Complex disposition of methylthioninium redox forms determines efficacy in tau aggregation inhibitor therapy for Alzheimer's disease
Baddeley, Thomas C, McCaffrey, Jennifer, Storey, John M D, Cheung, John K S, Melis, Valeria, Horsley, David, Harrington, Charles R, Wischik, Claude M
Published in The Journal of pharmacology and experimental therapeutics (01.01.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2015)
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Mitochondrial Effects of Hydromethylthionine, Rivastigmine and Memantine in Tau-Transgenic Mice
Kondak, Constantin, Leith, Michael, Baddeley, Thomas C, Santos, Renato X, Harrington, Charles R, Wischik, Claude M, Riedel, Gernot, Klein, Jochen
Published in International journal of molecular sciences (28.06.2023)
Published in International journal of molecular sciences (28.06.2023)
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A Protein Aggregation Inhibitor, Leuco-Methylthioninium Bis(Hydromethanesulfonate), Decreases α-Synuclein Inclusions in a Transgenic Mouse Model of Synucleinopathy
Schwab, Karima, Frahm, Silke, Horsley, David, Rickard, Janet E, Melis, Valeria, Goatman, Elizabeth A, Magbagbeolu, Mandy, Douglas, Morag, Leith, Michael G, Baddeley, Thomas C, Storey, John M D, Riedel, Gernot, Wischik, Claude M, Harrington, Charles R, Theuring, Franz
Published in Frontiers in molecular neuroscience (10.01.2018)
Published in Frontiers in molecular neuroscience (10.01.2018)
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HMTM-Mediated Enhancement of Brain Bioenergetics in a Mouse Tauopathy Model Is Blocked by Chronic Administration of Rivastigmine
Santos, Renato X, Melis, Valeria, Goatman, Elizabeth A, Leith, Michael, Baddeley, Thomas C, Storey, John M D, Riedel, Gernot, Wischik, Claude M, Harrington, Charles R
Published in Biomedicines (07.04.2022)
Published in Biomedicines (07.04.2022)
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Concentration-Dependent Activity of Hydromethylthionine on Cognitive Decline and Brain Atrophy in Mild to Moderate Alzheimer’s Disease
Schelter, Bjoern O., Shiells, Helen, Baddeley, Thomas C., Rubino, Christopher M., Ganesan, Harish, Hammel, Jeffrey, Vuksanovic, Vesna, Staff, Roger T., Murray, Alison D., Bracoud, Luc, Riedel, Gernot, Gauthier, Serge, Jia, Jianping, Bentham, Peter, Kook, Karin, Storey, John M.D., Harrington, Charles R., Wischik, Claude M.
Published in Journal of Alzheimer's disease (01.01.2019)
Published in Journal of Alzheimer's disease (01.01.2019)
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Concentration-Dependent Activity of Hydromethylthionine on Clinical Decline and Brain Atrophy in a Randomized Controlled Trial in Behavioral Variant Frontotemporal Dementia
Shiells, Helen, Schelter, Bjoern O., Bentham, Peter, Baddeley, Thomas C., Rubino, Christopher M., Ganesan, Harish, Hammel, Jeffrey, Vuksanovic, Vesna, Staff, Roger T., Murray, Alison D., Bracoud, Luc, Wischik, Damon J., Riedel, Gernot, Gauthier, Serge, Jia, Jianping, Moebius, Hans J., Hardlund, Jiri, Kipps, Christopher M., Kook, Karin, Storey, John M.D., Harrington, Charles R., Wischik, Claude M.
Published in Journal of Alzheimer's disease (01.01.2020)
Published in Journal of Alzheimer's disease (01.01.2020)
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Crystal structures and Hirshfeld surface analyses of the di- and tri-hydrates of (5α,17E)-17-hydrazonoandrostan-3-ol: Significant differences in the hydrogen bonding patterns and supramolecular arrangements
Gomes, Ligia R., Low, John N., Turner, Alan B., Baddeley, Thomas C., Wardell, James L.
Published in Steroids (01.12.2018)
Published in Steroids (01.12.2018)
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Crystal structures and Hirshfeld surface analyses of a des-A-B-aromatic steroidal compound, and two of its derivatives, having a trans-2,3,4,5-tetrahydro-3a-methyl-7-methoxybenz[e]indane skeleton – structural comparisons with reported tetrahydrobenz[e]indene derivatives
Gomes, Ligia R., Low, John N., Turner, Alan B., Nowicki, Alexander W., Baddeley, Thomas C., Wardell, James L.
Published in Zeitschrift für Naturforschung. B, A journal of chemical sciences (2019)
Published in Zeitschrift für Naturforschung. B, A journal of chemical sciences (2019)
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N '-(1,3-Benzo-thia-zol-2-yl)benzene-sulfono-hydrazide: crystal structure, Hirshfeld surface analysis and computational chemistry
Baddeley, Thomas C, de Souza, Marcus V N, Wardell, James L, Jotani, Mukesh M, Tiekink, Edward R T
Published in Acta crystallographica. Section E, Crystallographic communications (01.04.2019)
Published in Acta crystallographica. Section E, Crystallographic communications (01.04.2019)
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N ′-(1,3-Benzothiazol-2-yl)benzenesulfonohydrazide: crystal structure, Hirshfeld surface analysis and computational chemistry
Baddeley, Thomas C., Souza, Marcus V. N. de, Wardell, James L., Jotani, Mukesh M., Tiekink, Edward R. T.
Published in Acta crystallographica. Section E, Crystallographic communications (01.04.2019)
Published in Acta crystallographica. Section E, Crystallographic communications (01.04.2019)
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Variation in supramolecular arrangements of hydrazones, o-H2NC6H4CMeNNHC6H4X (XH, o-, m- and p-NO2), derived from o-aminoacetophenone and phenylhydrazines
Alan Howie, R., Baddeley, Thomas C., Wardell, James L., Wardell, Solange M.S.V.
Published in Journal of molecular structure (08.08.2012)
Published in Journal of molecular structure (08.08.2012)
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Tautomers and polymorphs of pyrazolinone derivatives, generated from reactions of arylhydrazines, ArNHNH2, with 1,3-dicarbonyl compounds
Baddeley, Thomas C., Howie, R. Alan, de Lima, Geraldo M., Wardell, James L., Wardell, Solange M. S. V.
Published in Zeitschrift für Kristallographie. Crystalline materials (01.02.2013)
Published in Zeitschrift für Kristallographie. Crystalline materials (01.02.2013)
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Journal Article
1,3-Diphenyl-4,5-dihydro-1H-pyrazol-5-one
Baddeley, Thomas C, Wardell, Solange M S V, Tiekink, Edward R T, Wardell, James L
Published in Acta crystallographica. Section E, Structure reports online (01.04.2012)
Published in Acta crystallographica. Section E, Structure reports online (01.04.2012)
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Co-crystallised α- and β-Anomers of 2,3,4,6-Tetra-acetyl-d-glucopyranose, in which the α- and β-Anomers are Randomly Distributed in the Hydrogen-bonded Chains of Molecules
Baddeley, Thomas C., Harrison, William T. A., Howie, R. Alan, Skakle, Janet M. S., Wardell, James L.
Published in Journal of chemical crystallography (01.12.2007)
Published in Journal of chemical crystallography (01.12.2007)
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1,2,3,4-Tetra-O-acetyl-β-d-glucopyranuronic acid monohydrate at 120 K and anhydrous 1,2,3,4-tetra-O-acetyl-β-d-glucopyranose at 292 K
Baddeley, Thomas C., Howie, R. Alan, Skakle, Janet M. S., Wardell, James L.
Published in Acta crystallographica. Section C, Crystal structure communications (01.12.2005)
Published in Acta crystallographica. Section C, Crystal structure communications (01.12.2005)
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Journal Article
1,2,3,4-Tetra-O-acetyl-β-D-glucopyranuronic acid monohydrate at 120 K and anhydrous 1,2,3,4-tetra-O-acetyl-β-D-glucopyranose at 292 K
BADDELEY, Thomas C, HOWIE, R. Alan, SKAKLE, Janet M. S, WARDELL, James L
Published in Acta crystallographica. Section C, Crystal structure communications (01.12.2005)
Published in Acta crystallographica. Section C, Crystal structure communications (01.12.2005)
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Journal Article
Crystal structures and Hirshfeld surface analyses of a des-A-B-aromatic steroidal compound, and two of its derivatives, having a trans -2,3,4,5-tetrahydro-3 a -methyl-7-methoxybenz[ e ]indane skeleton – structural comparisons with reported tetrahydrobenz[ e ]indene derivatives
Gomes, Ligia R., Low, John N., Turner, Alan B., Nowicki, Alexander W., Baddeley, Thomas C., Wardell, James L.
Published in Zeitschrift für Naturforschung. B, A journal of chemical sciences (25.09.2019)
Published in Zeitschrift für Naturforschung. B, A journal of chemical sciences (25.09.2019)
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Synthesis, potent anti-TB activity against M. tuberculosis ATTC 27294, crystal structures and complex formation of selected 2-arylidenehydrazinylbenzothiazole derivatives
Pinheiro, Alessandra.C., de Souza, Marcus.V.N., Lourenço, Maria.C.S., da Costa, Cristiane F., Baddeley, Thomas C., Low, John N., Wardell, Solange.M.S.V., Wardell, James L.
Published in Journal of molecular structure (15.02.2019)
Published in Journal of molecular structure (15.02.2019)
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