Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876
Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Müller, Thomas, Bauser, Marcus, Buchmann, Bernd
Published in ChemMedChem (19.10.2016)
Published in ChemMedChem (19.10.2016)
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Total Synthesis and Antitumor Activity of ZK-EPO: The First Fully Synthetic Epothilone in Clinical Development
Klar, Ulrich, Buchmann, Bernd, Schwede, Wolfgang, Skuballa, Werner, Hoffmann, Jens, Lichtner, Rosemarie B.
Published in Angewandte Chemie International Edition (04.12.2006)
Published in Angewandte Chemie International Edition (04.12.2006)
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Discovery of BAY-405: An Azaindole-Based MAP4K1 Inhibitor for the Enhancement of T‑Cell Immunity against Cancer
Mowat, Jeffrey, Carretero, Rafael, Leder, Gabriele, Aiguabella Font, Nuria, Neuhaus, Roland, Berndt, Sandra, Günther, Judith, Friberg, Anders, Schäfer, Martina, Briem, Hans, Raschke, Marian, Miyatake Ondozabal, Hideki, Buchmann, Bernd, Boemer, Ulf, Kreft, Bertolt, Hartung, Ingo V., Offringa, Rienk
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Published in Journal of medicinal chemistry (10.10.2024)
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Identification of novel GLUT inhibitors
Siebeneicher, Holger, Bauser, Marcus, Buchmann, Bernd, Heisler, Iring, Müller, Thomas, Neuhaus, Roland, Rehwinkel, Hartmut, Telser, Joachim, Zorn, Ludwig
Published in Bioorganic & medicinal chemistry letters (01.04.2016)
Published in Bioorganic & medicinal chemistry letters (01.04.2016)
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Abstract 4333: Identification and optimization of the first highly selective GLUT-1 inhibitors
Bauser, Marcus, Buchmann, Bernd, Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Mueller, Thomas, Kopitz, Charlotte Christine
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Abstract 1164: Metabolic responses in cancer cells with differential susceptibility to GLUT1 inhibition
Gruenewald, Sylvia, Rennefahrt, Ulrike, Maldonado, Sandra G., Walter, Alexander, Petrul, Heike, Héroult, Mélanie, Heisler, Iring, Quanz, Maria, Steigemann, Patrick, Buchmann, Bernd, Haegebarth, Andrea
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Cover Picture: Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876 (ChemMedChem 20/2016)
Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Müller, Thomas, Bauser, Marcus, Buchmann, Bernd
Published in ChemMedChem (19.10.2016)
Published in ChemMedChem (19.10.2016)
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Abstract 4746: Pharmacological characterization of BAY-876, a novel highly selective inhibitor of glucose transporter (GLUT)-1 in vitro and in vivo
Kopitz, Charlotte, Toschi, Luisella, Algire, Carolyn, Héroult, Mélanie, Frisk, Anna-Lena, Meyer, Kirstin, Schmitz, Arndt, Lagkadinou, Eleni, Petrul, Heike, Heisler, Iring, Neuhaus, Roland, Buchmann, Bernd, Himmel, Herbert, Bauser, Marcus, Haegebarth, Andrea, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Improved Cellular Pharmacokinetics and Pharmacodynamics Underlie the Wide Anticancer Activity of Sagopilone
HOFFMANN, Jens, VILALE, Ilio, PANARETAKIS, Theocharis, SIEMEISTER, Gerhard, LAGE, Hermann, NANTY, Lisa, HAMMER, Stefanie, MITTELSTAEDT, Kevin, WINSEL, Sebastian, ESCHENBRENNER, Julia, CASTEDO, Maria, DEMARCHE, Carine, BUCHMANN, Bernd, KLAR, Ulrich, KROEMER, Guido, GALLUZZI, Lorenzo, SCHWEDE, Wolfgang, SENOVILLA, Laura, SKUBALLA, Werner, VIVET, Sonia, LICHTNER, Rosemarie B, VICENCIO, José M
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[1,2,4]트리아졸로[1,5-c]퀴나졸린-5-아민
BADER BENJAMIN, GUENTHER JUDITH, ZORN LUDWIG, MEIER ROBIN MICHAEL, GUTCHER ILONA, BAUMANN DANIEL, BUCHMANN BERND, SCHMEES NORBERT, GORJANACZ MATYAS, HERBERT SIMON ANTHONY, STOECKIGT DETLEF, PLATTEN MICHAEL, LEFRANC JULIEN, KOBER CHRISTINA, BOTHE ULRICH, BOEHME STEPHAN, ROESE LARS
Year of Publication 13.04.2022
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Abstract 1026: Novel Tie2 inhibitor with in vivo efficacy in disseminated hematological tumor models in mice
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Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Abstract 1442: Effects of selective and broad glucose transporter (GLUT) inhibition on glucose distribution in tumor bearing mice
Heroult, Melanie, Steinke, Wolfram, Frisk, Anna-Lena, Borkowski, Sandra, Meyer, Kirstin, Petrul, Heike, Heisler, Iring, Quanz, Maria, Neuhaus, Roland, Buchmann, Bernd, Mueller, Thomas, Bauser, Marcus, Haegebarth, Andrea, Brands, Michael, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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The Role of Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 in the p38/TNF-α Pathway of Systemic and Cutaneous Inflammation
Schottelius, Arndt J., Zügel, Ulrich, Döcke, Wolf-Dietrich, Zollner, Thomas M., Röse, Lars, Mengel, Anne, Buchmann, Bernd, Becker, Andreas, Grütz, Gerald, Naundorf, Sandra, Friedrich, Anke, Gaestel, Matthias, Asadullah, Khusru
Published in Journal of investigative dermatology (01.02.2010)
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PHARMACEUTICAL COMPOSITION AND THE USE THEREOF, AND APPLICATION REGIME OF SAID PHARMACEUTICAL COMPOSITION FOR ON-DEMAND CONTRACEPTION
SERNO PETER, ROTGERI ANDREA, BUCHMANN BERND, ROEHN ULRIKE, TER LAAK ANTONIUS, LINDENTHAL BERNHARD, FUHRMANN ULRIKE, BRAEUER NICO, MENGEL ANNE
Year of Publication 11.02.2016
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ROTGERI ANDREA, BUCHMANN BERND, ROEHN ULRIKE, TER LAAK ANTONIUS, LINDENTHAL BERNHARD, BRAEUER NICO, MENGEL ANNE
Year of Publication 27.08.2014
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Year of Publication 27.08.2014
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The Role of Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 in the p38/TNF-[alpha] Pathway of Systemic and Cutaneous Inflammation
Schottelius, Arndt J, Zügel, Ulrich, Döcke, Wolf-dietrich, Zollner, Thomas M, Röse, Lars, Mengel, Anne, Buchmann, Bernd, Becker, Andreas, Grütz, Gerald, Naundorf, Sandra, Friedrich, Anke, Gaestel, Matthias, Asadullah, Khusru
Published in Journal of investigative dermatology (01.02.2010)
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Cover Picture: Total Synthesis and Antitumor Activity of ZK-EPO: The First Fully Synthetic Epothilone in Clinical Development (Angew. Chem. Int. Ed. 47/2006)
Klar, Ulrich, Buchmann, Bernd, Schwede, Wolfgang, Skuballa, Werner, Hoffmann, Jens, Lichtner, Rosemarie B.
Published in Angewandte Chemie International Edition (04.12.2006)
Published in Angewandte Chemie International Edition (04.12.2006)
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Synthesis of 3H-labeled Efomycine M
Bader, Ben, von Bonin, Arne, Buchmann, Bernd, Gay, Juergen, Gruendemann, Stephan, Guenther, Judith, Schaefer, Martina, Spellig, Tilman, Zollner, Thomas M., Zorn, Ludwig
Published in Tetrahedron letters (20.08.2007)
Published in Tetrahedron letters (20.08.2007)
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JOERISSEN HANNAH, SUESSMEIER FRANK, TELSER JOACHIM, LOBELL MARIO, HEROULT MELANIE, GRUENEWALD SYLVIA, BUCHMANN BERND, LUSTIG KLEMENS, LINDNER NIELS, HAERTER MICHAEL, KAHNERT ANTJE
Year of Publication 07.10.2014
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Year of Publication 07.10.2014
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Efficient chiral pool synthesis of the C1-C6 fragment of epothilones
Klar, U, Rohr, B, Kuczynski, F, Schwede, W, Berger, M, Skuballa, W, Buchmann, B
Published in Synthesis (Stuttgart) (01.02.2005)
Published in Synthesis (Stuttgart) (01.02.2005)
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