Evaluation of Cytotoxicity and α-Glucosidase Inhibitory Activity of Amide and Polyamino-Derivatives of Lupane Triterpenoids
Kazakova, Oxana B, Giniyatullina, Gul'nara V, Mustafin, Akhat G, Babkov, Denis A, Sokolova, Elena V, Spasov, Alexander A
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Published in Molecules (Basel, Switzerland) (20.10.2020)
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6-(Tetrazol-5-yl)-7-aminoazolo[1,5- a ]pyrimidines as Novel Potent CK2 Inhibitors
Urakov, Grigoriy V, Savateev, Konstantin V, Kotovskaya, Svetlana K, Rusinov, Vladimir L, Spasov, Alexandr A, Babkov, Denis A, Sokolova, Elena V
Published in Molecules (Basel, Switzerland) (08.12.2022)
Published in Molecules (Basel, Switzerland) (08.12.2022)
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3-Arylidene-2-oxindoles as Potent NRH:Quinone Oxidoreductase 2 Inhibitors
Lozinskaya, Natalia A, Bezsonova, Elena N, Dubar, Meriam, Melekhina, Daria D, Bazanov, Daniil R, Bunev, Alexander S, Grigor'eva, Olga B, Klochkov, Vladlen G, Sokolova, Elena V, Babkov, Denis A, Spasov, Alexander A, Sosonyuk, Sergey E
Published in Molecules (Basel, Switzerland) (25.01.2023)
Published in Molecules (Basel, Switzerland) (25.01.2023)
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Anti-Inflammatory Activity of Soluble Epoxide Hydrolase Inhibitors Based on Selenoureas Bearing an Adamantane Moiety
Burmistrov, Vladimir, Morisseau, Christophe, Babkov, Denis A., Golubeva, Tatiana, Pitushkin, Dmitry, Sokolova, Elena V., Vasipov, Vladimir, Kuznetsov, Yaroslav, Bazhenov, Sergey V., Novoyatlova, Uliana S., Bondarev, Nikolay A., Manukhov, Ilya V., Osipova, Victoria, Berberova, Nadezhda, Spasov, Alexander A., Butov, Gennady M., Hammock, Bruce D.
Published in International journal of molecular sciences (14.09.2022)
Published in International journal of molecular sciences (14.09.2022)
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Ru(III) Complexes with Lonidamine-Modified Ligands
Shutkov, Ilya A, Okulova, Yulia N, Tyurin, Vladimir Yu, Sokolova, Elena V, Babkov, Denis A, Spasov, Alexander A, Gracheva, Yulia A, Schmidt, Claudia, Kirsanov, Kirill I, Shtil, Alexander A, Redkozubova, Olga M, Shevtsova, Elena F, Milaeva, Elena R, Ott, Ingo, Nazarov, Alexey A
Published in International journal of molecular sciences (15.12.2021)
Published in International journal of molecular sciences (15.12.2021)
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CK2 Inhibition and Antitumor Activity of 4,7-Dihydro-6-nitroazolo[1,5-a]pyrimidines
Lyapustin, Daniil N., Kotovskaya, Svetlana K., Butorin, Ilya I., Ulomsky, Evgeny N., Rusinov, Vladimir L., Babkov, Denis A., Pokhlebin, Alexander A., Spasov, Alexander A., Melekhin, Vsevolod V., Tokhtueva, Maria D., Shcheglova, Anna V., Makeev, Oleg G.
Published in Molecules (Basel, Switzerland) (01.08.2022)
Published in Molecules (Basel, Switzerland) (01.08.2022)
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Development of New Antimicrobial Oleanonic Acid Polyamine Conjugates
Khusnutdinova, Elmira F, Sinou, Véronique, Babkov, Denis A, Kazakova, Oxana, Brunel, Jean Michel
Published in Antibiotics (Basel) (01.01.2022)
Published in Antibiotics (Basel) (01.01.2022)
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New Organometallic Ru(II) Compounds with Lonidamine Motif as Antitumor Agents
Shutkov, Ilya A, Okulova, Yulia N, Mazur, Dmitrii M, Melnichuk, Nikolai A, Babkov, Denis A, Sokolova, Elena V, Spasov, Alexander A, Milaeva, Elena R, Nazarov, Alexey A
Published in Pharmaceutics (29.04.2023)
Published in Pharmaceutics (29.04.2023)
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α-Glucosidase Inhibitors Based on Oleanolic Acid for the Treatment of Immunometabolic Disorders
Petrova, Anastasiya V, Babkov, Denis A, Khusnutdinova, Elmira F, Baikova, Irina P, Kazakova, Oxana B, Sokolova, Elena V, Spasov, Alexander A
Published in Applied sciences (01.08.2023)
Published in Applied sciences (01.08.2023)
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Synthesis, in vitro and in vivo evaluation of 2-aryl-4H-chromene and 3-aryl-1H-benzo[f]chromene derivatives as novel α-glucosidase inhibitors
Spasov, Alexander A., Babkov, Denis A., Osipov, Dmitry V., Klochkov, Vladlen G., Prilepskaya, Diana R., Demidov, Maxim R., Osyanin, Vitaly A., Klimochkin, Yuri N.
Published in Bioorganic & medicinal chemistry letters (01.01.2019)
Published in Bioorganic & medicinal chemistry letters (01.01.2019)
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Towards multi-target antidiabetic agents: In vitro and in vivo evaluation of 3,5-disubstituted indolin-2-one derivatives as novel α-glucosidase inhibitors
Klochkov, Vladlen G., Bezsonova, Elena N., Dubar, Meriam, Melekhina, Daria D., Temnov, Victor V., Zaryanova, Ekaterina V., Lozinskaya, Natalia A., Babkov, Denis A., Spasov, Alexander A.
Published in Bioorganic & medicinal chemistry letters (01.01.2022)
Published in Bioorganic & medicinal chemistry letters (01.01.2022)
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Towards multi-target antidiabetic agents: Discovery of biphenyl-benzimidazole conjugates as AMPK activators
Babkov, Denis A., Zhukowskaya, Olga N., Borisov, Alexander V., Babkova, Valentina A., Sokolova, Elena V., Brigadirova, Anastasia A., Litvinov, Roman A., Kolodina, Alexandra A., Morkovnik, Anatolii S., Sochnev, Vadim S., Borodkin, Gennady S., Spasov, Alexander A.
Published in Bioorganic & medicinal chemistry letters (01.09.2019)
Published in Bioorganic & medicinal chemistry letters (01.09.2019)
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Synthesis and biological evaluation of 3-substituted 2-oxindole derivatives as new glycogen synthase kinase 3β inhibitors
Lozinskaya, Natalia A., Babkov, Denis A., Zaryanova, Ekaterina V., Bezsonova, Elena N., Efremov, Alexander M., Tsymlyakov, Michael D., Anikina, Lada V., Zakharyascheva, Olga Yu, Borisov, Alexander V., Perfilova, Valentina N., Tyurenkov, Ivan N., Proskurnina, Marina V., Spasov, Alexander A.
Published in Bioorganic & medicinal chemistry (01.05.2019)
Published in Bioorganic & medicinal chemistry (01.05.2019)
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Structural modifications of 2,3-indolobetulinic acid: Design and synthesis of highly potent α-glucosidase inhibitors
Khusnutdinova, Elmira F., Petrova, Anastasiya V., Thu, Ha Nguyen Thi, Tu, Anh Le Thi, Thanh, Tra Nguyen, Thi, Cham Ba, Babkov, Denis A., Kazakova, Oxana B.
Published in Bioorganic chemistry (01.07.2019)
Published in Bioorganic chemistry (01.07.2019)
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Discovery and evaluation of biphenyl derivatives of 2‐iminobenzimidazoles as prototype dual PTP1B inhibitors and AMPK activators with in vivo antidiabetic activity
Babkov, Denis A., Zhukovskaya, Olga N., Brigadirova, Anastasia A., Prilepskaya, Diana R., Kolodina, Alexandra A., Abbas, Abbas Haider S., Morkovnik, Anatolii S., Sobhia, M. Elizabeth, Ghosh, Ketan, Spasov, Alexander A.
Published in Chemical biology & drug design (01.04.2023)
Published in Chemical biology & drug design (01.04.2023)
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Synthesis and biological evaluation of 2‐acylbenzofuranes as novel α‐glucosidase inhibitors with hypoglycemic activity
Spasov, Alexander A., Babkov, Denis A., Prokhorova, Tatyana Yu, Sturova, Ekaterina A., Muleeva, Diana R., Demidov, Maxim R., Osipov, Dmitry V., Osyanin, Vitaly A., Klimochkin, Yuri N.
Published in Chemical biology & drug design (01.12.2017)
Published in Chemical biology & drug design (01.12.2017)
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Pyridoxine dipharmacophore derivatives as potent glucokinase activators for the treatment of type 2 diabetes mellitus
Dzyurkevich, Mikhail S, Babkov, Denis A, Shtyrlin, Nikita V, Mayka, Olga Yu, Iksanova, Alfiya G, Vassiliev, Pavel M, Balakin, Konstantin V, Spasov, Alexander A, Tarasov, Vadim V, Barreto, George, Shtyrlin, Yurii G, Aliev, Gjumrakch
Published in Scientific reports (22.11.2017)
Published in Scientific reports (22.11.2017)
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6‐Nitroazolo[1,5‐a]pyrimidin‐7(4H)‐ones as Antidiabetic Agents
Spasov, Alexander A., Babkov, Denis A., Sysoeva, Valentina A., Litvinov, Roman A., Shamshina, Darya D., Ulomsky, Evgeny N., Savateev, Konstantin V., Fedotov, Viktor V., Slepukhin, Pavel A., Chupakhin, Oleg N., Charushin, Valery N., Rusinov, Vladimir L.
Published in Archiv der Pharmazie (Weinheim) (01.12.2017)
Published in Archiv der Pharmazie (Weinheim) (01.12.2017)
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Toward the discovery of dual HCMV–VZV inhibitors: Synthesis, structure activity relationship analysis, and cytotoxicity studies of long chained 2-uracil-3-yl-N-(4-phenoxyphenyl)acetamides
Babkov, Denis A., Khandazhinskaya, Anastasia L., Chizhov, Alexander O., Andrei, Graciela, Snoeck, Robert, Seley-Radtke, Katherine L., Novikov, Mikhail S.
Published in Bioorganic & medicinal chemistry (01.11.2015)
Published in Bioorganic & medicinal chemistry (01.11.2015)
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Synthesis and Evaluation of Novel [1,2,4]Triazolo[5,1‐c][1,2,4]‐triazines and Pyrazolo[5,1‐c][1,2,4]triazines as Potential Antidiabetic Agents
Rusinov, Vladimir L., Sapozhnikova, Irina M., Bliznik, Anastasiya M., Chupakhin, Oleg N., Charushin, Valery N., Spasov, Alexander A., Vassiliev, Pavel M., Kuznetsova, Valentina A., Rashchenko, Andrey I., Babkov, Denis A.
Published in Archiv der Pharmazie (Weinheim) (01.05.2017)
Published in Archiv der Pharmazie (Weinheim) (01.05.2017)
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