Peptidomimetic α‑Acyloxymethylketone Warheads with Six-Membered Lactam P1 Glutamine Mimic: SARS-CoV‑2 3CL Protease Inhibition, Coronavirus Antiviral Activity, and in Vitro Biological Stability
Bai, Bing, Belovodskiy, Alexandr, Hena, Mostofa, Kandadai, Appan Srinivas, Joyce, Michael A, Saffran, Holly A, Shields, Justin A, Khan, Muhammad Bashir, Arutyunova, Elena, Lu, Jimmy, Bajwa, Sardeev K, Hockman, Darren, Fischer, Conrad, Lamer, Tess, Vuong, Wayne, van Belkum, Marco J, Gu, Zhengxian, Lin, Fusen, Du, Yanhua, Xu, Jia, Rahim, Mohammad, Young, Howard S, Vederas, John C, Tyrrell, D. Lorne, Lemieux, M. Joanne, Nieman, James A
Published in Journal of medicinal chemistry (24.02.2022)
Published in Journal of medicinal chemistry (24.02.2022)
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