Pharmacological comparison of muscarinic ligands : Historical versus more recent muscarinic M1-preferring receptor agonists
HEINRICH, Julia N, BUTERA, John A, TSENG, Eugene, UVEGES, Albert J, MAYER, Scott C, CARRICK, Tikva, KRAMER, Angela, KOWAL, Dianne, LOCK, Tim, MARQUIS, Karen L, PAUSCH, Mark H, POPIOLEK, Mike, SUN, Shaiu-Ching
Published in European journal of pharmacology (01.03.2009)
Published in European journal of pharmacology (01.03.2009)
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Journal Article
Synthesis and bladder smooth muscle relaxing properties of substituted 3-amino-4-aryl-(and aralkyl-)cyclobut-3-ene-1,2-diones
Butera, John A., Jenkins, Douglas J., Lennox, Joseph R., Sheldon, Jeffrey H., Norton, N. Wesley, Warga, Dawn, Argentieri, Thomas M.
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
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Journal Article
Identification of pyridazino[4,5- b]indolizines as selective PDE4B inhibitors
Donnell, Andrew F., Dollings, Paul J., Butera, John A., Dietrich, Arlene J., Lipinski, Kerri K., Ghavami, Afshin, Hirst, Warren D.
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
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Journal Article
Novel progesterone receptor modulators with gene selective and context-dependent partial agonism
Berrodin, Thomas J., Jelinsky, Scott A., Graciani, Nilsa, Butera, John A., Zhang, Zhiming, Nagpal, Sunil, Winneker, Richard C., Yudt, Matthew R.
Published in Biochemical pharmacology (15.01.2009)
Published in Biochemical pharmacology (15.01.2009)
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Journal Article
Prodrugs of Perzinfotel with Improved Oral Bioavailability
Baudy, Reinhardt B, Butera, John A, Abou-Gharbia, Magid A, Chen, Hong, Harrison, Boyd, Jain, Uday, Magolda, Ronald, Sze, Jean Y, Brandt, Michael R, Cummons, Terri A, Kowal, Diane, Pangalos, Menelas N, Zupan, Bojana, Hoffmann, Matthew, May, Michael, Mugford, Cheryl, Kennedy, Jeffrey, Childers, Wayne E
Published in Journal of medicinal chemistry (12.02.2009)
Published in Journal of medicinal chemistry (12.02.2009)
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Journal Article
Design, Synthesis, and Biological Evaluation of Thio-Containing Compounds with Serum HDL-Cholesterol-Elevating Properties
Elokdah, Hassan, Sulkowski, Theodore S, Abou-Gharbia, Magid, Butera, John A, Chai, Sie-Yearl, McFarlane, Geraldine R, McKean, Mar-Lee, Babiak, John L, Adelman, Steven J, Quinet, Elaine M
Published in Journal of medicinal chemistry (29.01.2004)
Published in Journal of medicinal chemistry (29.01.2004)
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Journal Article
Discovery of a class of potent gap-junction modifiers as novel antiarrhythmic agents
Piatnitski Chekler, Eugene L., Butera, John A., Di, Li, Swillo, Robert E., Morgan, Gwen A., Rossman, Eric I., Huselton, Christine, Larsen, Bjarne D., Hennan, James K.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
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Journal Article
Synthesis and potassium channel opening activity of substituted 10H-benzo[4,5]furo[3,2-b]indole- and 5,10-dihydro-indeno[1,2-b]indole-1-carboxylic acids
BUTERA, John A, ANTANE, Schuyler A, HIRTH, Bradford, LENNOX, Joseph R, SHELDON, Jeffrey H, NORTON, N. Wesley, WARGA, Dawn, ARGENTIERI, Thomas M
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
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Journal Article
Discovery of (2S,4R)-1-(2-Aminoacetyl)-4-benzamidopyrrolidine-2-carboxylic Acid Hydrochloride (GAP-134)13, an Orally Active Small Molecule Gap-Junction Modifier for the Treatment of Atrial Fibrillation
Butera, John A, Larsen, Bjarne Due, Hennan, James K, Kerns, Edward, Di, Li, Alimardanov, Asaf, Swillo, Robert E, Morgan, Gwen A, Liu, Kun, Wang, Qiang, Rossman, Eric I, Unwalla, Rayomand, McDonald, Leonard, Huselton, Christine, Petersen, Jørgen S
Published in Journal of medicinal chemistry (26.02.2009)
Published in Journal of medicinal chemistry (26.02.2009)
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Journal Article
Ion channel screening plates: design, construction, and maintenance
Mayer, Scott C, Butera, John A, Diller, David J, Dunlop, John, Ellingboe, John, Fan, Kristi Yi, Kaftan, Edward, Mekonnen, Belew, Mobilio, Dominick, Paslay, Jeff, Tawa, Gregory, Vasilyev, Dmitry, Bowlby, Mark R
Published in Assay and drug development technologies (01.08.2010)
Published in Assay and drug development technologies (01.08.2010)
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Journal Article
Synthesis and selective class III antiarrhythmic activity of novel N-heteroaralkyl-substituted 1-(aryloxy)-2-propanolamine and related propylamine derivatives
Butera, John A, Spinelli, Walter, Anantharaman, Viji, Marcopulos, Nicholas, Parsons, Roderick W, Moubarak, Issam F, Cullinan, Catherine, Bagli, Jehan F
Published in Journal of medicinal chemistry (01.11.1991)
Published in Journal of medicinal chemistry (01.11.1991)
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Journal Article
Comparison of the Potassium Channel Openers, WAY-133537, ZD6169, and Celikalim on Isolated Bladder Tissue and In Vivo Bladder Instability in Rat
Wojdan, A, Freeden, C, Woods, M, Oshiro, G, Spinelli, W, Colatsky, T J, Sheldon, J H, Norton, N W, Warga, D, Antane, M M, Antane, S A, Butera, J A, Argentieri, T M
Published in The Journal of pharmacology and experimental therapeutics (01.06.1999)
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Published in The Journal of pharmacology and experimental therapeutics (01.06.1999)
Journal Article
Design and SAR of Novel Potassium Channel Openers Targeted for Urge Urinary Incontinence. 1. N-Cyanoguanidine Bioisosteres Possessing in Vivo Bladder Selectivity
Butera, John A, Antane, Madelene M, Antane, Schuyler A, Argentieri, Thomas M, Freeden, Chris, Graceffa, Russell F, Hirth, Bradford H, Jenkins, Douglas, Lennox, Joseph R, Matelan, Edward, Norton, N. Wesley, Quagliato, Dominick, Sheldon, Jeffrey H, Spinelli, Walter, Warga, Dawn, Wojdan, Alexandra, Woods, Morgan
Published in Journal of medicinal chemistry (23.03.2000)
Published in Journal of medicinal chemistry (23.03.2000)
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Journal Article
Design and SAR of Novel Potassium Channel Openers Targeted for Urge Urinary Incontinence. 2. Selective and Potent Benzylamino Cyclobutenediones
Gilbert, Adam M, Antane, Madelene M, Argentieri, Thomas M, Butera, John A, Francisco, Gerardo D, Freeden, Chris, Gundersen, Eric G, Graceffa, Russell F, Herbst, David, Hirth, Bradford H, Lennox, Joseph R, McFarlane, Geraldine, Norton, N. Wesley, Quagliato, Dominick, Sheldon, Jeffrey H, Warga, Dawn, Wojdan, Alexandra, Woods, Morgan
Published in Journal of medicinal chemistry (23.03.2000)
Published in Journal of medicinal chemistry (23.03.2000)
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Journal Article
Synthesis and potassium channel opening activity of substituted 10H-Benzofuro[3,2-b]indole- and 5,10-Dihydro-indeno[1,2-b]indole-1-carboxylic acids
Butera, John A., Antane, Schuyler A., Hirth, Bradford, Lennox, Joseph R., Sheldon, Jeffrey H., Norton, N.Wesley, Warga, Dawn, Argentieri, Thomas M.
Published in Bioorganic & medicinal chemistry letters (01.08.2001)
Published in Bioorganic & medicinal chemistry letters (01.08.2001)
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Journal Article
Pharmacological comparison of muscarinic ligands: Historical versus more recent muscarinic M 1-preferring receptor agonists
Heinrich, Julia N., Butera, John A., Carrick, Tikva, Kramer, Angela, Kowal, Dianne, Lock, Tim, Marquis, Karen L., Pausch, Mark H., Popiolek, Mike, Sun, Shaiu-Ching, Tseng, Eugene, Uveges, Albert J., Mayer, Scott C.
Published in European journal of pharmacology (01.03.2009)
Published in European journal of pharmacology (01.03.2009)
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Journal Article