Discovery of GSK2193874: An Orally Active, Potent, and Selective Blocker of Transient Receptor Potential Vanilloid 4
Cheung, Mui, Bao, Weike, Behm, David J, Brooks, Carl A, Bury, Michael J, Dowdell, Sarah E, Eidam, Hilary S, Fox, Ryan M, Goodman, Krista B, Holt, Dennis A, Lee, Dennis, Roethke, Theresa J, Willette, Robert N, Xu, Xiaoping, Ye, Guosen, Thorneloe, Kevin S
Published in ACS medicinal chemistry letters (11.05.2017)
Published in ACS medicinal chemistry letters (11.05.2017)
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Journal Article
Discovery of GSK3527497: A Candidate for the Inhibition of Transient Receptor Potential Vanilloid‑4 (TRPV4)
Brooks, Carl A, Barton, Linda S, Behm, David J, Brnardic, Edward J, Costell, Melissa H, Holt, Dennis A, Jolivette, Larry J, Matthews, Jay M, McAtee, John J, McCleland, Brent W, Patterson, Jaclyn R, Pero, Joseph E, Rivero, Ralph A, Roethke, Theresa J, Sanchez, Robert M, Shenje, Raynold, Terrell, Lamont R, Lawhorn, Brian G
Published in Journal of medicinal chemistry (24.10.2019)
Published in Journal of medicinal chemistry (24.10.2019)
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Journal Article
Discovery of GSK2798745: A Clinical Candidate for Inhibition of Transient Receptor Potential Vanilloid 4 (TRPV4)
Brooks, Carl A, Barton, Linda S, Behm, David J, Eidam, Hilary S, Fox, Ryan M, Hammond, Marlys, Hoang, Tram H, Holt, Dennis A, Hilfiker, Mark A, Lawhorn, Brian G, Patterson, Jaclyn R, Stoy, Patrick, Roethke, Theresa J, Ye, Guosen, Zhao, Steve, Thorneloe, Kevin S, Goodman, Krista B, Cheung, Mui
Published in ACS medicinal chemistry letters (08.08.2019)
Published in ACS medicinal chemistry letters (08.08.2019)
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Journal Article
TRPV4 길항제
LI PENG, MATTHEWS JAY M, LAWHORN BRIAN GRIFFIN, BRNARDIC EDWARD J, TERRELL LAMONT ROSCOE, SENDER MATTHEW ROBERT, PERO JOSEPH E, MCATEE JOHN JEFFREY, BEHM DAVID J, BROOKS CARL A
Year of Publication 09.05.2019
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Year of Publication 09.05.2019
Patent
TRPV4 길항제
MATTHEWS JAY M, LAWHORN BRIAN GRIFFIN, SANCHEZ ROBERT, YE GUOSEN, TERRELL LAMONT ROSCOE, PATTERSON JACLYN R, PERO JOSEPH E, SENDER MATTHEW ROBERT, MCATEE JOHN JEFFREY, BARTON LINDA S, THOMAS JAMES V, BRNARDIC EDWARD J, BUDZIK BRIAN W, BEHM DAVID J, BROOKS CARL A
Year of Publication 08.05.2019
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Year of Publication 08.05.2019
Patent