Pregnenolone Can Protect the Brain from Cannabis Intoxication
Vallée, Monique, Vitiello, Sergio, Bellocchio, Luigi, Hébert-Chatelain, Etienne, Monlezun, Stéphanie, Martin-Garcia, Elena, Kasanetz, Fernando, Baillie, Gemma L., Panin, Francesca, Cathala, Adeline, Roullot-Lacarrière, Valérie, Fabre, Sandy, Hurst, Dow P., Lynch, Diane L., Shore, Derek M., Deroche-Gamonet, Véronique, Spampanato, Umberto, Revest, Jean-Michel, Maldonado, Rafael, Reggio, Patricia H., Ross, Ruth A., Marsicano, Giovanni, Piazza, Pier Vincenzo
Published in Science (American Association for the Advancement of Science) (03.01.2014)
Published in Science (American Association for the Advancement of Science) (03.01.2014)
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Journal Article
A Cannabinoid CB1 Receptor-Positive Allosteric Modulator Reduces Neuropathic Pain in the Mouse with No Psychoactive Effects
Ignatowska-Jankowska, Bogna M, Baillie, Gemma L, Kinsey, Steven, Crowe, Molly, Ghosh, Sudeshna, Owens, Robert A, Damaj, Imad M, Poklis, Justin, Wiley, Jenny L, Zanda, Matteo, Zanato, Chiara, Greig, Iain R, Lichtman, Aron H, Ross, Ruth A
Published in Neuropsychopharmacology (New York, N.Y.) (01.12.2015)
Published in Neuropsychopharmacology (New York, N.Y.) (01.12.2015)
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Journal Article
The Discovery of New Inhibitors of Insulin-Regulated Aminopeptidase by a High-Throughput Screening of 400,000 Drug-like Compounds
Gising, Johan, Honarnejad, Saman, Bras, Maaike, Baillie, Gemma L, McElroy, Stuart P, Jones, Philip S, Morrison, Angus, Beveridge, Julia, Hallberg, Mathias, Larhed, Mats
Published in International journal of molecular sciences (01.04.2024)
Published in International journal of molecular sciences (01.04.2024)
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Journal Article
The Trifluoromethyl Group as a Bioisosteric Replacement of the Aliphatic Nitro Group in CB1 Receptor Positive Allosteric Modulators
Tseng, Chih-Chung, Baillie, Gemma, Donvito, Giulia, Mustafa, Mohammed A, Juola, Sophie E, Zanato, Chiara, Massarenti, Chiara, Dall’Angelo, Sergio, Harrison, William T. A, Lichtman, Aron H, Ross, Ruth A, Zanda, Matteo, Greig, Iain R
Published in Journal of medicinal chemistry (23.05.2019)
Published in Journal of medicinal chemistry (23.05.2019)
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Journal Article
Identification of a Novel, Small Molecule Partial Agonist for the Cyclic AMP Sensor, EPAC1
Parnell, Euan, McElroy, Stuart P, Wiejak, Jolanta, Baillie, Gemma L, Porter, Alison, Adams, David R, Rehmann, Holger, Smith, Brian O, Yarwood, Stephen J
Published in Scientific reports (22.03.2017)
Published in Scientific reports (22.03.2017)
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Journal Article
Allosteric modulation of a cannabinoid G protein-coupled receptor: binding site elucidation and relationship to G protein signaling
Shore, Derek M, Baillie, Gemma L, Hurst, Dow H, Navas, 3rd, Frank, Seltzman, Herbert H, Marcu, Jahan P, Abood, Mary E, Ross, Ruth A, Reggio, Patricia H
Published in The Journal of biological chemistry (28.02.2014)
Published in The Journal of biological chemistry (28.02.2014)
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Journal Article
Allosteric Modulation of the Cannabinoid CB1 Receptor
Price, Martin R, Baillie, Gemma L, Thomas, Adèle, Stevenson, Lesley A, Easson, Morag, Goodwin, Richard, McLean, Adèle, McIntosh, Lorraine, Goodwin, Gillian, Walker, Glenn, Westwood, Paul, Marrs, Julia, Thomson, Fiona, Cowley, Phillip, Christopoulos, Arthur, Pertwee, Roger G, Ross, Ruth A
Published in Molecular pharmacology (01.11.2005)
Published in Molecular pharmacology (01.11.2005)
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Journal Article
The F238L Point Mutation in the Cannabinoid Type 1 Receptor Enhances Basal Endocytosis via Lipid Rafts
Wickert, Melanie, Hildick, Keri L, Baillie, Gemma L, Jelinek, Ruth, Aparisi Rey, Alejandro, Monory, Krisztina, Schneider, Miriam, Ross, Ruth A, Henley, Jeremy M, Lutz, Beat
Published in Frontiers in molecular neuroscience (05.07.2018)
Published in Frontiers in molecular neuroscience (05.07.2018)
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Journal Article
Phosphorylation of ezrin on Thr567 is required for the synergistic activation of cell spreading by EPAC1 and protein kinase A in HEK293T cells
Parnell, Euan, Koschinski, Andreas, Zaccolo, Manuela, Cameron, Ryan T., Baillie, George S., Baillie, Gemma L., Porter, Alison, McElroy, Stuart P., Yarwood, Stephen J.
Published in Biochimica et biophysica acta (01.07.2015)
Published in Biochimica et biophysica acta (01.07.2015)
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Journal Article
Pyrazole-type cannabinoid ligands conjugated with fluoro-deoxy-carbohydrates as potential PET-imaging agents: Synthesis and CB1/CB2 receptor affinity evaluation
Frau, Simona, Dall’Angelo, Sergio, Baillie, Gemma L., Ross, Ruth A., Pira, Marilena, Tseng, Chih-Chung, Lazzari, Paolo, Zanda, Matteo
Published in Journal of fluorine chemistry (01.08.2013)
Published in Journal of fluorine chemistry (01.08.2013)
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Journal Article
Modulation of l-α-Lysophosphatidylinositol/GPR55 Mitogen-activated Protein Kinase (MAPK) Signaling by Cannabinoids
Anavi-Goffer, Sharon, Baillie, Gemma, Irving, Andrew J., Gertsch, Jürg, Greig, Iain R., Pertwee, Roger G., Ross, Ruth A.
Published in The Journal of biological chemistry (02.01.2012)
Published in The Journal of biological chemistry (02.01.2012)
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Journal Article
CB1 Receptor Allosteric Modulators Display Both Agonist and Signaling Pathway Specificity
Baillie, Gemma L., Horswill, James G., Anavi-Goffer, Sharon, Reggio, Patricia H., Bolognini, Daniele, Abood, Mary E., McAllister, Sean, Strange, Phillip G., Stephens, Gary J., Pertwee, Roger G., Ross, Ruth A.
Published in Molecular pharmacology (01.02.2013)
Published in Molecular pharmacology (01.02.2013)
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Journal Article
Synthesis and Structure‐Activity Relationships of N‐(4‐Benzamidino)‐Oxazolidinones: Potent and Selective Inhibitors of Kallikrein‐Related Peptidase 6
De Vita, Elena, Smits, Niels, Hurk, Helma, Beck, Elizabeth M., Hewitt, Joanne, Baillie, Gemma, Russell, Emily, Pannifer, Andrew, Hamon, Véronique, Morrison, Angus, McElroy, Stuart P., Jones, Philip, Ignatenko, Natalia A., Gunkel, Nikolas, Miller, Aubry K.
Published in ChemMedChem (07.01.2020)
Published in ChemMedChem (07.01.2020)
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Journal Article
4-Cyano-5-(2-thiophenyl)-pyrazoles are high affinity CB 1 receptor ligands
Altomonte, Stefano, Baillie, Gemma L., Ross, Ruth A., Zanda, Matteo
Published in RSC advances (2015)
Published in RSC advances (2015)
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Journal Article
The Trifluoromethyl Group as a Bioisosteric Replacement of the Aliphatic Nitro Group in CB 1 Receptor Positive Allosteric Modulators
Tseng, Chih-Chung, Baillie, Gemma, Donvito, Giulia, Mustafa, Mohammed A, Juola, Sophie E, Zanato, Chiara, Massarenti, Chiara, Dall'Angelo, Sergio, Harrison, William T A, Lichtman, Aron H, Ross, Ruth A, Zanda, Matteo, Greig, Iain R
Published in Journal of medicinal chemistry (23.05.2019)
Published in Journal of medicinal chemistry (23.05.2019)
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Journal Article
A critical review of both the synthesis approach and the receptor profile of the 8-chloro-1-(2′,4′-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide and analogue derivatives
Lazzari, Paolo, Distinto, Rita, Manca, Ilaria, Baillie, Gemma, Murineddu, Gabriele, Pira, Marilena, Falzoi, Matteo, Sani, Monica, Morales, Paula, Ross, Ruth, Zanda, Matteo, Jagerovic, Nadine, Pinna, Gérard Aimè
Published in European journal of medicinal chemistry (04.10.2016)
Published in European journal of medicinal chemistry (04.10.2016)
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Journal Article
A Cannabinoid CB sub(1) Receptor-Positive Allosteric Modulator Reduces Neuropathic Pain in the Mouse with No Psychoactive Effects
Ignatowska-Jankowska, Bogna M, Baillie, Gemma L, Kinsey, Steven, Crowe, Molly, Ghosh, Sudeshna, Owens, Robert A, Damaj, Imad M, Poklis, Justin, Wiley, Jenny L, Zanda, Matteo, Zanato, Chiara, Greig, Iain R, Lichtman, Aron H, Ross, Ruth A
Published in Neuropsychopharmacology (New York, N.Y.) (01.12.2015)
Published in Neuropsychopharmacology (New York, N.Y.) (01.12.2015)
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Journal Article
THE IDENTIFICATION AND CHARACTERISATION OF SMALL-MOLECULE HUMAN ABAD INHIBITORS AS THERAPEUTICS IN ALZHEIMER’S DISEASE
Aitken, Laura, Baillie, Gemma, Sethi, Ritika, Robinson, John S., Rajamanickam, Muralikrishnan, Pannifer, Andrew, Morrison, Angus, Jones, Philip S., Smith, Terry K., McElroy, Stuart P., Gunn-Moore, Frank J.
Published in Alzheimer's & dementia (01.07.2017)
Published in Alzheimer's & dementia (01.07.2017)
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