Evaluation of Cytochrome P450 3A4-Mediated Drug–Drug Interaction Potential for Cobimetinib Using Physiologically Based Pharmacokinetic Modeling and Simulation
Budha, Nageshwar R., Ji, Tao, Musib, Luna, Eppler, Steve, Dresser, Mark, Chen, Yuan, Jin, Jin Y.
Published in Clinical pharmacokinetics (01.11.2016)
Published in Clinical pharmacokinetics (01.11.2016)
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Journal Article
Prevalence of Acid-Reducing Agents (ARA) in Cancer Populations and ARA Drug–Drug Interaction Potential for Molecular Targeted Agents in Clinical Development
Smelick, Gillian S, Heffron, Timothy P, Chu, Laura, Dean, Brian, West, David A, DuVall, Scott L, Lum, Bert L, Budha, Nageshwar, Holden, Scott N, Benet, Leslie Z, Frymoyer, Adam, Dresser, Mark J, Ware, Joseph A
Published in Molecular pharmaceutics (04.11.2013)
Published in Molecular pharmaceutics (04.11.2013)
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Journal Article
Single- and multiple-dose pharmacokinetics, potential for CYP3A inhibition, and food effect in patients with cancer and healthy subjects receiving ipatasertib
Malhi, Vikram, Budha, Nageshwar, Sane, Rucha, Huang, Jian, Liederer, Bianca, Meng, Raymond, Patel, Premal, Deng, Yuzhong, Cervantes, Andres, Tabernero, Josep, Musib, Luna
Published in Cancer chemotherapy and pharmacology (01.12.2021)
Published in Cancer chemotherapy and pharmacology (01.12.2021)
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Journal Article
A tandem mass spectrometry assay for the simultaneous determination of acetaminophen, caffeine, phenytoin, ranitidine, and theophylline in small volume pediatric plasma specimens
Zhang, Yi, Mehrotra, Nitin, Budha, Nageshwar R., Christensen, Michael L., Meibohm, Bernd
Published in Clinica chimica acta (01.12.2008)
Published in Clinica chimica acta (01.12.2008)
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Journal Article
AdvanTIG-105: a phase I dose escalation study of the anti-TIGIT monoclonal antibody ociperlimab in combination with tislelizumab in patients with advanced solid tumors
Frentzas, Sophia, Kao, Steven, Gao, Rang, Zheng, Hao, Rizwan, Ahsan, Budha, Nageshwar, de la Hoz Pedroza, Luz, Tan, Wei, Meniawy, Tarek
Published in Journal for immunotherapy of cancer (01.10.2023)
Published in Journal for immunotherapy of cancer (01.10.2023)
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Journal Article
Clinical dose rationale of tislelizumab in patients with solid or hematological advanced tumors
Yu, Tian, Liu, Xiangyu, Wu, Chi‐Yuan, Tang, Zhiyu, Wang, Hongwei, Schnell, Patrick, Wan, Ya, Wang, Kun, Liu, Lucy, Gao, Yuying, Sahasranaman, Srikumar, Budha, Nageshwar
Published in Clinical and translational science (01.03.2024)
Published in Clinical and translational science (01.03.2024)
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Journal Article
Model‐based population pharmacokinetic analysis of tislelizumab in patients with advanced tumors
Budha, Nageshwar, Wu, Chi‐Yuan, Tang, Zhiyu, Yu, Tian, Liu, Lucy, Xu, Fengyan, Gao, Yuying, Li, Ruiying, Zhang, Qiuyang, Wan, Ya, Sahasranaman, Srikumar
Published in CPT: pharmacometrics and systems pharmacology (01.01.2023)
Published in CPT: pharmacometrics and systems pharmacology (01.01.2023)
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Journal Article
Biopharmaceutics, Pharmacokinetics and Pharmacodynamics of Antituberculosis Drugs
BUDHA, Nageshwar R, LEE, Richard E, MEIBOHM, Bernd
Published in Current medicinal chemistry (01.04.2008)
Published in Current medicinal chemistry (01.04.2008)
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Journal Article
Population pharmacokinetics and dosing implications for cobimetinib in patients with solid tumors
Han, Kelong, Jin, Jin Y., Marchand, Mathilde, Eppler, Stephen, Choong, Nicholas, Hack, Stephen P., Tikoo, Nalin, Bruno, Rene, Dresser, Mark, Musib, Luna, Budha, Nageshwar R.
Published in Cancer chemotherapy and pharmacology (01.11.2015)
Published in Cancer chemotherapy and pharmacology (01.11.2015)
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Journal Article
A phase 1 study to evaluate the safety and LDL cholesterol–lowering effects of RG7652, a fully human monoclonal antibody against proprotein convertase subtilisin/kexin type 9
Baruch, Amos, Luca, Diana, Kahn, Robert S., Cowan, Kyra J., Leabman, Maya, Budha, Nageshwar R., Chiu, Cecilia P.C., Wu, Yan, Kirchhofer, Daniel, Peterson, Andrew, Davis Jr, John C., Tingley, Whittemore G.
Published in Clinical cardiology (Mahwah, N.J.) (01.07.2017)
Published in Clinical cardiology (Mahwah, N.J.) (01.07.2017)
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Journal Article
Modeling and Simulation to Support Phase 2 Dose Selection for RG7652, a Fully Human Monoclonal Antibody Against Proprotein Convertase Subtilisin/Kexin Type 9
Budha, Nageshwar R., Leabman, Maya, Jin, Jin Y., Wada, D. Russell, Baruch, Amos, Peng, Kun, Tingley, Whittemore G., Davis, John D.
Published in The AAPS journal (01.07.2015)
Published in The AAPS journal (01.07.2015)
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Journal Article
Population repeated time‐to‐event analysis of exacerbations in asthma patients: A novel approach for predicting asthma exacerbations based on biomarkers, spirometry, and diaries/questionnaires
Svensson, Robin J, Ribbing, Jakob, Kotani, Naoki, Dolton, Michael, Vadhavkar, Shweta, Cheung, Dorothy, Staton, Tracy, Choy, David F, Putnam, Wendy, Jin, Jin, Budha, Nageshwar, Karlsson, Mats O., Quartino, Angelica, Zhu, Rui
Published in CPT: pharmacometrics and systems pharmacology (01.10.2021)
Published in CPT: pharmacometrics and systems pharmacology (01.10.2021)
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Journal Article
A microbiological assessment of novel nitrofuranylamides as anti-tuberculosis agents
Hurdle, Julian G., Lee, Robin B., Budha, Nageshwar R., Carson, Elizabeth I., Qi, Jianjun, Scherman, Michael S., Cho, Sang Hyun, McNeil, Michael R., Lenaerts, Anne J., Franzblau, Scott G., Meibohm, Bernd, Lee, Richard E.
Published in Journal of antimicrobial chemotherapy (01.11.2008)
Published in Journal of antimicrobial chemotherapy (01.11.2008)
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Journal Article
Gastric Reacidification with Betaine HCl in Healthy Volunteers with Rabeprazole-Induced Hypochlorhydria
Yago, Marc R, Frymoyer, Adam R, Smelick, Gillian S, Frassetto, Lynda A, Budha, Nageshwar R, Dresser, Mark J, Ware, Joseph A, Benet, Leslie Z
Published in Molecular pharmaceutics (04.11.2013)
Published in Molecular pharmaceutics (04.11.2013)
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Journal Article
Dogs are more sensitive to antagonists of inhibitor of apoptosis proteins than rats and humans: a translational toxicokinetic/toxicodynamic analysis
Wong, Harvey, Budha, Nageshwar R, West, Kristina, Blackwood, Elizabeth, Ware, Joseph A, Yu, Ron, Darbonne, Walter C, Gould, Stephen E, Steigerwalt, Ronald, Erickson, Rebecca, Hop, Cornelis E A C, LoRusso, Patricia, Eckhardt, S Gail, Wagner, Andrew, Chan, Iris T, Mamounas, Michael, Flygare, John A, Fairbrother, Wayne J
Published in Toxicological sciences (01.11.2012)
Published in Toxicological sciences (01.11.2012)
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Journal Article
Critical role of bioanalytical strategies in investigation of clinical PK observations, a Phase I case study
Peng, Kun, Xu, Keyang, Liu, Luna, Hendricks, Robert, Delarosa, Reginald, Erickson, Rich, Budha, Nageshwar, Leabman, Maya, Song, An, Kaur, Surinder, Fischer, Saloumeh K
Published in mAbs (02.11.2014)
Published in mAbs (02.11.2014)
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Journal Article