Nigratine as dual inhibitor of necroptosis and ferroptosis regulated cell death
Delehouzé, Claire, Comte, Arnaud, Leon-Icaza, Stephen Adonai, Cougoule, Céline, Hauteville, Marcelle, Goekjian, Peter, Bulinski, Jeannette Chloë, Dimanche-Boitrel, Marie-Thérèse, Meunier, Etienne, Rousselot, Morgane, Bach, Stéphane
Published in Scientific reports (24.03.2022)
Published in Scientific reports (24.03.2022)
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Journal Article
New Quinoxaline Derivatives as Dual Pim-1/2 Kinase Inhibitors: Design, Synthesis and Biological Evaluation
Oyallon, Bruno, Brachet-Botineau, Marie, Logé, Cédric, Robert, Thomas, Bach, Stéphane, Ibrahim, Sajida, Raoul, William, Croix, Cécile, Berthelot, Pascal, Guillon, Jean, Pinaud, Noël, Gouilleux, Fabrice, Viaud-Massuard, Marie-Claude, Denevault-Sabourin, Caroline
Published in Molecules (Basel, Switzerland) (06.02.2021)
Published in Molecules (Basel, Switzerland) (06.02.2021)
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New Fusarochromanone Derivatives from the Marine Fungus Fusarium equiseti UBOCC-A-117302
Pham, Giang Nam, Josselin, Béatrice, Cousseau, Arnaud, Baratte, Blandine, Dayras, Marie, Le Meur, Christophe, Debaets, Stella, Weill, Amélie, Robert, Thomas, Burgaud, Gaëtan, Probert, Ian, Abdoul-Latif, Fatouma Mohamed, Boyer, Laurent, Bach, Stéphane, Mehiri, Mohamed
Published in Marine drugs (28.09.2024)
Published in Marine drugs (28.09.2024)
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Journal Article
Design and biological evaluation of substituted 5,7-dihydro-6H-indolo[2,3-c]quinolin-6-one as novel selective Haspin inhibitors
Avula, Sreenivas, Peng, Xudan, Lang, Xingfen, Tortorella, Micky, Josselin, Béatrice, Bach, Stéphane, Bourg, Stephane, Bonnet, Pascal, Buron, Frédéric, Ruchaud, Sandrine, Routier, Sylvain, Neagoie, Cleopatra
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2022)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2022)
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Journal Article
Betulin, a Newly Characterized Compound in Acacia auriculiformis Bark, Is a Multi-Target Protein Kinase Inhibitor
Ahmadu, Augustine A., Delehouzé, Claire, Haruna, Anas, Mustapha, Lukman, Lawal, Bilqis A., Udobre, Aniefiok, Baratte, Blandine, Triscornia, Camilla, Autret, Axelle, Robert, Thomas, Bulinski, Jeannette Chloë, Rousselot, Morgane, Simoes Eugénio, Mélanie, Dimanche-Boitrel, Marie-Thérèse, Petzer, Jacobus P., Legoabe, Lesetja J., Bach, Stéphane
Published in Molecules (Basel, Switzerland) (29.07.2021)
Published in Molecules (Basel, Switzerland) (29.07.2021)
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Journal Article
Delayed treatment with systemic (S)-roscovitine provides neuroprotection and inhibits in vivo CDK5 activity increase in animal stroke models
Menn, Bénédicte, Bach, Stéphane, Blevins, Teri L, Campbell, Mark, Meijer, Laurent, Timsit, Serge
Published in PloS one (12.08.2010)
Published in PloS one (12.08.2010)
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Journal Article
Bioprospecting marine plankton
Abida, Heni, Ruchaud, Sandrine, Rios, Laurent, Humeau, Anne, Probert, Ian, De Vargas, Colomban, Bach, Stéphane, Bowler, Chris
Published in Marine Drugs (14.11.2013)
Published in Marine Drugs (14.11.2013)
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Journal Article
Book Review
Structure Activity Relationship Studies around DB18, a Potent and Selective Inhibitor of CLK Kinases
Brahmaiah, Dabbugoddu, Bhavani, Anagani Kanaka Durga, Aparna, Pasula, Kumar, Nangunoori Sampath, Solhi, Hélène, Le Guevel, Rémy, Baratte, Blandine, Robert, Thomas, Ruchaud, Sandrine, Bach, Stéphane, Jadav, Surender Singh, Reddy, Chada Raji, Mosset, Paul, Gouault, Nicolas, Levoin, Nicolas, Grée, René
Published in Molecules (Basel, Switzerland) (20.09.2022)
Published in Molecules (Basel, Switzerland) (20.09.2022)
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Journal Article
Dibenzofuran Derivatives Inspired from Cercosporamide as Dual Inhibitors of Pim and CLK1 Kinases
Dao, Viet Hung, Ourliac-Garnier, Isabelle, Logé, Cédric, McCarthy, Florence O, Bach, Stéphane, da Silva, Teresinha Gonçalves, Denevault-Sabourin, Caroline, Thiéfaine, Jérôme, Baratte, Blandine, Robert, Thomas, Gouilleux, Fabrice, Brachet-Botineau, Marie, Bazin, Marc-Antoine, Marchand, Pascal
Published in Molecules (Basel, Switzerland) (30.10.2021)
Published in Molecules (Basel, Switzerland) (30.10.2021)
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Journal Article
Synthesis and biological evaluation of selected 7-azaindole derivatives as CDK9/Cyclin T and Haspin inhibitors
Pieterse, Lianie, Legoabe, Lesetja J., Beteck, Richard M., Josselin, Béatrice, Bach, Stéphane, Ruchaud, Sandrine
Published in Medicinal chemistry research (01.08.2020)
Published in Medicinal chemistry research (01.08.2020)
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Journal Article
Kinase-Based Screening of Marine Natural Extracts Leads to the Identification of a Cytotoxic High Molecular Weight Metabolite from the Mediterranean Sponge Crambe tailliezi
Nguyen, Thi-Ngoc-Dung, Feizbakhsh, Omid, Sfecci, Estelle, Baratte, Blandine, Delehouzé, Claire, Garcia, Adrien, Moulin, Corentin, Colas, Pierre, Ruchaud, Sandrine, Mehiri, Mohamed, Bach, Stéphane
Published in Marine drugs (09.10.2019)
Published in Marine drugs (09.10.2019)
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Journal Article
Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation
Elie, Jonathan, Feizbakhsh, Omid, Desban, Nathalie, Josselin, Béatrice, Baratte, Blandine, Bescond, Amandine, Duez, Julien, Fant, Xavier, Bach, Stéphane, Marie, Dominique, Place, Matthieu, Ben Salah, Sami, Chartier, Agnes, Berteina-Raboin, Sabine, Chaikuad, Apirat, Knapp, Stefan, Carles, Fabrice, Bonnet, Pascal, Buron, Frédéric, Routier, Sylvain, Ruchaud, Sandrine
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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Journal Article
The pyrazolo[4,3-c]pyrazole core as a novel and versatile scaffold for developing dual DYRK1A-CLK1 inhibitors targeting key processes of Alzheimer's disease pathology
Bakalakou, Vaia-Argyro, Mavroidi, Barbara, Kalampaliki, Amalia D., Josselin, Béatrice, Bach, Stéphane, Skaltsounis, Alexios-Leandros, Marakos, Panagiotis, Pouli, Nicole, Pelecanou, Maria, Myrianthopoulos, Vassilios, Ruchaud, Sandrine, Kostakis, Ioannis K.
Published in European journal of medicinal chemistry reports (01.12.2024)
Published in European journal of medicinal chemistry reports (01.12.2024)
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Journal Article
Overexpression of Eimeria tenella Rhoptry Kinase 2 Induces Early Production of Schizonts
Ribeiro E Silva, Adeline, Diallo, Mamadou Amadou, Sausset, Alix, Robert, Thomas, Bach, Stéphane, Bussière, Françoise I, Laurent, Fabrice, Lacroix-Lamandé, Sonia, Silvestre, Anne
Published in Microbiology spectrum (17.08.2023)
Published in Microbiology spectrum (17.08.2023)
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Journal Article
Web Resource
The Anti- Candida albicans Agent 4-AN Inhibits Multiple Protein Kinases
Masłyk, Maciej, Janeczko, Monika, Martyna, Aleksandra, Czernik, Sławomir, Tokarska-Rodak, Małgorzata, Chwedczuk, Marta, Foll-Josselin, Béatrice, Ruchaud, Sandrine, Bach, Stéphane, Demchuk, Oleg M, Kubiński, Konrad
Published in Molecules (Basel, Switzerland) (02.01.2019)
Published in Molecules (Basel, Switzerland) (02.01.2019)
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Journal Article
Marine Natural Products from New Caledonia--A Review
Motuhi, Sofia-Eléna, Mehiri, Mohamed, Payri, Claude Elisabeth, La Barre, Stéphane, Bach, Stéphane
Published in Marine drugs (16.03.2016)
Published in Marine drugs (16.03.2016)
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Journal Article
Potassium 6-Oxo-7,13,16,22-tetraazatetracyclo[12.6.2.18,12.017,21]tricosa-1(20),8(23),9,11,14,16,18,21-octaen-2-yne-15-carboxylate
Blouet, Camille, Letast, Stéphanie, Robert, Thomas, Bach, Stéphane, Pinaud, Noël, Joubert, Nicolas, Viaud-Massuard, Marie-Claude, Guillon, Jean, Logé, Cédric, Denevault-Sabourin, Caroline
Published in MolBank (01.12.2023)
Published in MolBank (01.12.2023)
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Journal Article
Improved tumor control through circadian clock induction by seliciclib, a cyclin-dependent kinase inhibitor
IURISCI, Ida, FILIPSKI, Elisabeth, REINHARDT, Jens, BACH, Stéphane, GIANELLA-BORRADORI, Athos, IACOBELLI, Stefano, MEIJER, Laurent, LEVI, Francis
Published in Cancer research (Chicago, Ill.) (15.11.2006)
Published in Cancer research (Chicago, Ill.) (15.11.2006)
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Journal Article
Antihypertensive drug guanabenz is active in vivo against both yeast and mammalian prions
Tribouillard-Tanvier, Déborah, Béringue, Vincent, Desban, Nathalie, Gug, Fabienne, Bach, Stéphane, Voisset, Cécile, Galons, Hervé, Laude, Hubert, Vilette, Didier, Blondel, Marc
Published in PloS one (23.04.2008)
Published in PloS one (23.04.2008)
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Journal Article
Synthesis, antileishmanial activity and cytotoxicity of 2,3-diaryl- and 2,3,8-trisubstituted imidazo[1,2-a]pyrazines
Marchand, Pascal, Bazin, Marc-Antoine, Pagniez, Fabrice, Rivière, Guillaume, Bodero, Lizeth, Marhadour, Sophie, Nourrisson, Marie-Renée, Picot, Carine, Ruchaud, Sandrine, Bach, Stéphane, Baratte, Blandine, Sauvain, Michel, Pareja, Denis Castillo, Vaisberg, Abraham J., Le Pape, Patrice
Published in European journal of medicinal chemistry (20.10.2015)
Published in European journal of medicinal chemistry (20.10.2015)
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