Pimavanserin reverses multiple measures of anxiety in a rodent model of post-traumatic stress disorder
Malin, David H., Tsai, Ping-Hsun, Campbell, Joseph R., Moreno, Georgina L., Chapman, Holly L., Suzaki, Aoi, Keivan, Mehrshad S., Gibbons, Kaitlyn M., Morales, Erica R., Burstein, Ethan S., Ward, Christopher P.
Published in European journal of pharmacology (15.01.2023)
Published in European journal of pharmacology (15.01.2023)
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Imaging the 5-HT2C receptor with PET: Evaluation of 5-HT2C and 5-HT2A affinity of pimavanserin in the primate brain
Ridler, Khanum, Rizzo, Gaia, Burstein, Ethan S, sberg Morén, Anton, Stepanov, Vladimir, Halldin, Christer, Rabiner, Eugenii A
Published in Journal of cerebral blood flow and metabolism (21.08.2024)
Published in Journal of cerebral blood flow and metabolism (21.08.2024)
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Low Dose Bexarotene Treatment Rescues Dopamine Neurons and Restores Behavioral Function in Models of Parkinson’s Disease
McFarland, Krista, Spalding, Tracy A, Hubbard, David, Ma, Jian-Nong, Olsson, Roger, Burstein, Ethan S
Published in ACS chemical neuroscience (20.11.2013)
Published in ACS chemical neuroscience (20.11.2013)
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Inverse agonists of the 5-HT2A receptor reduce nicotine withdrawal signs in rats
Malin, David, Henceroth, Mallori, Rao, Gadam Srinivas, Campbell, Joseph, Ma, Jian-Nong, Tsai, Ping-Hsun, Kishbaugh, Jordan C., Burstein, Ethan S.
Published in Neuroscience letters (20.11.2019)
Published in Neuroscience letters (20.11.2019)
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Pimavanserin, a 5HT2A receptor inverse agonist, rapidly suppresses Aβ production and related pathology in a mouse model of Alzheimer’s disease
Yuede, Carla M., Wallace, Clare E., Davis, Todd A., Gardiner, Woodrow D., Hettinger, Jane C., Edwards, Hannah M., Hendrix, Rachel D., Doherty, Brookelyn M., Yuede, Kayla M., Burstein, Ethan S., Cirrito, John R.
Published in Journal of neurochemistry (01.03.2021)
Published in Journal of neurochemistry (01.03.2021)
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Pimavanserin Promotes Trophic Factor Release and Protects Cultured Primary Dopaminergic Neurons Exposed to MPP+ in a GDNF-Dependent Manner
Lavigne, Elodie Gras, Buttigieg, Dorothée, Steinschneider, Rémy, Burstein, Ethan S
Published in ACS chemical neuroscience (16.06.2021)
Published in ACS chemical neuroscience (16.06.2021)
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The impact of pimavanserin on psychotic phenotypes and tau phosphorylation in the P301L/COMT– and rTg(P301L)4510 mouse models of Alzheimer's disease
Jimenez, Heidy, Adrien, Leslie, Wolin, Adam, Eun, John, Chang, Eric H., Burstein, Ethan S., Gomar, Jesus, Davies, Peter, Koppel, Jeremy
Published in Alzheimer's & dementia : translational research & clinical interventions (2022)
Published in Alzheimer's & dementia : translational research & clinical interventions (2022)
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Pimavanserin, a 5HT 2A receptor inverse agonist, rapidly suppresses Aβ production and related pathology in a mouse model of Alzheimer's disease
Yuede, Carla M, Wallace, Clare E, Davis, Todd A, Gardiner, Woodrow D, Hettinger, Jane C, Edwards, Hannah M, Hendrix, Rachel D, Doherty, Brookelyn M, Yuede, Kayla M, Burstein, Ethan S, Cirrito, John R
Published in Journal of neurochemistry (01.03.2021)
Published in Journal of neurochemistry (01.03.2021)
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Estrogen Receptor Beta Selective Agonists as Agents to Treat Chemotherapeutic-Induced Neuropathic Pain
Ma, Jian-Nong, McFarland, Krista, Olsson, Roger, Burstein, Ethan S
Published in ACS chemical neuroscience (21.09.2016)
Published in ACS chemical neuroscience (21.09.2016)
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Bexarotene prodrugs: Targeting through cleavage by NQO1 (DT-diaphorase)
Schafer, Anja, Burstein, Ethan S., Olsson, Roger
Published in Bioorganic & medicinal chemistry letters (15.04.2014)
Published in Bioorganic & medicinal chemistry letters (15.04.2014)
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The protease activated receptor 2 (PAR2) polymorphic variant F240S constitutively activates PAR2 receptors and potentiates responses to small-molecule PAR2 agonists
Ma, Jian-Nong, Burstein, Ethan S
Published in The Journal of pharmacology and experimental therapeutics (01.12.2013)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2013)
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Chiral Dihydrobenzofuran Acids Show Potent Retinoid X Receptor–Nuclear Receptor Related 1 Protein Dimer Activation
Sundén, Henrik, Schäfer, Anja, Scheepstra, Marcel, Leysen, Seppe, Malo, Marcus, Ma, Jian-Nong, Burstein, Ethan S, Ottmann, Christian, Brunsveld, Luc, Olsson, Roger
Published in Journal of medicinal chemistry (11.02.2016)
Published in Journal of medicinal chemistry (11.02.2016)
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Characterization of highly efficacious allosteric agonists of the human calcium-sensing receptor
Ma, Jian-Nong, Owens, Michelle, Gustafsson, Magnus, Jensen, Jacob, Tabatabaei, Ali, Schmelzer, Kara, Olsson, Roger, Burstein, Ethan S
Published in The Journal of pharmacology and experimental therapeutics (01.04.2011)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2011)
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A subtype-specific neuropeptide FF receptor antagonist attenuates morphine and nicotine withdrawal syndrome in the rat
Malin, David H., Henceroth, Mallori M., Elayoubi, Joanne, Campbell, Joseph R., Anderson, Andrea, Goyarzu, Pilar, Izygon, Jonathan, Madison, Caitlin A., Ward, Christopher P., Burstein, Ethan S.
Published in Neuroscience letters (25.09.2018)
Published in Neuroscience letters (25.09.2018)
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Ligand Dependent Switch from RXR Homo- to RXR-NURR1 Heterodimerization
Scheepstra, Marcel, Andrei, Sebastian A, de Vries, Rens M. J. M, Meijer, Femke A, Ma, Jian-Nong, Burstein, Ethan S, Olsson, Roger, Ottmann, Christian, Milroy, Lech-Gustav, Brunsveld, Luc
Published in ACS chemical neuroscience (20.09.2017)
Published in ACS chemical neuroscience (20.09.2017)
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Pharmacology of N-desmethylclozapine
Lameh, Jelveh, Burstein, Ethan S, Taylor, Eve, Weiner, David M, Vanover, Kimberly E, Bonhaus, Douglas W
Published in Pharmacology & therapeutics (Oxford) (01.08.2007)
Published in Pharmacology & therapeutics (Oxford) (01.08.2007)
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