Efficient Preparation of ((3-Chloro-2-fluoro-phenyl)-[7-methoxy-8-(3-morpholin-4-yl-propoxy)-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo(a,d)cyclohepten-1-yl]-amine) for In-Vivo Study
Liu, Hu, Smith, Leon M., Mao, Yunyu, Pan, Weitao, Xu, Yong-Jiang, Burdzovic-Wizeman, Sabina, Duncton, Matthew A. J., Wong, Wai C.
Published in Synthetic communications (01.01.2006)
Published in Synthetic communications (01.01.2006)
Get full text
Journal Article
Preparation of Substituted Pyrimido[4,5-b]-1,4-benzoxazepines, Thiazepines, and Diazepines via a Pictet-Spengler Cyclization
Duncton, Matthew A. J., Smith, Leon M. II, Burdzovic-Wizeman, Sabina, Burns, Aaron, Liu, Hu, Mao, Yunyu, Wong, Wai C., Kiselyov, Alexander S.
Published in ChemInform (28.03.2006)
Published in ChemInform (28.03.2006)
Get full text
Journal Article
Novel tricyclic azepine derivatives: Biological evaluation of pyrimido[4,5- b]-1,4-benzoxazepines, thiazepines, and diazepines as inhibitors of the epidermal growth factor receptor tyrosine kinase
Smith, Leon, Wong, Wai C., Kiselyov, Alexander S., Burdzovic-Wizemann, Sabina, Mao, Yunyu, Xu, Yongjiang, Duncton, Matthew A.J., Kim, Ki, Piatnitski, Evgueni L., Doody, Jacqueline F., Wang, Ying, Rosler, Robin L., Milligan, Daniel, Columbus, John, Balagtas, Chris, Lee, Sui Ping, Konovalov, Andrey, Hadari, Yaron R.
Published in Bioorganic & medicinal chemistry letters (01.10.2006)
Published in Bioorganic & medicinal chemistry letters (01.10.2006)
Get full text
Journal Article
Efficient Preparation of ((3-Chloro-2-fluorophenyl)- [7-methoxy-8- (3-morpholin-4-yl-propoxy)-10,11-dihydro-5-oxa-2,4,11-triazadibenzo (a,d)cyclohepten-1-yl]amine) for in vivo Study
Liu, Hu, Smith, Leon M. II, Mao, Yunyu, Pan, Weitao, Xu, Yong-Jiang, Burdzovic-Wizeman, Sabina, Duncton, Matthew A. J., Wong, Wai C.
Published in ChemInform (06.06.2006)
Published in ChemInform (06.06.2006)
Get full text
Journal Article
Preparation of Substituted Pyrimido[4,5-b]-1,4-benzoxazepines, Thiazepines, and Diazepines via a Pictet−Spengler Cyclization
Duncton, Matthew A. J, Smith, Leon M, Burdzovic-Wizeman, Sabina, Burns, Aaron, Liu, Hu, Mao, Yunyu, Wong, Wai C, Kiselyov, Alexander S
Published in Journal of organic chemistry (11.11.2005)
Published in Journal of organic chemistry (11.11.2005)
Get full text
Journal Article
Tricyclic azepine derivatives: Pyrimido[4,5-b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitors
Smith, Leon, Piatnitski, Evgueni L., Kiselyov, Alexander S., Ouyang, Xiaohu, Chen, Xiaoling, Burdzovic-Wizemann, Sabina, Xu, Yongjiang, Wang, Ying, Rosler, Robin L., Patel, Sheetal N., Chiang, Hui-Hsien, Milligan, Daniel L., Columbus, John, Wong, Wai C., Doody, Jacqueline F., Hadari, Yaron R.
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Get full text
Journal Article
Corrigendum to “Tricyclic azepine derivatives: Pyrimido[4,5- b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitors” [Bioorg. Med. Chem. Lett. 16 (2006) 1643–1646]
Smith, Leon, Piatnitski, Evgueni L., Kiselyov, Alexander S., Ouyang, Xiaohu, Chen, Xiaoling, Burdzovic-Wizemann, Sabina, Xu, Yongjiang, Pan, Weitao, Chen, Xin, Wang, Ying, Rosler, Robin L., Patel, Sheetal N., Chiang, Hui-Hsien, Milligan, Daniel L., Columbus, John, Wong, Wai C., Doody, Jacqueline F., Hadari, Yaron R.
Published in Bioorganic & medicinal chemistry letters (15.07.2006)
Published in Bioorganic & medicinal chemistry letters (15.07.2006)
Get full text
Journal Article