Search Results - "BUSCHAUER, Armin" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Structural basis of small-molecule inhibition of human multidrug transporter ABCG2

Structural basis of small-molecule inhibition of human multidrug transporter ABCG2

by Jackson, Scott M., Manolaridis, Ioannis, Kowal, Julia, Zechner, Melanie, Taylor, Nicholas M. I., Bause, Manuel, Bauer, Stefanie, Bartholomaeus, Ruben, Bernhardt, Guenther, Koenig, Burkhard, Buschauer, Armin, Stahlberg, Henning, Altmann, Karl-Heinz, Locher, Kaspar P.
Published in Nature structural & molecular biology (01.04.2018)

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The extracellular loop 2 (ECL2) of the human histamine H4 receptor substantially contributes to ligand binding and constitutive activity

The extracellular loop 2 (ECL2) of the human histamine H4 receptor substantially contributes to ligand binding and constitutive activity

by Wifling, David, Bernhardt, Günther, Dove, Stefan, Buschauer, Armin
Published in PloS one (2015)

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Structural basis of ligand binding modes at the neuropeptide Y Y1 receptor

Structural basis of ligand binding modes at the neuropeptide Y Y1 receptor

by Yang, Zhenlin, Han, Shuo, Keller, Max, Kaiser, Anette, Bender, Brian J., Bosse, Mathias, Burkert, Kerstin, Kögler, Lisa M., Wifling, David, Bernhardt, Guenther, Plank, Nicole, Littmann, Timo, Schmidt, Peter, Yi, Cuiying, Li, Beibei, Ye, Sheng, Zhang, Rongguang, Xu, Bo, Larhammar, Dan, Stevens, Raymond C., Huster, Daniel, Meiler, Jens, Zhao, Qiang, Beck-Sickinger, Annette G., Buschauer, Armin, Wu, Beili
Published in Nature (London) (01.04.2018)

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Paradoxical stimulatory effects of the "standard" histamine H4-receptor antagonist JNJ7777120: the H4 receptor joins the club of 7 transmembrane domain receptors exhibiting functional selectivity

Paradoxical stimulatory effects of the "standard" histamine H4-receptor antagonist JNJ7777120: the H4 receptor joins the club of 7 transmembrane domain receptors exhibiting functional selectivity

by Seifert, Roland, Schneider, Erich H, Dove, Stefan, Brunskole, Irena, Neumann, Detlef, Strasser, Andrea, Buschauer, Armin
Published in Molecular pharmacology (01.04.2011)

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Dimeric carbamoylguanidine-type histamine H2 receptor ligands: A new class of potent and selective agonists

Dimeric carbamoylguanidine-type histamine H2 receptor ligands: A new class of potent and selective agonists

by Kagermeier, Nicole, Werner, Kristin, Keller, Max, Baumeister, Paul, Bernhardt, Günther, Seifert, Roland, Buschauer, Armin
Published in Bioorganic & medicinal chemistry (15.07.2015)

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Potent and Selective Inhibitors of Breast Cancer Resistance Protein (ABCG2) Derived from the p-Glycoprotein (ABCB1) Modulator Tariquidar

Potent and Selective Inhibitors of Breast Cancer Resistance Protein (ABCG2) Derived from the p-Glycoprotein (ABCB1) Modulator Tariquidar

by Kühnle, Matthias, Egger, Michael, Müller, Christine, Mahringer, Anne, Bernhardt, Günther, Fricker, Gert, König, Burkhard, Buschauer, Armin
Published in Journal of medicinal chemistry (26.02.2009)

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High Affinity Agonists of the Neuropeptide Y (NPY) Y4 Receptor Derived from the C‑Terminal Pentapeptide of Human Pancreatic Polypeptide (hPP): Synthesis, Stereochemical Discrimination, and Radiolabeling

High Affinity Agonists of the Neuropeptide Y (NPY) Y4 Receptor Derived from the C‑Terminal Pentapeptide of Human Pancreatic Polypeptide (hPP): Synthesis, Stereochemical Discrimination, and Radiolabeling

by Kuhn, Kilian K, Ertl, Thomas, Dukorn, Stefanie, Keller, Max, Bernhardt, Günther, Reiser, Oliver, Buschauer, Armin
Published in Journal of medicinal chemistry (14.07.2016)

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Highly Potent, Stable, and Selective Dimeric Hetarylpropylguanidine-Type Histamine H2 Receptor Agonists

Highly Potent, Stable, and Selective Dimeric Hetarylpropylguanidine-Type Histamine H2 Receptor Agonists

by Pockes, Steffen, Wifling, David, Keller, Max, Buschauer, Armin, Elz, Sigurd
Published in ACS omega (31.03.2018)

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Synthesis and dual histamine H₁ and H₂ receptor antagonist activity of cyanoguanidine derivatives

Synthesis and dual histamine H₁ and H₂ receptor antagonist activity of cyanoguanidine derivatives

by Sadek, Bassem, Alisch, Rudi, Buschauer, Armin, Elz, Sigurd
Published in Molecules (Basel, Switzerland) (15.11.2013)

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Synthesis and Structure−Activity Relationships of Cyanoguanidine-Type and Structurally Related Histamine H4 Receptor Agonists

Synthesis and Structure−Activity Relationships of Cyanoguanidine-Type and Structurally Related Histamine H4 Receptor Agonists

by Igel, Patrick, Geyer, Roland, Strasser, Andrea, Dove, Stefan, Seifert, Roland, Buschauer, Armin
Published in Journal of medicinal chemistry (22.10.2009)

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Fluorescence- and Radiolabeling of [Lys4,Nle17,30]hPP Yields Molecular Tools for the NPY Y4 Receptor

Fluorescence- and Radiolabeling of [Lys4,Nle17,30]hPP Yields Molecular Tools for the NPY Y4 Receptor

by Dukorn, Stefanie, Littmann, Timo, Keller, Max, Kuhn, Kilian, Cabrele, Chiara, Baumeister, Paul, Bernhardt, Günther, Buschauer, Armin
Published in Bioconjugate chemistry (19.04.2017)

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Luciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readouts

Luciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readouts

by Nordemann, Uwe, Wifling, David, Schnell, David, Bernhardt, Günther, Stark, Holger, Seifert, Roland, Buschauer, Armin
Published in PloS one (2013)

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Dissociations in the effects of β2-adrenergic receptor agonists on cAMP formation and superoxide production in human neutrophils: support for the concept of functional selectivity

Dissociations in the effects of β2-adrenergic receptor agonists on cAMP formation and superoxide production in human neutrophils: support for the concept of functional selectivity

by Brunskole Hummel, Irena, Reinartz, Michael T, Kälble, Solveig, Burhenne, Heike, Schwede, Frank, Buschauer, Armin, Seifert, Roland
Published in PloS one (31.05.2013)

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[3H]UR-DE257: Development of a Tritium-Labeled Squaramide-Type Selective Histamine H2 Receptor Antagonist

[3H]UR-DE257: Development of a Tritium-Labeled Squaramide-Type Selective Histamine H2 Receptor Antagonist

by Baumeister, Paul, Erdmann, Daniela, Biselli, Sabrina, Kagermeier, Nicole, Elz, Sigurd, Bernhardt, Günther, Buschauer, Armin
Published in ChemMedChem (01.01.2015)

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Autodisplay of Human Hyaluronidase Hyal-1 on Escherichia coli and Identification of Plant-Derived Enzyme Inhibitors

Autodisplay of Human Hyaluronidase Hyal-1 on Escherichia coli and Identification of Plant-Derived Enzyme Inhibitors

by Orlando, Zoya, Lengers, Isabelle, Melzig, Matthias F, Buschauer, Armin, Hensel, Andreas, Jose, Joachim
Published in Molecules (Basel, Switzerland) (26.08.2015)

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Synthesis and Functional Characterization of Imbutamine Analogs as Histamine H3 and H4 Receptor Ligands

Synthesis and Functional Characterization of Imbutamine Analogs as Histamine H3 and H4 Receptor Ligands

by Geyer, Roland, Kaske, Melanie, Baumeister, Paul, Buschauer, Armin
Published in Archiv der Pharmazie (Weinheim) (01.02.2014)

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The Neuropeptide Y Y1 Receptor: A Diagnostic Marker? Expression in MCF-7 Breast Cancer Cells Is Down-Regulated by Antiestrogens In Vitro and in Xenografts

The Neuropeptide Y Y1 Receptor: A Diagnostic Marker? Expression in MCF-7 Breast Cancer Cells Is Down-Regulated by Antiestrogens In Vitro and in Xenografts

by Memminger, Martin, Keller, Max, Lopuch, Miroslaw, Pop, Nathalie, Bernhardt, Günther, von Angerer, Erwin, Buschauer, Armin
Published in PloS one (07.12.2012)

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G protein-coupled receptors function as logic gates for nanoparticle binding and cell uptake

G protein-coupled receptors function as logic gates for nanoparticle binding and cell uptake

by Hild, Wolfgang, Pollinger, Klaus, Caporale, Andrea, Cabrele, Chiara, Keller, Max, Pluym, Nicola, Buschauer, Armin, Rachel, Reinhard, Tessmar, Joerg, Breunig, Miriam, Goepferich, Achim, Langer, Robert
Published in Proceedings of the National Academy of Sciences - PNAS (08.06.2010)

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Structure‐Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands

Structure‐Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands

by Pockes, Steffen, Wifling, David, Buschauer, Armin, Elz, Sigurd
Published in ChemistryOpen (Weinheim) (01.03.2019)

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Expression and functional properties of canine, rat, and murine histamine H4 receptors in Sf9 insect cells

Expression and functional properties of canine, rat, and murine histamine H4 receptors in Sf9 insect cells

by Schnell, David, Brunskole, Irena, Ladova, Katerina, Schneider, Erich H., Igel, Patrick, Dove, Stefan, Buschauer, Armin, Seifert, Roland
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.05.2011)

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