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Reeves, Jonathan T, Malapit, Christian A, Buono, Frederic G, Sidhu, Kanwar P, Marsini, Maurice A, Sader, C. Avery, Fandrick, Keith R, Busacca, Carl A, Senanayake, Chris H
Published in Journal of the American Chemical Society (29.07.2015)
Published in Journal of the American Chemical Society (29.07.2015)
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Shee, Yu, Li, Haote, Zhang, Pengpeng, Nikolic, Andrea M, Lu, Wenxin, Kelly, H Ray, Manee, Vidhyadhar, Sreekumar, Sanil, Buono, Frederic G, Song, Jinhua J, Newhouse, Timothy R, Batista, Victor S
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Published in Nature communications (06.09.2024)
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Autonomous Multi‐Step and Multi‐Objective Optimization Facilitated by Real‐Time Process Analytics
Sagmeister, Peter, Ort, Florian F., Jusner, Clemens E., Hebrault, Dominique, Tampone, Thomas, Buono, Frederic G., Williams, Jason D., Kappe, C. Oliver
Published in Advanced science (01.04.2022)
Published in Advanced science (01.04.2022)
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Carbamoyl Anion Addition to Azirines
Kerner, Michael J, Kuttruff, Christian A, Chevliakov, Maxim, Buono, Frederic G, Gao, Donghong A, Krawiec, Mariusz, Busacca, Carl A, Senanayake, Chris H, Wipf, Peter, Reeves, Jonathan T
Published in Organic letters (04.06.2021)
Published in Organic letters (04.06.2021)
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A Slug Flow Platform with Multiple Process Analytics Facilitates Flexible Reaction Optimization
Wagner, Florian, Sagmeister, Peter, Jusner, Clemens E., Tampone, Thomas G., Manee, Vidhyadhar, Buono, Frederic G., Williams, Jason D., Kappe, C. Oliver
Published in Advanced science (01.04.2024)
Published in Advanced science (01.04.2024)
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Sequential C–H Arylation and Enantioselective Hydrogenation Enables Ideal Asymmetric Entry to the Indenopiperidine Core of an 11β-HSD‑1 Inhibitor
Wei, Xudong, Qu, Bo, Zeng, Xingzhong, Savoie, Jolaine, Fandrick, Keith R, Desrosiers, Jean-Nicolas, Tcyrulnikov, Sergei, Marsini, Maurice A, Buono, Frederic G, Li, Zhibin, Yang, Bing-Shiou, Tang, Wenjun, Haddad, Nizar, Gutierrez, Osvaldo, Wang, Jun, Lee, Heewon, Ma, Shengli, Campbell, Scot, Lorenz, Jon C, Eckhardt, Matthias, Himmelsbach, Frank, Peters, Stefan, Patel, Nitinchandra D, Tan, Zhulin, Yee, Nathan K, Song, Jinhua J, Roschangar, Frank, Kozlowski, Marisa C, Senanayake, Chris H
Published in Journal of the American Chemical Society (30.11.2016)
Published in Journal of the American Chemical Society (30.11.2016)
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Scalable copper‐catalyzed preparation of imidazopyridinones from iodopyridinyl ureas
Rugg, Kyle W., Balk, Regina C., Paolillo, Joshua M., Yerkozhanov, Dauzhan, Tampone, Thomas G., Holan, Martin, Buono, Frederic G., Reeves, Jonathan T.
Published in Journal of heterocyclic chemistry (01.02.2023)
Published in Journal of heterocyclic chemistry (01.02.2023)
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Development of a concise, scalable synthesis of a CCR1 antagonist utilizing a continuous flow Curtius rearrangement
Marsini, Maurice A, Buono, Frederic G, Lorenz, Jon C, Yang, Bing-Shiou, Reeves, Jonathan T, Sidhu, Kanwar, Sarvestani, Max, Tan, Zhulin, Zhang, Yongda, Li, Ning, Lee, Heewon, Brazzillo, Jason, Nummy, Laurence J, Chung, J C, Luvaga, Irungu K, Narayanan, Bikshandarkoil A, Wei, Xudong, Song, Jinhua J, Roschangar, Frank, Yee, Nathan K, Senanayake, Chris H
Published in Green chemistry : an international journal and green chemistry resource : GC (2017)
Published in Green chemistry : an international journal and green chemistry resource : GC (2017)
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Efficient Iron-Catalyzed Kumada Cross-Coupling Reactions Utilizing Flow Technology under Low Catalyst Loadings
Buono, Frederic G., Zhang, Yongda, Tan, Zhulin, Brusoe, Andrew, Yang, Bing-Shiou, Lorenz, Jon C., Giovannini, Riccardo, Song, Jinhua J., Yee, Nathan K., Senanayake, Chris H.
Published in European Journal of Organic Chemistry (01.05.2016)
Published in European Journal of Organic Chemistry (01.05.2016)
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Synthesis of the 6‑Azaindole Containing HIV‑1 Attachment Inhibitor Pro-Drug, BMS-663068
Chen, Ke, Risatti, Christina, Bultman, Michael, Soumeillant, Maxime, Simpson, James, Zheng, Bin, Fanfair, Dayne, Mahoney, Michelle, Mudryk, Boguslaw, Fox, Richard J, Hsaio, Yi, Murugesan, Saravanababu, Conlon, David A, Buono, Frederic G, Eastgate, Martin D
Published in Journal of organic chemistry (19.09.2014)
Published in Journal of organic chemistry (19.09.2014)
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Amine-Tunable Ruthenium Catalysts for Asymmetric Reduction of Ketones
Rodríguez, Sonia, Qu, Bo, Fandrick, Keith R., Buono, Frederic, Haddad, Nizar, Xu, Yibo, Herbage, Melissa A., Zeng, Xingzhong, Ma, Shengli, Grinberg, Nelu, Lee, Heewon, Han, Zhengxu S., Yee, Nathan K., Senanayake, Chris H.
Published in Advanced synthesis & catalysis (10.02.2014)
Published in Advanced synthesis & catalysis (10.02.2014)
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In silico enzyme screening identifies an SDR ketoreductase from Thermus caliditerrae as an attractive biocatalyst and promising candidate for protein engineering
Sosa, Yvett, Kapur, Bhav, Hurtak, Jessica, Kingsley, Laura J., Wu, Hao, Gruber, Stefanie, Nar, Herbert, Khattabi, Saad, Moral, Jesus Seco, Lucas, Maria Fátima, Martin, Caterina, Lončar, Nikola, Buono, Frederic, Pefaur, Noah, Nixon, Andrew E., Song, Jinhua J.
Published in Frontiers in Chemical Biology (23.07.2024)
Published in Frontiers in Chemical Biology (23.07.2024)
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Feed-Forward Neural Network for Predicting Enantioselectivity of the Asymmetric Negishi Reaction
Cuomo, Abbigayle E., Ibarraran, Sebastian, Sreekumar, Sanil, Li, Haote, Eun, Jungmin, Menzel, Jan Paul, Zhang, Pengpeng, Buono, Frederic, Song, Jinhua J., Crabtree, Robert H., Batista, Victor S., Newhouse, Timothy R.
Published in ACS central science (27.09.2023)
Published in ACS central science (27.09.2023)
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Development of an Asymmetric Synthesis of a Chiral Quaternary FLAP Inhibitor
Fandrick, Keith R, Mulder, Jason A, Patel, Nitinchandra D, Gao, Joe, Konrad, Michael, Archer, Elizabeth, Buono, Frederic G, Duran, Adil, Schmid, Rolf, Daeubler, Juergen, Desrosiers, Jean-Nicolas, Zeng, Xingzhong, Rodriguez, Sonia, Ma, Shengli, Qu, Bo, Li, Zhibin, Fandrick, Daniel R, Grinberg, Nelu, Lee, Heewon, Bosanac, Todd, Takahashi, Hidenori, Chen, Zhidong, Bartolozzi, Alessandra, Nemoto, Peter, Busacca, Carl A, Song, Jinhua J, Yee, Nathan K, Mahaney, Paige E, Senanayake, Chris H
Published in Journal of organic chemistry (06.02.2015)
Published in Journal of organic chemistry (06.02.2015)
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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 4. Synthesis of the 6‑Azaindole Core
Bultman, Michael S, Fan, Junying, Fanfair, Dayne, Soltani, Michelle, Simpson, James, Murugesan, Saravanababu, Soumeillant, Maxime, Chen, Ke, Risatti, Christina, La Cruz, Thomas E, Buono, Frederic G, Hung, Victor, Schild, Richard L, Ivy, Sabrina, Sweeney, Jason T, Conlon, David A, Eastgate, Martin D
Published in Organic process research & development (18.08.2017)
Published in Organic process research & development (18.08.2017)
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Addressing the Configuration Stability of Lithiated Secondary Benzylic Carbamates for the Development of a Noncryogenic Stereospecific Boronate Rearrangement
Fandrick, Keith R, Patel, Nitinchandra D, Mulder, Jason A, Gao, Joe, Konrad, Michael, Archer, Elizabeth, Buono, Frederic G, Duran, Adil, Schmid, Rolf, Daeubler, Juergen, Fandrick, Daniel R, Ma, Shengli, Grinberg, Nelu, Lee, Heewon, Busacca, Carl A, Song, Jinhua J, Yee, Nathan K, Senanayake, Chris H
Published in Organic letters (05.09.2014)
Published in Organic letters (05.09.2014)
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A Practical Stereoselective Synthesis and Novel Cocrystallizations of an Amphiphatic SGLT-2 Inhibitor
Deshpande, Prashant P, Singh, Janak, Pullockaran, Annie, Kissick, Thomas, Ellsworth, Bruce A, Gougoutas, Jack Z, Dimarco, John, Fakes, Michael, Reyes, Mayra, Lai, Chiajen, Lobinger, Hidegard, Denzel, Theo, Ermann, Peter, Crispino, Gerard, Randazzo, Michael, Gao, Zenrong, Randazzo, Renee, Lindrud, Mark, Rosso, Victor, Buono, Frederic, Doubleday, Wendel W, Leung, Simon, Richberg, Pricilla, Hughes, David, Washburn, William N, Meng, Wei, Volk, Kevin J, Mueller, Richard H
Published in Organic process research & development (20.04.2012)
Published in Organic process research & development (20.04.2012)
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