Identification of a Selective Inverse Agonist for the Orphan Nuclear Receptor Estrogen-Related Receptor α
Busch, Brett B, Stevens, William C, Martin, Richard, Ordentlich, Peter, Zhou, Sihong, Sapp, Douglas W, Horlick, Robert A, Mohan, Raju
Published in Journal of medicinal chemistry (04.11.2004)
Published in Journal of medicinal chemistry (04.11.2004)
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Journal Article
Discovery of Highly Potent Liver X Receptor β Agonists
Kick, Ellen K, Busch, Brett B, Martin, Richard, Stevens, William C, Bollu, Venkataiah, Xie, Yinong, Boren, Brant C, Nyman, Michael C, Nanao, Max H, Nguyen, Lam, Plonowski, Artur, Schulman, Ira G, Yan, Grace, Zhang, Huiping, Hou, Xiaoping, Valente, Meriah N, Narayanan, Rangaraj, Behnia, Kamelia, Rodrigues, A. David, Brock, Barry, Smalley, James, Cantor, Glenn H, Lupisella, John, Sleph, Paul, Grimm, Denise, Ostrowski, Jacek, Wexler, Ruth R, Kirchgessner, Todd, Mohan, Raju
Published in ACS medicinal chemistry letters (08.12.2016)
Published in ACS medicinal chemistry letters (08.12.2016)
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Journal Article
Strategies for the modulation of phase II metabolism in a series of PKC epsilon inhibitors
Clemens, Jeremy J., Coon, Timothy, Busch, Brett B., Asgian, Juliana L., Hudson, Sarah, Termin, Andreas, Flores, Tina B., Tran, Dao, Chiang, Peggy, Sperry, Sam, Gross, Ray, Abt, Jeffrey, Heim, Roger, Lechner, Sandra, Twin, Heather, Studley, John, Brenchley, Guy, Collier, Philip N., Pierard, Francoise, Miller, Andrew, Mak, Chau, Dvornikovs, Vadims, Jimenez, Juan-Miguel, Stamos, Dean
Published in Bioorganic & medicinal chemistry letters (01.08.2014)
Published in Bioorganic & medicinal chemistry letters (01.08.2014)
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Journal Article
The Boron-Catalyzed Polymerization of Dimethylsulfoxonium Methylide. A Living Polymethylene Synthesis
Busch, Brett B, Paz, Manuel M, Shea, Kenneth J, Staiger, Chad L, Stoddard, Jonathan M, Walker, James R, Zhou, Xian-Zhi, Zhu, Huide
Published in Journal of the American Chemical Society (10.04.2002)
Published in Journal of the American Chemical Society (10.04.2002)
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Journal Article
Living Polymerization of Sulfur Ylides. Synthesis of Terminally Functionalized and Telechelic Polymethylene
Busch, Brett B, Staiger, Chad L, Stoddard, Jonathan M, Shea, Kenneth J
Published in Macromolecules (22.10.2002)
Published in Macromolecules (22.10.2002)
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Journal Article
Regulation of PPARγ Coactivator 1α (PGC-1α) Signaling by an Estrogen-Related Receptor α (ERRα) Ligand
Willy, Patricia J., Murray, Ian R., Qian, Jing, Busch, Brett B., Stevens, William C., Martin, Richard, Mohan, Raju, Zhou, Sihong, Ordentlich, Peter, Wei, Ping, Sapp, Douglas W., Horlick, Robert A., Heyman, Richard A., Schulman, Ira G., Spiegelman, Bruce M.
Published in Proceedings of the National Academy of Sciences - PNAS (15.06.2004)
Published in Proceedings of the National Academy of Sciences - PNAS (15.06.2004)
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Journal Article
Diastereoselective One-Pot Knoevenagel Condensation/Corey–Chaykovsky Cyclopropanation
Clemens, Jeremy J, Asgian, Juliana L, Busch, Brett B, Coon, Timothy, Ernst, Justin, Kaljevic, Leonard, Krenitsky, Paul J, Neubert, Timothy D, Schweiger, Edwin J, Termin, Andreas, Stamos, Dean
Published in Journal of organic chemistry (18.01.2013)
Published in Journal of organic chemistry (18.01.2013)
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Journal Article
Materials Characterization of Alternative Gate Dielectrics
Busch, Brett W., Pluchery, Olivier, Chabal, Yves J., Muller, David A., Opila, Robert L., Raynien Kwo, J., Garfunkel, Eric
Published in MRS bulletin (01.03.2002)
Published in MRS bulletin (01.03.2002)
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Journal Article
ASGPR 세포 표면 수용체 결합 화합물 및 접합체
BUSCH BRETT BRADLEY, TURTLE ERIC D, ERNST JUSTIN THOMAS, PACKARD GARRICK K, LEWIS JASON G
Year of Publication 20.03.2024
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Year of Publication 20.03.2024
Patent
세포 표면 수용체 결합 화합물 및 접합체
BUSCH BRETT BRADLEY, TURTLE ERIC D, ERNST JUSTIN THOMAS, PACKARD GARRICK K, LEWIS JASON G
Year of Publication 27.10.2022
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Year of Publication 27.10.2022
Patent
Liver X Receptor (LXR) partial agonists: Biaryl pyrazoles and imidazoles displaying a preference for LXR beta
Kick, Ellen, Martin, Richard, Xie, Yinong, Flatt, Brenton, Schweiger, Edwin, Wang, Tie-Lin, Busch, Brett, Nyman, Michael, Gu, Xiao-Hui, Yan, Grace, Wagner, Brandee, Nanao, Max, Lam Nguyen, Stout, Thomas, Plonowski, Artur, Schulman, Ira, Ostrowski, Jacek, Kirchgessner, Todd, Wexler, Ruth, Mohan, Raju
Published in Bioorganic & medicinal chemistry letters (15.01.2015)
Published in Bioorganic & medicinal chemistry letters (15.01.2015)
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Journal Article
MACROCYCLIC MOLECULES AS MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR, PHARMACEUTICAL COMPOSITIONS THEREOF, USE THEREOF IN TREATMENT OF CYSTIC FIBROSIS, AND PRODUCTION METHOD THEREOF
ZHOU JINGLAN, ANTON V GULEVICH, HARIPADA KATSUYA, MCCARTNEY JASON, JEREMY J CLEMENS, CARL V VOGEL, PETER GROOTENHUIS, SARA SABINA HADIDA RUAH, KANG PING, MARK THOMAS MILLER, FABRICE PIERRE, FREEMAN BRIAN, PRASUNA PARASELLI, CHEN WEICHAO G, TIMOTHY RICHARD COON, COREY DON ANDERSON, THOMAS CLEVELAND, ALEXANDER RUSSELL ABELA, CLARA KUANG-JU HSIA, SENAIT G GHIRMAI, SARA E SWIFT, ANDREAS TERMIN, JOHNNY UY, BUSCH BRETT B
Year of Publication 10.04.2024
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Year of Publication 10.04.2024
Patent
낭성 섬유증 막관통 전도도 조절자의 조절제
HADIDA RUAH SARA SABINA, GHIRMAI SENAIT G, ZHOU JINGLAN, BOOKSER BRETT C, PIERRE FABRICE, MCCARTNEY JASON, VOGEL CARL V, PARASELLI PRASUNA, CLEVELAND THOMAS, KHATUYA HARIPADA, UY JOHNNY, ABELA ALEXANDER RUSSELL, SWIFT SARA E, MILLER MARK THOMAS, TERMIN ANDREAS, GROOTENHUIS PETER, ANDERSON COREY DON, FRIEMAN BRYAN, COON TIMOTHY RICHARD, BUSCH BRETT B, CLEMENS JEREMY J, GULEVICH ANTON V, ISHIHARA YOSHIHIRO
Year of Publication 24.05.2022
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Year of Publication 24.05.2022
Patent
낭포성 섬유증 막관통 전도성 조절인자의 조절제로서의 매크로사이클, 그의 약제학적 조성물, 낭포성 섬유증의 치료에서의 그의 용도, 및 그의 제조 방법
HADIDA RUAH SARA SABINA, GHIRMAI SENAIT G, ZHOU JINGLAN, CHEN WEICHAO GEORGE, PIERRE FABRICE, MCCARTNEY JASON, VOGEL CARL V, PARASELLI PRASUNA, CLEVELAND THOMAS, KHATUYA HARIPADA, UY JOHNNY, ABELA ALEXANDER RUSSELL, KANG PING, SWIFT SARA E, MILLER MARK THOMAS, TERMIN ANDREAS, GROOTENHUIS PETER, HSIA CLARA KUANG JU, ANDERSON COREY DON, FRIEMAN BRYAN, COON TIMOTHY RICHARD, BUSCH BRETT B, CLEMENS JEREMY J, GULEVICH ANTON V
Year of Publication 23.11.2020
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Year of Publication 23.11.2020
Patent
낭포성 섬유증 막횡단 전도 조절자의 조절제, 제약 조성물, 치료 방법, 및 상기 조절제의 제조 방법
HADIDA RUAH SARA SABINA, BUSCH BRETT BRADLEY, MCCARTNEY JASON, JOSHI PRAMOD VIRUPAX, HUGHES ROBERT M, BAEK MINSON, PARASELLI PRASUNA, PIERRE FABRICE JEAN DENIS, KHATUYA HARIPADA, UY JOHNNY, KESHAVARZ SHOKRI ALI, GROOTENHUIS PETER, VAN GOOR FREDRICK, KRENITSKY PAUL JOHN, MCAULEY AOKI RACHEL, FRIEMAN BRYAN A, TERMIN ANDREAS P, SIESEL DAVID ANDREW, ZHOU JINGLAN, ANDERSON COREY, MELILLO VITO, CLEVELAND THOMAS, ALCACIO TIMOTHY, ABELA ALEXANDER RUSSELL, ZHANG BEILI, MILLER MARK THOMAS
Year of Publication 17.06.2019
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Year of Publication 17.06.2019
Patent
M6PR CELL SURFACE RECEPTOR BINDING COMPOUNDS AND CONJUGATES
PACKARD, Garrick, ERNST, Justin, BUSCH, Brett, LEWIS, Jason, TURTLE, Eric
Year of Publication 25.01.2024
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Year of Publication 25.01.2024
Patent
ASGPR CELL SURFACE RECEPTOR BINDING COMPOUNDS AND CONJUGATES
PACKARD, Garrick, ERNST, Justin, BUSCH, Brett, LEWIS, Jason, TURTLE, Eric
Year of Publication 25.01.2024
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Year of Publication 25.01.2024
Patent
ASGPR CELL SURFACE RECEPTOR BINDING COMPOUNDS AND CONJUGATES
PACKARD, Garrick, ERNST, Justin, BUSCH, Brett, LEWIS, Jason, TURTLE, Eric
Year of Publication 22.06.2023
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Year of Publication 22.06.2023
Patent
LXR MODULATORS
KICK ELLEN K, MOHAN RAJU, BOLLU VENKATAIAH, MARTIN RICHARD, BUSCH BRETT B, STEVENS WILLIAM C. JR, ZHANG HAIYING
Year of Publication 14.05.2012
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Year of Publication 14.05.2012
Patent