Development of a Multiplexed Activity-Based Protein Profiling Assay to Evaluate Activity of Endocannabinoid Hydrolase Inhibitors
Janssen, Antonius P. A, van der Vliet, Daan, Bakker, Alexander T, Jiang, Ming, Grimm, Sebastian H, Campiani, Giuseppe, Butini, Stefania, van der Stelt, Mario
Published in ACS chemical biology (21.09.2018)
Published in ACS chemical biology (21.09.2018)
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Journal Article
Identification of α,β-Hydrolase Domain Containing Protein 6 as a Diacylglycerol Lipase in Neuro-2a Cells
van Esbroeck, Annelot C M, Kantae, Vasudev, Di, Xinyu, van der Wel, Tom, den Dulk, Hans, Stevens, Anna F, Singh, Simar, Bakker, Alexander T, Florea, Bogdan I, Stella, Nephi, Overkleeft, Herman S, Hankemeier, Thomas, van der Stelt, Mario
Published in Frontiers in molecular neuroscience (26.11.2019)
Published in Frontiers in molecular neuroscience (26.11.2019)
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Journal Article
Development of a Retinal-Based Probe for the Profiling of Retinaldehyde Dehydrogenases in Cancer Cells
Koenders, Sebastiaan T. A, Wijaya, Lukas S, Erkelens, Martje N, Bakker, Alexander T, van der Noord, Vera E, van Rooden, Eva J, Burggraaff, Lindsey, Putter, Pasquale C, Botter, Else, Wals, Kim, van den Elst, Hans, den Dulk, Hans, Florea, Bogdan I, van de Water, Bob, van Westen, Gerard J. P, Mebius, Reina E, Overkleeft, Herman S, Le Dévédec, Sylvia E, van der Stelt, Mario
Published in ACS central science (26.12.2019)
Published in ACS central science (26.12.2019)
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Journal Article
A Suite of Activity-Based Probes To Dissect the KLK Activome in Drug-Resistant Prostate Cancer
Lovell, Scott, Zhang, Leran, Kryza, Thomas, Neodo, Anna, Bock, Nathalie, De Vita, Elena, Williams, Elizabeth D, Engelsberger, Elisabeth, Xu, Congyi, Bakker, Alexander T, Maneiro, Maria, Tanaka, Reiko J, Bevan, Charlotte L, Clements, Judith A, Tate, Edward W
Published in Journal of the American Chemical Society (16.06.2021)
Published in Journal of the American Chemical Society (16.06.2021)
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Journal Article
Chemical Proteomics Reveals Antibiotic Targets of Oxadiazolones in MRSA
Bakker, Alexander T., Kotsogianni, Ioli, Mirenda, Liza, Straub, Verena M., Avalos, Mariana, van den Berg, Richard J. B. H. N., Florea, Bogdan I., van Wezel, Gilles P., Janssen, Antonius P. A., Martin, Nathaniel I., van der Stelt, Mario
Published in Journal of the American Chemical Society (18.01.2023)
Published in Journal of the American Chemical Society (18.01.2023)
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Journal Article
Synthetic studies with the brevicidine and laterocidine lipopeptide antibiotics including analogues with enhanced properties and in vivo efficacy
Al Ayed, Karol, Ballantine, Ross D, Hoekstra, Michael, Bann, Samantha J, Wesseling, Charlotte M J, Bakker, Alexander T, Zhong, Zheng, Li, Yong-Xin, Brüchle, Nora C, van der Stelt, Mario, Cochrane, Stephen A, Martin, Nathaniel I
Published in Chemical science (Cambridge) (24.03.2022)
Published in Chemical science (Cambridge) (24.03.2022)
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Journal Article
Discovery of isoquinoline sulfonamides as allosteric gyrase inhibitors with activity against fluoroquinolone-resistant bacteria
Bakker, Alexander T., Kotsogianni, Ioli, Avalos, Mariana, Punt, Jeroen M., Liu, Bing, Piermarini, Diana, Gagestein, Berend, Slingerland, Cornelis J., Zhang, Le, Willemse, Joost J., Ghimire, Leela B., van den Berg, Richard J. H. B. N., Janssen, Antonius P. A., Ottenhoff, Tom H. M., van Boeckel, Constant A. A., van Wezel, Gilles P., Ghilarov, Dmitry, Martin, Nathaniel I., van der Stelt, Mario
Published in Nature chemistry (01.09.2024)
Published in Nature chemistry (01.09.2024)
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Journal Article
Chemical Proteomics Reveals Off-Targets of the Anandamide Reuptake Inhibitor WOBE437
Gagestein, Berend, Stevens, Anna F., Fazio, Domenico, Florea, Bogdan I., van der Wel, Tom, Bakker, Alexander T., Fezza, Filomena, Dulk, Hans den, Overkleeft, Herman S., Maccarrone, Mauro, van der Stelt, Mario
Published in ACS chemical biology (20.05.2022)
Published in ACS chemical biology (20.05.2022)
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Journal Article
Biochemical and Cellular Characterization of the Function of Fluorophosphonate-Binding Hydrolase H (FphH) in Staphylococcus aureus Support a Role in Bacterial Stress Response
Fellner, Matthias, Walsh, Annabel, Dela Ahator, Stephen, Aftab, Nadia, Sutherland, Ben, Tan, Eng W., Bakker, Alexander T., Martin, Nathaniel I., van der Stelt, Mario, Lentz, Christian S.
Published in ACS infectious diseases (10.11.2023)
Published in ACS infectious diseases (10.11.2023)
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Journal Article
Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice
Mock, Elliot D, Mustafa, Mohammed, Gunduz-Cinar, Ozge, Cinar, Resat, Petrie, Gavin N, Kantae, Vasudev, Di, Xinyu, Ogasawara, Daisuke, Varga, Zoltan V, Paloczi, Janos, Miliano, Cristina, Donvito, Giulia, van Esbroeck, Annelot C M, van der Gracht, Anouk M F, Kotsogianni, Ioli, Park, Joshua K, Martella, Andrea, van der Wel, Tom, Soethoudt, Marjolein, Jiang, Ming, Wendel, Tiemen J, Janssen, Antonius P A, Bakker, Alexander T, Donovan, Colleen M, Castillo, Laura I, Florea, Bogdan I, Wat, Jesse, van den Hurk, Helma, Wittwer, Matthias, Grether, Uwe, Holmes, Andrew, van Boeckel, Constant A A, Hankemeier, Thomas, Cravatt, Benjamin F, Buczynski, Matthew W, Hill, Matthew N, Pacher, Pal, Lichtman, Aron H, van der Stelt, Mario
Published in Nature chemical biology (01.06.2020)
Published in Nature chemical biology (01.06.2020)
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Journal Article
Synthetic studies with the brevicidine and laterocidine lipopeptide antibiotics including analogues with enhanced properties and efficacy
Al Ayed, Karol, Ballantine, Ross D, Hoekstra, Michael, Bann, Samantha J, Wesseling, Charlotte M. J, Bakker, Alexander T, Zhong, Zheng, Li, Yong-Xin, Brüchle, Nora C, van der Stelt, Mario, Cochrane, Stephen A, Martin, Nathaniel I
Published in Chemical science (Cambridge) (24.03.2022)
Published in Chemical science (Cambridge) (24.03.2022)
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Journal Article
DNA GYRASE INHIBITORS
VAN DER STELT, Mario, MARTIN, Nathaniel I, PIERMARINI, Diana, KOTSOGIANNI, Ioli, LIU, Bing, VAN DEN BERG, Richard J.H.B.N, AVALOS, Mariana, VAN BOECKEL, Constant A.A, VAN WEZEL, Gilles P, PUNT, Jeroen M, BAKKER, Alexander T, GHILAROV, Dmitry
Year of Publication 30.05.2024
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Year of Publication 30.05.2024
Patent
DNA Gyrase Inhibitors
RICHARD J.H.B.N VAN DEN BERG, IOLI KOTSOGIANNI, NATHANIEL I. MARTIN, JEROEN M. PUNT, MARIANA AVALOS, GILLES P. VAN WEZEL, ALEXANDER T. BAKKER, CONSTANT A.A. VAN BOECKEL, DMITRY GHILAROV, DIANA PIERMARINI, MARIO VAN DER STELT, BING LIU
Year of Publication 30.05.2024
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Year of Publication 30.05.2024
Patent
A suite of activity-based probes to dissect the KLK activome in drug-resistant prostate cancer
Lovell, Scott, Zhang, Leran, Kryza, Thomas, Neodo, Anna, Bock, Nathalie, Williams, Elizabeth D, Engelsberger, Elisabeth, Xu, Congyi, Bakker, Alexander T, De Vita, Elena, Maneiro, Maria, Tanaka, Reiko J, Bevan, Charlotte L, Clements, Judith A, Tate, Edward William
Published in bioRxiv (15.04.2021)
Published in bioRxiv (15.04.2021)
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Paper
Modified human variable domains
BAKKER ALEXANDER BERTHOLD HENRIK, SILVERMAN PETER BRIAN, KRAMER ROBERT ARJAN
Year of Publication 27.06.2023
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Year of Publication 27.06.2023
Patent
Modified human variable domains
BAKKER ALEXANDER BERTHOLD HENRIK, SILVERMAN PETER BRIAN, KRAMER ROBERT ARJAN
Year of Publication 25.03.2022
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Year of Publication 25.03.2022
Patent
ANTIBODY COMPOSITIONS
ALVENTE TUDOR, BAKKER ALEXANDER BERTHOLD HENDRIK, HENDRIKS LINDA JOHANNA ALEIDA, DALPIN, GUILLAUME, DESIREE, POIRIER, EMILY, BRIGITTE, DOORNBOS, ROBERT, PAUL
Year of Publication 22.09.2023
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Year of Publication 22.09.2023
Patent