3-(7-Azaindolyl)-4-arylmaleimides as potent, selective inhibitors of glycogen synthase kinase-3
Zhang, Han-Cheng, Ye, Hong, Conway, Bruce R., Derian, Claudia K., Addo, Michael F., Kuo, Gee-Hong, Hecker, Leonard R., Croll, Diane R., Li, Jian, Westover, Lori, Xu, Jun Z., Look, Richard, Demarest, Keith T., Andrade-Gordon, Patricia, Damiano, Bruce P., Maryanoff, Bruce E.
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Synthesis and evaluation of 3-anilino-quinoxalinones as glycogen phosphorylase inhibitors
Dudash, Joseph, Zhang, Yongzheng, Moore, John B., Look, Richard, Liang, Yin, Beavers, Mary Pat, Conway, Bruce R., Rybczynski, Philip J., Demarest, Keith T.
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
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Synthesis and Discovery of Macrocyclic Polyoxygenated Bis-7-azaindolylmaleimides as a Novel Series of Potent and Highly Selective Glycogen Synthase Kinase-3β Inhibitors
Kuo, Gee-Hong, Prouty, Catherine, DeAngelis, Alan, Shen, Lan, O'Neill, David J, Shah, Chandra, Connolly, Peter J, Murray, William V, Conway, Bruce R, Cheung, Peter, Westover, Lori, Xu, Jun Z, Look, Richard A, Demarest, Keith T, Emanuel, Stuart, Middleton, Steven A, Jolliffe, Linda, Beavers, Mary Pat, Chen, Xin
Published in Journal of medicinal chemistry (11.09.2003)
Published in Journal of medicinal chemistry (11.09.2003)
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Novel Indolylindazolylmaleimides as Inhibitors of Protein Kinase C-β: Synthesis, Biological Activity, and Cardiovascular Safety
Zhang, Han-Cheng, Derian, Claudia K, McComsey, David F, White, Kimberly B, Ye, Hong, Hecker, Leonard R, Li, Jian, Addo, Michael F, Croll, Diane, Eckardt, Annette J, Smith, Charles E, Li, Quan, Cheung, Wai-Man, Conway, Bruce R, Emanuel, Stuart, Demarest, Keith T, Andrade-Gordon, Patricia, Damiano, Bruce P, Maryanoff, Bruce E
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Heteroaryl- O-glucosides as novel sodium glucose co-transporter 2 inhibitors. Part 1
Zhang, Xiaoyan, Urbanski, Maud, Patel, Mona, Zeck, Roxanne E., Cox, Geoffrey G., Bian, Haiyan, Conway, Bruce R., Pat Beavers, Mary, Rybczynski, Philip J., Demarest, Keith T.
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
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Indole-glucosides as novel sodium glucose co-transporter 2 (SGLT2) inhibitors. Part 2
Zhang, Xiaoyan, Urbanski, Maud, Patel, Mona, Cox, Geoffrey G., Zeck, Roxanne E., Bian, Haiyan, Conway, Bruce R., Beavers, Mary Pat, Rybczynski, Philip J., Demarest, Keith T.
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
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Macrocyclic bisindolylmaleimides as inhibitors of protein kinase C and glycogen synthase kinase-3
Zhang, Han-Cheng, White, Kimberly B., Ye, Hong, McComsey, David F., Derian, Claudia K., Addo, Michael F., Andrade-Gordon, Patricia, Eckardt, Annette J., Conway, Bruce R., Westover, Lori, Xu, Jun Z., Look, Richard, Demarest, Keith T., Emanuel, Stuart, Maryanoff, Bruce E.
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
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Glycosylated dihydrochalcones as potent and selective sodium glucose co-transporter 2 (SGLT2) inhibitors
Dudash, Joseph, Zhang, Xiaoyan, Zeck, Roxanne E., Johnson, Sigmond G., Cox, Geoffrey G., Conway, Bruce R., Rybczynski, Philip J., Demarest, Keith T.
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
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Synthesis and biological evaluation of novel macrocyclic bis-7-azaindolylmaleimides as potent and highly selective glycogen synthase kinase-3β (GSK-3β) inhibitors
SHEN, Lan, PROUTY, Catherine, DEMAREST, Keith T, KUO, Gee-Hong, CONWAY, Bruce R, WESTOVER, Lori, XU, Jun Z, LOOK, Richard A, XIN CHEN, BEAVERS, Mary Pat, ROBERTS, Jerry, MURRAY, William V
Published in Bioorganic & medicinal chemistry (01.03.2004)
Published in Bioorganic & medicinal chemistry (01.03.2004)
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Quantification of G-Protein Coupled Receptor Internalization Using G-Protein Coupled Receptor-Green Fluorescent Protein Conjugates with the ArrayScan™ High-Content Screening System
Conway, Bruce R., Minor, Lisa K., Xu, Jun Z., Gunnet, Joseph W., DeBiasio, Robbin, D’Andrea, Michael R., Rubin, Richard, DeBiasio, Richard, Giuliano, Ken, Zhou, Lubing, Demaresti, Keith T.
Published in SLAS discovery (01.04.1999)
Published in SLAS discovery (01.04.1999)
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Functional Roles for the Pleckstrin and Dbl Homology Regions in the Ras Exchange Factor Son-of-sevenless (∗)
McCollam, Linda, Bonfini, Laura, Karlovich, Chris A., Conway, Bruce R., Kozma, Lynn M., Banerjee, Utpal, Czech, Michael P.
Published in The Journal of biological chemistry (07.07.1995)
Published in The Journal of biological chemistry (07.07.1995)
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Validation of a cell-based screen for insulin receptor modulators by quantification of insulin receptor phosphorylation
Minor, Lisa K, Westover, Lori, Kong, Yan, Patel, Darpana, Wildey, Mary Jo, Conway, Bruce R, Demarest, Keith T
Published in Journal of biomolecular screening (01.08.2003)
Published in Journal of biomolecular screening (01.08.2003)
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Interactions of Cbl with Grb2 and phosphatidylinositol 3'-kinase in activated Jurkat cells
Meisner, Herman, Conway, Bruce R., Hartley, David, Czech, Michael P.
Published in Molecular and Cellular Biology (01.07.1995)
Published in Molecular and Cellular Biology (01.07.1995)
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Design, synthesis, and biological evaluation of novel 7-azaindolyl-heteroaryl-maleimides as potent and selective glycogen synthase kinase-3β (GSK-3β) inhibitors
O'Neill, David J., Shen, Lan, Prouty, Catherine, Conway, Bruce R., Westover, Lori, Xu, Jun Z., Zhang, Han-Cheng, Maryanoff, Bruce E., Murray, William V., Demarest, Keith T., Kuo, Gee-Hong
Published in Bioorganic & medicinal chemistry (15.06.2004)
Published in Bioorganic & medicinal chemistry (15.06.2004)
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Quantitative analysis of agonist-dependent parathyroid hormone receptor trafficking in whole cells using a functional green fluorescent protein conjugate
Conway, Bruce R., Minor, Lisa K., Xu, Jun Z., D'Andrea, Michael R., Ghosh, Richik N., Demarest, Keith T.
Published in Journal of cellular physiology (01.12.2001)
Published in Journal of cellular physiology (01.12.2001)
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Novel indolylindazolylmaleimides as inhibitors of protein kinase C- : Synthesis, biological activity, and cardiovascular safety
ZHANG, Han-Cheng, DERIAN, Claudia K, SMITH, Charles E, QUAN LI, CHEUNG, Wai-Man, CONWAY, Bruce R, EMANUEL, Stuart, DEMAREST, Keith T, ANDRADE-GORDON, Patricia, DAMIANO, Bruce P, MARYANOFF, Bruce E, MCCOMSEY, David F, WHITE, Kimberly B, HONG YE, HECKER, Leonard R, JIAN LI, ADDO, Michael F, CROLL, Diane, ECKARDT, Annette J
Published in Journal of medicinal chemistry (2005)
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Published in Journal of medicinal chemistry (2005)
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Design, synthesis, and biological evaluation of novel 7-azaindolyl-heteroaryl-maleimides as potent and selective glycogen synthase kinase-3beta (GSK-3beta) inhibitors
O'Neill, David J, Shen, Lan, Prouty, Catherine, Conway, Bruce R, Westover, Lori, Xu, Jun Z, Zhang, Han-Cheng, Maryanoff, Bruce E, Murray, William V, Demarest, Keith T, Kuo, Gee-Hong
Published in Bioorganic & medicinal chemistry (15.06.2004)
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Published in Bioorganic & medicinal chemistry (15.06.2004)
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