Dual targeting of polyamine synthesis and uptake in diffuse intrinsic pontine gliomas
Khan, Aaminah, Gamble, Laura D., Upton, Dannielle H., Ung, Caitlin, Yu, Denise M. T., Ehteda, Anahid, Pandher, Ruby, Mayoh, Chelsea, Hébert, Steven, Jabado, Nada, Kleinman, Claudia L., Burns, Mark R., Norris, Murray D., Haber, Michelle, Tsoli, Maria, Ziegler, David S.
Published in Nature communications (12.02.2021)
Published in Nature communications (12.02.2021)
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Journal Article
Inhibition of polyamine synthesis and uptake reduces tumor progression and prolongs survival in mouse models of neuroblastoma
Gamble, Laura D, Purgato, Stefania, Murray, Jayne, Xiao, Lin, Yu, Denise M T, Hanssen, Kimberley M, Giorgi, Federico M, Carter, Daniel R, Gifford, Andrew J, Valli, Emanuele, Milazzo, Giorgio, Kamili, Alvin, Mayoh, Chelsea, Liu, Bing, Eden, Georgina, Sarraf, Sara, Allan, Sophie, Di Giacomo, Simone, Flemming, Claudia L, Russell, Amanda J, Cheung, Belamy B, Oberthuer, Andre, London, Wendy B, Fischer, Matthias, Trahair, Toby N, Fletcher, Jamie I, Marshall, Glenn M, Ziegler, David S, Hogarty, Michael D, Burns, Mark R, Perini, Giovanni, Norris, Murray D, Haber, Michelle
Published in Science translational medicine (30.01.2019)
Published in Science translational medicine (30.01.2019)
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Journal Article
De novo synthesis and salvage pathway coordinately regulate polyamine homeostasis and determine T cell proliferation and function
Wu, Ruohan, Chen, Xuyong, Kang, Siwen, Wang, Tingting, Gnanaprakasam, Jn Rashida, Yao, Yufeng, Liu, Lingling, Fan, Gaofeng, Burns, Mark R, Wang, Ruoning
Published in Science advances (01.12.2020)
Published in Science advances (01.12.2020)
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Journal Article
Polyamine Analogs with Xylene Rings Induce Antizyme Frameshifting, Reduce ODC Activity, and Deplete Cellular Polyamines
Petros, Lorin M, Graminski, Gerard F, Robinson, Susan, Burns, Mark R, Kisiel, Nicholas, Gesteland, Raymond F, Atkins, John F, Kramer, Debora L, Howard, Michael T, Weeks, Reitha S
Published in Journal of biochemistry (Tokyo) (01.11.2006)
Published in Journal of biochemistry (Tokyo) (01.11.2006)
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Journal Article
Lipophilic Lysine−Spermine Conjugates Are Potent Polyamine Transport Inhibitors for Use in Combination with a Polyamine Biosynthesis Inhibitor
Burns, Mark R, Graminski, Gerard F, Weeks, Reitha S, Chen, Yan, O’Brien, Thomas G
Published in Journal of medicinal chemistry (09.04.2009)
Published in Journal of medicinal chemistry (09.04.2009)
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Journal Article
Combination therapy with 2‐difluoromethylornithine and a polyamine transport inhibitor against murine squamous cell carcinoma
Chen, Yan, Weeks, Reitha S., Burns, Mark R., Boorman, David W., Klein‐Szanto, Andres, O'Brien, Thomas G.
Published in International journal of cancer (01.05.2006)
Published in International journal of cancer (01.05.2006)
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Journal Article
Polycationic Sulfonamides for the Sequestration of Endotoxin
Burns, Mark R, Jenkins, Scott A, Kimbrell, Matthew R, Balakrishna, Rajalakshmi, Nguyen, Thuan B, Abbo, Benjamin G, David, Sunil A
Published in Journal of medicinal chemistry (22.02.2007)
Published in Journal of medicinal chemistry (22.02.2007)
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Journal Article
Structural correlation between lipophilicity and lipopolysaccharide-sequestering activity in spermine-sulfonamide analogs
Burns, Mark R., Jenkins, Scott A., Vermeulen, Nicolas M., Balakrishna, Rajalakshmi, Nguyen, Thuan B., Kimbrell, Matthew R., David, Sunil A.
Published in Bioorganic & medicinal chemistry letters (15.12.2006)
Published in Bioorganic & medicinal chemistry letters (15.12.2006)
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Journal Article
Amino Acid/Spermine Conjugates: Polyamine Amides as Potent Spermidine Uptake Inhibitors
Burns, Mark R, Carlson, C. Lance, Vanderwerf, Scott M, Ziemer, Josh R, Weeks, Reitha S, Cai, Feng, Webb, Heather K, Graminski, Gerard F
Published in Journal of medicinal chemistry (25.10.2001)
Published in Journal of medicinal chemistry (25.10.2001)
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Journal Article
Structure−Activity Relationships in Lipopolysaccharide Neutralizers: Design, Synthesis, and Biological Evaluation of a 540-Membered Amphipathic Bisamide Library
Burns, Mark R, Jenkins, Scott A, Wood, Stewart J, Miller, Kelly, David, Sunil A
Published in Journal of combinatorial chemistry (01.01.2006)
Published in Journal of combinatorial chemistry (01.01.2006)
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Journal Article
Induction of apoptosis by aryl-substituted diamines: role of aromatic group substituents and distance between nitrogens
Burns, Mark R, LaTurner, Solveig, Ziemer, Josh, McVean, Maralee, Devens, Bruce, Carlson, C.Lance, Graminski, Gerard F, Vanderwerf, Scott M, Weeks, Reitha S, Carreon, Jay
Published in Bioorganic & medicinal chemistry letters (06.05.2002)
Published in Bioorganic & medicinal chemistry letters (06.05.2002)
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Journal Article
Anti-endotoxin agents. 3. Rapid identification of high-affinity lipopolysaccharide-binding compounds in a substituted polyamine library
Wood, Stewart J, Miller, Kelly A, Lushington, Gerald H, Burns, Mark R, David, Sunil A
Published in Combinatorial chemistry & high throughput screening (01.01.2006)
Published in Combinatorial chemistry & high throughput screening (01.01.2006)
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Journal Article
Synthesis of bis-spermine dimers that are potent polyamine transport inhibitors
Graminski, Gerard F., Carlson, C.Lance, Ziemer, Josh R., Cai, Feng, Vermeulen, Nicolaas M.J., Vanderwerf, Scott M., Burns, Mark R.
Published in Bioorganic & medicinal chemistry letters (07.01.2002)
Published in Bioorganic & medicinal chemistry letters (07.01.2002)
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Journal Article