Chiral N super(G)-acylated hetarylpropylguanidine-type histamine H sub(2) receptor agonists do not show significant stereoselectivity
Ghorai, Prasanta, Kraus, Anja, Birnkammer, Tobias, Geyer, Roland, Bernhardt, Guenther, Dove, Stefan, Seifert, Roland, Elz, Sigurd, Buschauer, Armin
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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Synthesis and pharmacological characterization of novel fluorescent histamine H 2-receptor ligands derived from aminopotentidine
Xie, Sheng-Xue, Petrache, Georgiana, Schneider, Erich, Ye, Qi-Zhuang, Bernhardt, Günther, Seifert, Roland, Buschauer, Armin
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
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Guanidine−Acylguanidine Bioisosteric Approach in the Design of Radioligands: Synthesis of a Tritium-Labeled NG-Propionylargininamide ([3H]-UR-MK114) as a Highly Potent and Selective Neuropeptide Y Y1 Receptor Antagonist
KELLER, Max, POP, Nathalie, HUTZLER, Christoph, BECK-SICKINGER, Annette G., BERNHARDT, Günther, BUSCHAUER, Armin
Published in Journal of medicinal chemistry (25.12.2008)
Published in Journal of medicinal chemistry (25.12.2008)
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N(ω)-Carbamoylation of the Argininamide Moiety: An Avenue to Insurmountable NPY Y1 Receptor Antagonists and a Radiolabeled Selective High-Affinity Molecular Tool ([(3)H]UR-MK299) with Extended Residence Time
Keller, Max, Weiss, Stefan, Hutzler, Christoph, Kuhn, Kilian K, Mollereau, Catherine, Dukorn, Stefanie, Schindler, Lisa, Bernhardt, Günther, König, Burkhard, Buschauer, Armin
Published in Journal of medicinal chemistry (25.11.2015)
Published in Journal of medicinal chemistry (25.11.2015)
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Luciferase Reporter Gene Assay on Human, Murine and Rat Histamine H4 Receptor Orthologs: Correlations and Discrepancies between Distal and Proximal Readouts: e73961
Nordemann, Uwe, Wifling, David, Schnell, David, Bernhardt, Guenther, Stark, Holger, Seifert, Roland, Buschauer, Armin
Published in PloS one (01.09.2013)
Published in PloS one (01.09.2013)
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Dissociations in the Effects of beta 2-Adrenergic Receptor Agonists on cAMP Formation and Superoxide Production in Human Neutrophils: Support for the Concept of Functional Selectivity. e64556
Hummel, Irena Brunskole, Reinartz, Michael T, Kaelble, Solveig, Burhenne, Heike, Schwede, Frank, Buschauer, Armin, Seifert, Roland
Published in PloS one (01.05.2013)
Published in PloS one (01.05.2013)
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Functional Expression of the Interleukin-11 Receptor α-Chain and Evidence of Antiapoptotic Effects in Human Colonic Epithelial Cells
Kiessling, Stephan, Muller-Newen, Gerhard, Leeb, Sandra N., Hausmann, Martin, Rath, Heiko C., Strater, Jorn, Spottl, Tanja, Schlottmann, Klaus, Grossmann, Johannes, Montero-Julian, F.A., Scholmerich, Jurgen, Andus, Tilo, Buschauer, Armin, Heinrich, Peter C., Rogler, Gerhard
Published in The Journal of biological chemistry (12.03.2004)
Published in The Journal of biological chemistry (12.03.2004)
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Replacement of Thr32 and Gln34 in the C-terminal neuropeptide Y fragment 25-36 by cis-cyclobutane and cis-cyclopentane β-amino acids shifts selectivity toward the Y(4) receptor
Berlicki, Lukasz, Kaske, Melanie, Gutiérrez-Abad, Raquel, Bernhardt, Günther, Illa, Ona, Ortuño, Rosa M, Cabrele, Chiara, Buschauer, Armin, Reiser, Oliver
Published in Journal of medicinal chemistry (14.11.2013)
Published in Journal of medicinal chemistry (14.11.2013)
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Tariquidar Analogues: Synthesis by Cu I ‐Catalysed N/O–Aryl Coupling and Inhibitory Activity against the ABCB1 Transporter
Egger, Michael, Li, Xuqin, Müller, Christine, Bernhardt, Günther, Buschauer, Armin, König, Burkhard
Published in European journal of organic chemistry (01.06.2007)
Published in European journal of organic chemistry (01.06.2007)
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Fluorescence- and luminescence-based methods for the determination of affinity and activity of neuropeptide Y sub(2) receptor ligands
Ziemek, Ralf, Brennauer, Albert, Schneider, Erich, Cabrele, Chiara, Beck-Sickinger, Annette G, Bernhardt, Guenther, Buschauer, Armin
Published in European journal of pharmacology (01.12.2006)
Published in European journal of pharmacology (01.12.2006)
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Distinct Interaction of Human and Guinea Pig Histamine H2-Receptor with Guanidine-Type Agonists
Kelley, M T, Bürckstümmer, T, Wenzel-Seifert, K, Dove, S, Buschauer, A, Seifert, R
Published in Molecular pharmacology (01.12.2001)
Published in Molecular pharmacology (01.12.2001)
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N(G)-Acyl-argininamides as NPY Y(1) receptor antagonists: Influence of structurally diverse acyl substituents on stability and affinity
Weiss, Stefan, Keller, Max, Bernhardt, Günther, Buschauer, Armin, König, Burkhard
Published in Bioorganic & medicinal chemistry (01.09.2010)
Published in Bioorganic & medicinal chemistry (01.09.2010)
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