Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (BAY-598) for the Protein Lysine Methyltransferase SMYD2
Eggert, Erik, Hillig, Roman C, Koehr, Silke, Stöckigt, Detlef, Weiske, Jörg, Barak, Naomi, Mowat, Jeffrey, Brumby, Thomas, Christ, Clara D, ter Laak, Antonius, Lang, Tina, Fernandez-Montalvan, Amaury E, Badock, Volker, Weinmann, Hilmar, Hartung, Ingo V, Barsyte-Lovejoy, Dalia, Szewczyk, Magdalena, Kennedy, Steven, Li, Fengling, Vedadi, Masoud, Brown, Peter J, Santhakumar, Vijayaratnam, Arrowsmith, Cheryl H, Stellfeld, Timo, Stresemann, Carlo
Published in Journal of medicinal chemistry (26.05.2016)
Published in Journal of medicinal chemistry (26.05.2016)
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Neutral W(V) Complexes Featuring the W2O2(µ-O)2 Core and Amino Acids or EDTA Derivatives as Ligands: Synthesis and Structural Characterization
Varbanov, Hristo P., Belaj, Ferdinand, Glasnov, Toma, Herbert, Simon, Brumby, Thomas, Mösch-Zanetti, Nadia C.
Published in Inorganics (01.03.2023)
Published in Inorganics (01.03.2023)
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The Lab Oddity Prevails: Discovery of Pan-CDK Inhibitor (R)-S-Cyclopropyl-S-(4-{[4-{[(1R,2R)-2-hydroxy-1-methylpropyl]oxy}-5-(trifluoromethyl)pyrimidin-2-yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer
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Published in ChemMedChem (01.07.2013)
Published in ChemMedChem (01.07.2013)
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New strategies towards advanced CT contrast agents. Development of neutral and monoanionic sulfur-bridged W() dimeric complexes
Varbanov, Hristo P, Glasnov, Toma, Belaj, Ferdinand, Herbert, Simon, Brumby, Thomas, Mösch-Zanetti, Nadia C
Published in Dalton transactions : an international journal of inorganic chemistry (26.07.2022)
Published in Dalton transactions : an international journal of inorganic chemistry (26.07.2022)
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표적화 방사선요법에 사용하기 위한 다량체 킬레이트화제화합물
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Year of Publication 10.10.2023
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Year of Publication 10.10.2023
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PANKNIN OLAF, JOST GREGOR, LOHRKE JESSICA, FRENZEL THOMAS, BERGER MARKUS, BRUMBY THOMAS, HERBERT SIMON ANTHONY, WITTROCK SVEN, GREEN CLAUDIA, PIETSCH HUBERTUS
Year of Publication 16.11.2023
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Year of Publication 16.11.2023
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조영 매체의 제형 및 그의 제조 방법
JOST GREGOR, FRENZEL THOMAS, LOHRKE JESSICA, BRUMBY THOMAS, HOLZSCHUH STEPHAN, EBERT WOLFGANG, HALFBRODT WOLFGANG
Year of Publication 30.07.2021
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Year of Publication 30.07.2021
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Efficient Routes to a Diverse Array of Amino Alcohol-Derived Chiral Fragments
Haftchenary, Sina, Nelson, Shawn D, Furst, Laura, Dandapani, Sivaraman, Ferrara, Steven J, Bošković, Žarko V, Figueroa Lazú, Samuel, Guerrero, Adrian M, Serrano, Juan C, Crews, DeMarcus K, Brackeen, Cristina, Mowat, Jeffrey, Brumby, Thomas, Bauser, Marcus, Schreiber, Stuart L, Phillips, Andrew J
Published in ACS combinatorial science (12.09.2016)
Published in ACS combinatorial science (12.09.2016)
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From the Insoluble Dye Indirubin towards Highly Active, Soluble CDK2-Inhibitors
Jautelat, Rolf, Brumby, Thomas, Schäfer, Martina, Briem, Hans, Eisenbrand, Gerhard, Schwahn, Stefan, Krüger, Martin, Lücking, Ulrich, Prien, Olaf, Siemeister, Gerhard
Published in Chembiochem : a European journal of chemical biology (01.03.2005)
Published in Chembiochem : a European journal of chemical biology (01.03.2005)
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치환된 디히드로피라졸로 피라진 카르복스아미드 유도체
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Year of Publication 03.02.2021
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Year of Publication 03.02.2021
Patent
Cover Picture: The Lab Oddity Prevails: Discovery of Pan-CDK Inhibitor (R)-S-Cyclopropyl-S-(4-{[4-{[(1R,2R)-2-hydroxy-1-methylpropyl]oxy}-5-(trifluoromethyl)pyrimidin-2-yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer (ChemMedChem 7/2013)
Lücking, Ulrich, Jautelat, Rolf, Krüger, Martin, Brumby, Thomas, Lienau, Philip, Schäfer, Martina, Briem, Hans, Schulze, Julia, Hillisch, Alexander, Reichel, Andreas, Wengner, Antje Margret, Siemeister, Gerhard
Published in ChemMedChem (01.07.2013)
Published in ChemMedChem (01.07.2013)
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Intra- and intermolecular hetero-Diels-Alder reactions. 17. Intramolecular hetero-Diels-Alder reaction of alkylidene- and benzylidenepyrazolones and benzylideneisoxazolones. Investigations toward the conformation of the transition state
Tietze, Lutz F., Brumby, Thomas, Pretor, Martina, Remberg, Gerd
Published in Journal of organic chemistry (01.02.1988)
Published in Journal of organic chemistry (01.02.1988)
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RADIOLABELED AMINO ACIDS FOR DIAGNOSTIC IMAGING
STELLFELD TIMO, KETTSCHAU GEORG, SCHMITT WILLICH HERIBERT, BRUMBY THOMAS, BERNDT MATHIAS, KRUEGER MARTIN, LEHMANN LUTZ, GRAHAM KEITH, MUELLER ANDRE, HASSFELD JORMA
Year of Publication 20.05.2014
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Year of Publication 20.05.2014
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METHOD FOR PRODUCTION OF F-18 LABELED GLUTAMIC ACID DERIVATIVES
FRIEBE MATTHIAS, WESTER HANS JUERGEN, SCHMITT WILLICH HERIBERT, BRUMBY THOMAS, BERNDT MATHIAS, HULTSCH CHRISTINA, GRAHAM KEITH, WAGNER FRANZISKA
Year of Publication 13.09.2012
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Year of Publication 13.09.2012
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FORMULATION OF CONTRAST MEDIA AND PROCESS OF PREPARATION THEREOF
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Year of Publication 01.08.2024
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Year of Publication 01.08.2024
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MULTIMERIC CHELATOR COMPOUNDS FOR USE IN TARGETED RADIOTHERAPY
KRISTIAN, Alexander, CRUCIANI, Véronique, KROGSTIE, Vilde Roko, RAFIQUE, Waqas, CUTHBERTSON, Alan, INDREVOLL, Bård, BRUMBY, Thomas
Year of Publication 30.05.2024
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Year of Publication 30.05.2024
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