Development of a P-Glycoprotein Knockout Model in Rodents to Define Species Differences in its Functional Effect at the Blood–brain Barrier
Cutler, Leanne, Howes, Colin, Deeks, Nigel J., Buck, Tania L., Jeffrey, Phil
Published in Journal of pharmaceutical sciences (01.09.2006)
Published in Journal of pharmaceutical sciences (01.09.2006)
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Oral administration of a potent and selective non-peptidic BACE-1 inhibitor decreases β-cleavage of amyloid precursor protein and amyloid-β production in vivo
Hussain, Ishrut, Hawkins, Julie, Harrison, David, Hille, Christopher, Wayne, Gareth, Cutler, Leanne, Buck, Tania, Walter, Daryl, Demont, Emmanuel, Howes, Colin, Naylor, Alan, Jeffrey, Philip, Gonzalez, Maria I, Dingwall, Colin, Michel, Anton, Redshaw, Sally, Davis, John B
Published in Journal of neurochemistry (01.02.2007)
Published in Journal of neurochemistry (01.02.2007)
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Bicyclic heteroarylpiperazines as selective brain penetrant 5-HT 6 receptor antagonists
Ahmed, Mahmood, Briggs, Michael A., Bromidge, Steven M., Buck, Tania, Campbell, Lorraine, Deeks, Nigel J., Garner, Ashley, Gordon, Laurie, Hamprecht, Dieter W., Holland, Vicky, Johnson, Christopher N., Medhurst, Andrew D., Mitchell, Darren J., Moss, Stephen F., Powles, Jenifer, Seal, Jon T., Stean, Tania O., Stemp, Geoffrey, Thompson, Mervyn, Trail, Brenda, Upton, Neil, Winborn, Kim, Witty, David R.
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
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Bicyclic heteroarylpiperazines as selective brain penetrant 5-HT6 receptor antagonists
AHMED, Mahmood, BRIGGS, Michael A, JOHNSON, Christopher N, MEDHURST, Andrew D, MITCHELL, Darren J, MOSS, Stephen F, POWLES, Jenifer, SEAL, Jon T, STEAN, Tania O, STEMP, Geoffrey, THOMPSON, Mervyn, TRAIL, Brenda, BROMIDGE, Steven M, UPTON, Neil, WINBORN, Kim, WITTY, David R, BUCK, Tania, CAMPBELL, Lorraine, DEEKS, Nigel J, GARNER, Ashley, GORDON, Laurie, HAMPRECHT, Dieter W, HOLLAND, Vicky
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
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Journal Article
Oral administration of a potent and selective non-peptidic BACE-1 inhibitor decreases [beta]-cleavage of amyloid precursor protein and amyloid-[beta] production in vivo
Hussain, Ishrut, Hawkins, Julie, Harrison, David, Hille, Christopher, Wayne, Gareth, Cutler, Leanne, Buck, Tania, Walter, Daryl, Demont, Emmanuel, Howes, Colin, Naylor, Alan, Philip, Jeffrey, Gonzalez, Maria I, Dingwall, Colin, Anton, Michel, Redshaw, Sally
Published in Journal of neurochemistry (01.02.2007)
Published in Journal of neurochemistry (01.02.2007)
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Journal Article
WITHDRAWN: Bicyclic heteroarylpiperazines as selective brain penetrant 5-HT6 receptor antagonists
Ahmed, Mahmood, Briggs, Michael A., Bromidge, Steven M., Buck, Tania, Campbell, Lorraine, Deeks, Nigel J., Garner, Ashley, Gordon, Laurie, Hamprecht, Dieter W., Holland, Vicky, Johnson, Christopher N., Medhurst, Andrew D., Mitchell, Darren J., Moss, Stephen F., Powles, Jenifer, Seal, Jon T., Stean, Tania O., Stemp, Geoffrey, Thompson, Mervyn, Trail, Brenda, Upton, Neil, Winborn, Kim, Witty, David R.
Published in Bioorganic & medicinal chemistry (01.07.2005)
Published in Bioorganic & medicinal chemistry (01.07.2005)
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