrishnareddy, Gundala, Bilugudi, Prasad, Tangella, Sai Krishna, Patil, Sandeep, Gowda, Nagesh, Aithal, Kiran, Balasubramanian, Wesley Roy, Dhudashiya, Amit, Dodheri, Samiulla, Nellore, Kavitha, Samajdar, Susanta, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
A simple method for the production of recombinant proteins from mammalian cells
Wu, Chia-Hung, Balasubramanian, Wesley Roy, Ko, Ya-Ping, Hsu, George, Chang, Shih-En, Prijovich, Zeljko M, Chen, Kai-Chuan, Roffler, Steve R
Published in Biotechnology and applied biochemistry (01.10.2004)
Published in Biotechnology and applied biochemistry (01.10.2004)
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Journal Article
Targeting ALK for cancer therapy: high throughput screening assays
Abdul Kadir, Mohamad Fairus, Alagapan, Pratheev, Lim, Yang Jin, Kong, Wai Mun, Balan, Dharvind, Dorasamy, Mathura Subangari, Balasubramanian, Wesley Roy, Marappan, Sivapriya, Subramaniam, Umarani, Nellore, Kavitha, Anthony, Thomas
Published in Frontiers in pharmacology (2018)
Published in Frontiers in pharmacology (2018)
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Journal Article
Abstract C191: Efficacy of novel IRAK4 inhibitors in ABC-DLBCL and AML models
Rao, Venkateshwar, Balasubramanian, Wesley Roy, Nellore, Kavitha, Marappan, Sivapriya, Basavaraju, Aravind, Raja Ainan, Bharathi, Daginakatte, Girish, Gopinath, Sreevalsam, Giri, Sanjeev, Antony, Thomas, Chelur, Shekar, Samajdar, Susanta, Pandit, Chetan, Ramachandra, Murali
Published in Molecular cancer therapeutics (01.12.2015)
Published in Molecular cancer therapeutics (01.12.2015)
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Journal Article
혈액 장애를 치료하기 위한 화합물 및 조성물
NELLORE KAVITHA, GUMMADI VENKATESHWAR RAO, SAMAJDAR SUSANTA, DAGINAKATTE GIRISH, BALASUBRAMANIAN WESLEY ROY
Year of Publication 20.11.2019
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Year of Publication 20.11.2019
Patent
Discovery of selective RORγ inverse agonists and demonstration of efficacy in inflammatory disease models
Damarla, Ravi Krishna Babu, Ujjinamatada, Ravi K, Nellore, Kavitha, Dodheri, Samiulla S, Chelur, Shekar, Charamanna, K.B, Mukherjee, Subhendu, Reddy, CH Sandeep, Balasubramanian, Wesley Roy, Rathod, Sanjay B, Lakshminarasimhan, Anirudha, Rao, K Narasimha, Ramanathan, Anuradha, Mahalingam, Natarajan, Girish, AR, Samajdar, Susanta, Pandit, Chetan, Ramachandra, Murali
Published in The Journal of immunology (1950) (01.05.2016)
Published in The Journal of immunology (1950) (01.05.2016)
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Journal Article
Efficacy of selective RAR-related orphan receptor gamma (RORγ) inverse agonists in psoriasis and asthma models (CCR6P.278)
Nellore, Kavitha, Bejugam, Mallesham, Damarla, Ravi Krishna Babu, Hegde, Pragathi, Dodheri, Samiulla, Mukherjee, Subhendu, Rao, Narasimha, Lakshminarasimhan, Anirudha, Ramanathan, Anuradha, Balasubramanian, Wesley, Mattegunta, Suresh Babu, Mahalingam, Natarajan, Samajdar, Susanta, Subramanya, Hosahalli
Published in The Journal of immunology (1950) (01.05.2014)
Published in The Journal of immunology (1950) (01.05.2014)
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Journal Article
Compounds and compositions for treating hematological disorders
Gummadi, Venkateshwar Rao, Daginakatte, Girish, Nellore, Kavitha, Samajdar, Susanta, Balasubramanian, Wesley Roy
Year of Publication 04.07.2024
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Year of Publication 04.07.2024
Patent
Compounds and compositions for treating hematological disorders
Gummadi, Venkateshwar Rao, Daginakatte, Girish, Nellore, Kavitha, Samajdar, Susanta, Balasubramanian, Wesley Roy
Year of Publication 02.05.2024
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Year of Publication 02.05.2024
Patent
COMPOUNDS AND COMPOSITIONS FOR TREATING HEMATOLOGICAL DISORDERS
SAMAJDAR, Susanta, BALASUBRAMANIAN, Wesley Roy, NELLORE, Kavitha, DAGINAKATTE, Girish, GUMMADI, Venkateshwar Rao
Year of Publication 13.12.2023
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Year of Publication 13.12.2023
Patent