A Small Molecule RAS-Mimetic Disrupts RAS Association with Effector Proteins to Block Signaling
Athuluri-Divakar, Sai Krishna, Vasquez-Del Carpio, Rodrigo, Dutta, Kaushik, Baker, Stacey J., Cosenza, Stephen C., Basu, Indranil, Gupta, Yogesh K., Reddy, M.V. Ramana, Ueno, Lynn, Hart, Jonathan R., Vogt, Peter K., Mulholland, David, Guha, Chandan, Aggarwal, Aneel K., Reddy, E. Premkumar
Published in Cell (21.04.2016)
Published in Cell (21.04.2016)
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Journal Article
TGFβ reprograms TNF stimulation of macrophages towards a non-canonical pathway driving inflammatory osteoclastogenesis
Xia, Yuhan, Inoue, Kazuki, Du, Yong, Baker, Stacey J, Reddy, E Premkumar, Greenblatt, Matthew B, Zhao, Baohong
Published in Nature communications (07.07.2022)
Published in Nature communications (07.07.2022)
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Journal Article
Simultaneous CK2/TNIK/DYRK1 inhibition by 108600 suppresses triple negative breast cancer stem cells and chemotherapy-resistant disease
Sato, Katsutoshi, Padgaonkar, Amol A, Baker, Stacey J, Cosenza, Stephen C, Rechkoblit, Olga, Subbaiah, D R C Venkata, Domingo-Domenech, Josep, Bartkowski, Alison, Port, Elisa R, Aggarwal, Aneel K, Ramana Reddy, M V, Irie, Hanna Y, Reddy, E Premkumar
Published in Nature communications (03.08.2021)
Published in Nature communications (03.08.2021)
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Journal Article
ON01910, a non-ATP-competitive small molecule inhibitor of Plk1, is a potent anticancer agent
Gumireddy, Kiranmai, Reddy, M.V. Ramana, Cosenza, Stephen C., Nathan, R. Boomi, Baker, Stacey J., Papathi, Nabisa, Jiang, Jiandong, Holland, James, Reddy, E. Premkumar
Published in Cancer cell (01.03.2005)
Published in Cancer cell (01.03.2005)
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Journal Article
B-myb is an essential regulator of hematopoietic stem cell and myeloid progenitor cell development
Baker, Stacey J., Ma'ayan, Avi, Lieu, Yen K., John, Premila, Reddy, M. V. Ramana, Chen, Edward Y., Duan, Qiaonan, Snoeck, Hans-Willem, Reddy, E. Premkumar
Published in Proceedings of the National Academy of Sciences - PNAS (25.02.2014)
Published in Proceedings of the National Academy of Sciences - PNAS (25.02.2014)
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Journal Article
A Non-ATP-Competitive Inhibitor of BCR-ABL Overrides Imatinib Resistance
Gumireddy, Kiranmai, Baker, Stacey J., Cosenza, Stephen C., John, Premila, Kang, Anthony D., Robell, Kimberly A., M. V. Ramana Reddy, Reddy, E. Premkumar, Vogt, Peter K.
Published in Proceedings of the National Academy of Sciences - PNAS (08.02.2005)
Published in Proceedings of the National Academy of Sciences - PNAS (08.02.2005)
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Journal Article
A Contaminant Impurity, Not Rigosertib, Is a Tubulin Binding Agent
Baker, Stacey J., Cosenza, Stephen C., Athuluri-Divakar, Saikrishna, Reddy, M.V. Ramana, Vasquez-Del Carpio, Rodrigo, Jain, Rinku, Aggarwal, Aneel K., Reddy, E. Premkumar
Published in Molecular cell (02.07.2020)
Published in Molecular cell (02.07.2020)
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Journal Article
CDK4: a master regulator of the cell cycle and its role in cancer
Baker, Stacey J, Poulikakos, Poulikos I, Irie, Hanna Y, Parekh, Samir, Reddy, E Premkumar
Published in Genes & cancer (25.08.2022)
Published in Genes & cancer (25.08.2022)
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Journal Article
Discovery of 8‑Cyclopentyl-2-[4-(4-methyl-piperazin-1-yl)-phenylamino]-7-oxo-7,8-dihydro-pyrido[2,3‑d]pyrimidine-6-carbonitrile (7x) as a Potent Inhibitor of Cyclin-Dependent Kinase 4 (CDK4) and AMPK-Related Kinase 5 (ARK5)
Reddy, M. V. Ramana, Akula, Balireddy, Cosenza, Stephen C, Athuluridivakar, Saikrishna, Mallireddigari, Muralidhar R, Pallela, Venkat R, Billa, Vinay K, Subbaiah, D. R. C. Venkata, Bharathi, E. Vijaya, Vasquez-Del Carpio, Rodrigo, Padgaonkar, Amol, Baker, Stacey J, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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Journal Article
Targeting protein kinase CK2 and CDK4/6 pathways with a multi-kinase inhibitor ON108110 suppresses pro-survival signaling and growth in mantle cell lymphoma and T-acute lymphoblastic leukemia
Padgaonkar, Amol, Rechkoblit, Olga, Vasquez-Del Carpio, Rodgrigo, Pallela, Venkat, Venkata Subbaiah, Drc, Cosenza, Stephen C, Baker, Stacey J, Ramana Reddy, M V, Aggarwal, Aneel, Reddy, E Premkumar
Published in Oncotarget (28.12.2018)
Published in Oncotarget (28.12.2018)
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Journal Article
p89c-Myb is not required for fetal or adult hematopoiesis
Baker, Stacey J., Kumar, Atul, Reddy, E. Premkumar
Published in Genesis (New York, N.Y. : 2000) (01.05.2010)
Published in Genesis (New York, N.Y. : 2000) (01.05.2010)
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