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Christoph, Thomas, Bahrenberg, Gregor, De Vry, Jean, Englberger, Werner, Erdmann, Volker A., Frech, Moritz, Kögel, Babette, Röhl, Thomas, Schiene, Klaus, Schröder, Wolfgang, Seibler, Jost, Kurreck, Jens
Published in Molecular and cellular neuroscience (01.03.2008)
Published in Molecular and cellular neuroscience (01.03.2008)
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Quantitative trait loci for obesity and insulin resistance (Nob1, Nob2) and their interaction with the leptin receptor allele (LeprA720T/T10441) in New Zealand obese mice
KLUGE, R, GIESEN, K, BAHRENBERG, G, PLUM, L, ORTLEPP, J. R, JOOST, H.-G
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Published in Diabetologia (01.12.2000)
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(223) Evidence for a combined mode of action underlying the broad efficacy profile of tapentadol, a novel centrally acting analgesic
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Published in The journal of pain (2008)
Published in The journal of pain (2008)
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A New Class of Spiegelmers Containing 2′-Fluoro-nucleotides
Helmling, S., Moyroud, E., Schroeder, W., Roehl, I., Kleinjung, F., Stark, S., Bahrenberg, G., Gillen, C., Klussmann, S., Vonhoff, S.
Published in Nucleosides, nucleotides & nucleic acids (01.10.2003)
Published in Nucleosides, nucleotides & nucleic acids (01.10.2003)
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Pyrazole C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists
Lee, Sunho, Kim, Changhoon, Ann, Jihyae, Thorat, Shivaji A., Kim, Eunhye, Park, Jongmi, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, Jeewoo
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
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4-Aminophenyl acetamides and propanamides as potent transient receptor potential vanilloid 1 (TRPV1) ligands
Kim, Changhoon, Ann, Jihyae, Lee, Sunho, Kim, Eunhye, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, Jeewoo
Published in Bioorganic & medicinal chemistry (15.08.2018)
Published in Bioorganic & medicinal chemistry (15.08.2018)
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A hydrophobic residue in position 15 of the rP2X3 receptor slows desensitization and reveals properties beneficial for pharmacological analysis and high-throughput screening
Hausmann, Ralf, Bahrenberg, Gregor, Kuhlmann, Daniel, Schumacher, Michaela, Braam, Ursula, Bieler, Dagmar, Schlusche, Ilka, Schmalzing, Günther
Published in Neuropharmacology (01.04.2014)
Published in Neuropharmacology (01.04.2014)
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Discovery of 2-(3,5-difluoro-4-methylsulfonaminophenyl)propanamides as potent TRPV1 antagonists
Kim, Changhoon, Ann, Jihyae, Lee, Sunho, Sun, Wei, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, Jeewoo
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
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t-Butyl pyridine and phenyl C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists
Lee, Sunho, Kang, Dong Wook, Ryu, HyungChul, Kim, Changhoon, Ann, Jihyae, Lee, Hobin, Kim, Eunhye, Hong, Sunhye, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, Jeewoo
Published in Bioorganic & medicinal chemistry (15.04.2017)
Published in Bioorganic & medicinal chemistry (15.04.2017)
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Molecular determinants of potent P2X2 antagonism identified by functional analysis, mutagenesis, and homology docking
Wolf, Christian, Rosefort, Christiane, Fallah, Ghada, Kassack, Matthias U, Hamacher, Alexandra, Bodnar, Mandy, Wang, Haihong, Illes, Peter, Kless, Achim, Bahrenberg, Gregor, Schmalzing, Günther, Hausmann, Ralf
Published in Molecular pharmacology (01.04.2011)
Published in Molecular pharmacology (01.04.2011)
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Salt bridge switching from Arg290/Glu167 to Arg290/ATP promotes the closed-to-open transition of the P2X2 receptor
Hausmann, Ralf, Günther, Janka, Kless, Achim, Kuhlmann, Daniel, Kassack, Matthias U, Bahrenberg, Gregor, Markwardt, Fritz, Schmalzing, Günther
Published in Molecular pharmacology (01.01.2013)
Published in Molecular pharmacology (01.01.2013)
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RNA interference-based functional knockdown of the voltage-gated potassium channel Kv7.2 in dorsal root ganglion neurons after in vitro and in vivo gene transfer by adeno-associated virus vectors
Valdor, Markus, Wagner, Anke, Röhrs, Viola, Berg, Johanna, Fechner, Henry, Schröder, Wolfgang, Tzschentke, Thomas M, Bahrenberg, Gregor, Christoph, Thomas, Kurreck, Jens
Published in Molecular pain (01.01.2018)
Published in Molecular pain (01.01.2018)
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Pyridine C-region analogs of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists
Ryu, HyungChul, Seo, Sejin, Lee, Jee-Young, Ha, Tae-Hwan, Lee, Sunho, Jung, Aeran, Ann, Jihyae, Kim, Sung-Eun, Yoon, Suyoung, Hong, Mannkyu, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Schiene, Klaus, Stockhausen, Hannelore, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo
Published in European journal of medicinal chemistry (26.03.2015)
Published in European journal of medicinal chemistry (26.03.2015)
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α-Substituted 2-(3-fluoro-4-methylsulfonamidophenyl)acetamides as potent TRPV1 antagonists
Tran, Phuong-Thao, Kim, Ho Shin, Ann, Jihyae, Kim, Sung-Eun, Kim, Changhoon, Hong, Mannkyu, Hoang, Van-Hai, Ngo, Van T.H., Hong, Sunhye, Cui, Minghua, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, Jeewoo
Published in Bioorganic & medicinal chemistry letters (01.06.2015)
Published in Bioorganic & medicinal chemistry letters (01.06.2015)
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Structure activity relationships of benzyl C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists
Ann, Jihyae, Jung, Aeran, Kim, Mi-Yeon, Kim, Hyuk-Min, Ryu, HyungChul, Kim, Sunjoo, Kang, Dong Wook, Hong, Sunhye, Cui, Minghua, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, Jeewoo
Published in Bioorganic & medicinal chemistry (01.11.2015)
Published in Bioorganic & medicinal chemistry (01.11.2015)
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2-Alkyl/alkenyl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists
Ryu, HyungChul, Seo, Sejin, Cho, Seong-Hee, Kim, Ho Shin, Jung, Aeran, Kang, Dong Wook, Son, Karam, Cui, Minghua, Hong, Sun-hye, Sharma, Pankaz Kumar, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Schiene, Klaus, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo
Published in Bioorganic & medicinal chemistry letters (15.08.2014)
Published in Bioorganic & medicinal chemistry letters (15.08.2014)
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Journal Article
2-Aryl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists
Ryu, HyungChul, Seo, Sejin, Kim, Myeong Seop, Kim, Mi-Yeon, Kim, Ho Shin, Ann, Jihyae, Tran, Phuong-Thao, Hoang, Van-Hai, Byun, Jieun, Cui, Minghua, Son, Karam, Sharma, Pankaz Kumar, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Koegel, Babette-Yvonne, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo
Published in Bioorganic & medicinal chemistry letters (15.08.2014)
Published in Bioorganic & medicinal chemistry letters (15.08.2014)
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Journal Article
6,6-Fused heterocyclic ureas as highly potent TRPV1 antagonists
Sun, Wei, Kim, Hyo-Shin, Lee, Sunho, Jung, Aeran, Kim, Sung-Eun, Ann, Jihyae, Yoon, Suyoung, Choi, Sun, Lee, Jin Hee, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Schiene, Klaus, Stockhausen, Hannelore, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo
Published in Bioorganic & medicinal chemistry letters (15.02.2015)
Published in Bioorganic & medicinal chemistry letters (15.02.2015)
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