Synthesis and biological activity of oxo-7H-benzo[E]perimidine-4-carboxylic acid derivatives as potent, nonpeptide corticotropin releasing factor (CRF) receptor antagonists
LUTHIN, D. R, RABINOVICH, A. K, BHUMRALKAR, D. R, YOUNGBLOOD, K. L, BYCHOWSKI, R. A, DHANOA, D. S, MAY, J. M
Published in Bioorganic & medicinal chemistry letters (08.03.1999)
Published in Bioorganic & medicinal chemistry letters (08.03.1999)
Get full text
Journal Article
NICHTPEPTIDISCHE ANTAGONISTEN DES GLP-1 REZEPTORS UND VERWENDUNGSMETHODEN
CHOU, TSO-SHENG, BYCHOWSKI, A, LING, L, KUKI, ATSUO, KIEL, DAN, HONG, YUFENG, DHANOA, S, TRUESDALE, KENNETH, GONZALEZ, JAVIER, GREGOR, EDWARD, RAJAPAKSE, JAGATH, TENG, MIN, JOHNSON, DAVID
Year of Publication 23.06.2005
Get full text
Year of Publication 23.06.2005
Patent
Synthesis and biological activity of oxo-7 H-benzo[ e]perimidine-4-carboxylic acid derivatives as potent, nonpeptide corticotropin releasing factor (CRF) receptor antagonists
Luthin, David R, Rabinovich, Aleksandr K, Bhumralkar, Dilip R, Youngblood, Kenna L, Bychowski, Richard A, Dhanoa, Daljit S, May, John M
Published in Bioorganic & medicinal chemistry letters (1999)
Published in Bioorganic & medicinal chemistry letters (1999)
Get full text
Journal Article
Benzoperimidine-carboxylic acids and derivatives thereof
DAVID R. LUTHIN, DILIP R. BHUMRALKAR, RICHARD A. BYCHOWSKI, ALEKSANDR K. RABINOVICH, DALE S. DHANOA
Year of Publication 19.03.1998
Get full text
Year of Publication 19.03.1998
Patent
Non-peptide antagonists of GLP-1 receptor and methods of use
ATSUO KUKI, LARRY KENNETH TRUESDALE, MIN TENG, RICHARD A. BYCHOWSKI, TSO-SHENG CHOU, VLAD EDWARD GREGOR, RANJAN JAGATH RAJAPAKSE, MICHAEL DAVID JOHNSON, ANTHONY L. LING, JAVIER GONZALEZ, DAN KIEL, DALJIT S. DHANOA, YUFENG HONG
Year of Publication 03.04.2003
Get full text
Year of Publication 03.04.2003
Patent
Non-peptide antagonists of GLP-1 receptor and methods of use
ATSUO KUKI, LARRY KENNETH TRUESDALE, MIN TENG, RICHARD A. BYCHOWSKI, TSO-SHENG CHOU, VLAD EDWARD GREGOR, RANJAN JAGATH RAJAPAKSE, MICHAEL DAVID JOHNSON, ANTHONY L. LING, JAVIER GONZALEZ, DAN KIEL, DALJIT S. DHANOA, YUFENG HONG
Year of Publication 21.05.2002
Get full text
Year of Publication 21.05.2002
Patent
Non-peptide antagonists of glp-1 receptor and methods of use
ATSUO KUKI, LARRY KENNETH TRUESDALE, MIN TENG, RICHARD A. BYCHOWSKI, TSO-SHENG CHOU, VLAD EDWARD GREGOR, RANJAN JAGATH RAJAPAKSE, MICHAEL DAVID JOHNSON, ANTHONY L. LING, JAVIER GONZALEZ, DAN KIEL, DALJIT S. DHANOA, YUFENG HONG
Year of Publication 26.06.2000
Get full text
Year of Publication 26.06.2000
Patent
Compostos antagonistas de receptores não peptìdicos de glp-1, seus derivados, composto útil derivado dos mesmos, composição farmacêutica, método para regular a secreção de insulina em mamìferos, método de inibição da atividade de glp-1, método de inibição da ligação de glp-1 ao receptor de glp-1 e método de inibição da ativação do receptor de glp-1
ATSUO KUKI, LARRY KENNETH TRUESDALE, MIN TENG, RICHARD A. BYCHOWSKI, TSO-SHENG CHOU, VLAD EDWARD GREGOR, RANJAN JAGATH RAJAPAKSE, MICHAEL DAVID JOHNSON, ANTHONY L. LING, JAVIER GONZALEZ, DAN KIEL, DALJIT S. DHANOA, YUFENG HONG
Year of Publication 06.11.2001
Get full text
Year of Publication 06.11.2001
Patent
Benzoperimidine-carboxylic acids and derivatives thereof
LUTHIN; DAVID R, BHUMRALKAR; DILIP R, DHANOA; DALE S, BYCHOWSKI; RICHARD A, RABINOVICH; ALEKSANDR K
Year of Publication 19.01.1999
Get full text
Year of Publication 19.01.1999
Patent
BENZOPERIMIDINE-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF
RABINOVICH, ALEKSANDR, K, LUTHIN, DAVID, R, BHUMRALKAR, DILIP, R, DHANOA, DALE, S, BYCHOWSKI, RICHARD, A
Year of Publication 05.03.1998
Get full text
Year of Publication 05.03.1998
Patent
ANTAGONISTAS NAO-PEPTIDICOS DO RECEPTOR DE GLP-1 E METODOS DE UTILIZACAO
DHANOA, DALJIT, S, GREGOR, VLAD, EDWARD, CHOU, TSO-SHENG, BYCHOWSKI, RICHARD, A, JOHNSON, MICHAEL, DAVID, TRUESDALE, LARRY, KENNETH, RAJAPAKSE, RANJAN, JAGATH, LING, ANTHONY, L, KUKI, ATSUO, KIEL, DAN, GONZALEZ, JAVIER, TENG, MIN, YUFENG HONG
Year of Publication 31.05.2005
Get full text
Year of Publication 31.05.2005
Patent
NICHTPEPTIDISCHE ANTAGONISTEN DES GLP-1 REZEPTORS UND VERWENDUNGSMETHODEN
DHANOA, DALJIT, S, GREGOR, VLAD, EDWARD, CHOU, TSO-SHENG, BYCHOWSKI, RICHARD, A, JOHNSON, MICHAEL, DAVID, TRUESDALE, LARRY, KENNETH, RAJAPAKSE, RANJAN, JAGATH, LING, ANTHONY, L, KUKI, ATSUO, KIEL, DAN, HONG, YUFENG, GONZALEZ, JAVIER, TENG, MIN
Year of Publication 15.02.2005
Get full text
Year of Publication 15.02.2005
Patent
NON-PEPTIDE ANTAGONISTS OF GLP-1 RECEPTOR AND METHODS OF USE
DHANOA, DALJIT, S, GREGOR, VLAD, EDWARD, CHOU, TSO-SHENG, BYCHOWSKI, RICHARD, A, JOHNSON, MICHAEL, DAVID, TRUESDALE, LARRY, KENNETH, RAJAPAKSE, RANJAN, JAGATH, LING, ANTHONY, L, KUKI, ATSUO, KIEL, DAN, HONG, YUFENG, GONZALEZ, JAVIER, TENG, MIN
Year of Publication 02.02.2005
Get full text
Year of Publication 02.02.2005
Patent
Pyrrolo-pyridine antagonists of GLP-1 receptor
LING,ANTHONY L, CHOU, TSO-SHENG, GREGOR, VLAD EDWARD, RAJAPAKSE, RANJAN JAGATH, GONZALEZ,JAVIER, DHANOA, DALJIT S, BYCHOWSKI, RICHARD A, KUKI, ATSUO, HONG, YUFENG, IEL, DAN, RUESDALE, LARRY KENNETH, TENG, MIN, JOHNSON, MICHAEL DAVID
Year of Publication 26.09.2003
Get full text
Year of Publication 26.09.2003
Patent
Non-peptide antagonists of GLP-1 receptor and methods of use
JOHNSON MICHAEL DAVID, GREGOR VLAD EDWARD, KIEL DAN, DHANOA DALJIT S, CHOU TSO-SHENG, LING ANTHONY L, TENG MIN, BYCHOWSKI RICHARD A, GONZALEZ JAVIER, RAJAPAKSE RANJAN JAGATH, TRUESDALE LARRY KENNETH, KUKI ATSUO, HONG YUFENG
Year of Publication 22.10.2002
Get full text
Year of Publication 22.10.2002
Patent